Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design
Dietrich, Justin D, Longenecker, Kenton L, Wilson, Noel S, Goess, Christian, Panchal, Sanjay C, Swann, Steven L, Petros, Andrew M, Hobson, Adrian D, Ihle, David, Song, Danying, Richardson, Paul, Comess, Kenneth M, Cox, Philip B, Dombrowski, Amanda, Sarris, Kathy, Donnelly-Roberts, Diana L, Duignan, David B, Gomtsyan, Arthur, Jung, Paul, Krueger, A Chris, Mathieu, Suzanne, McClure, Andrea, Stoll, Vincent S, Wetter, Jill, Mankovich, John A, Hajduk, Philip J, Vasudevan, Anil, Stoffel, Robert H, Sun, Chaohong
Published in Journal of medicinal chemistry (14.01.2021)
Published in Journal of medicinal chemistry (14.01.2021)
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Journal Article
Merits and Pitfalls in the Characterization of Covalent Inhibitors of Bruton’s Tyrosine Kinase
Harris, Christopher M., Foley, Sage E., Goedken, Eric R., Michalak, Mark, Murdock, Sara, Wilson, Noel S.
Published in SLAS discovery (01.12.2018)
Published in SLAS discovery (01.12.2018)
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Journal Article
A scalable approach to diaminopyrazoles using flow chemistry
Wilson, Noel S., Osuma, Augustine T., Camp, Jennifer A.Van, Xu, Xiangdong
Published in Tetrahedron letters (22.08.2012)
Published in Tetrahedron letters (22.08.2012)
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Journal Article
Development and Applications of a Practical Continuous Flow Microwave Cell
Wilson, Noel S., Sarko, Christopher R., Roth, Gregory P.
Published in Organic process research & development (01.05.2004)
Published in Organic process research & development (01.05.2004)
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Journal Article
Hit-to-lead studies on benzimidazole inhibitors of ITK: Discovery of a novel class of kinase inhibitors
Snow, Roger J., Abeywardane, Asitha, Campbell, Scot, Lord, John, Kashem, Mohammed A., Khine, Hnin Hnin, King, Josephine, Kowalski, Jennifer A., Pullen, Steven S., Roma, Teresa, Roth, Gregory P., Sarko, Christopher R., Wilson, Noel S., Winters, Michael P., Wolak, John P., Cywin, Charles L.
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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Journal Article
Construction and Validation of an Automated Flow Hydrogenation Instrument for Application in High-Throughput Organic Chemistry
Clapham, Bruce, Wilson, Noel S, Michmerhuizen, Melissa J, Blanchard, David P, Dingle, David M, Nemcek, Thomas A, Pan, Jeffrey Y, Sauer, Daryl R
Published in Journal of combinatorial chemistry (01.01.2008)
Published in Journal of combinatorial chemistry (01.01.2008)
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Journal Article
Solid phase synthesis of chiral 2-amino-benzimidazoles
Lee, Jinbo, Doucette, Amanda, Wilson, Noel S, Lord, John
Published in Tetrahedron letters (02.04.2001)
Published in Tetrahedron letters (02.04.2001)
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Journal Article
PRIMARY CARBOXAMIDES AS BTK INHIBITORS
NOEL S WILSON, ANIL VASUDEVAN, STACY A VAN EPPS, JII WAN, MICHAEL M FRIEDMAN, AUGUSTINE OSUMA, RAYMOND HUNTLEY, GAGANDEEP K SOMAL, J MARTIN HEROLD, XU XIANGDONG, GRIER A WALLACE, WANG LU, HEATHER M DAVIS, MICHAEL Z HOEMANN, GEORGE SHEPPARD, DOMINIQUE BONAFOUX, KRISTINE E FRANK, JENNIFER VAN CAMP
Year of Publication 07.01.2021
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Year of Publication 07.01.2021
Patent
PRIMARY CARBOXAMIDES AS BTK INHIBITORS
NOEL S WILSON, ANIL VASUDEVAN, STACY A VAN EPPS, JII WAN, MICHAEL M FRIEDMAN, AUGUSTINE OSUMA, RAYMOND HUNTLEY, GAGANDEEP K SOMAL, J MARTIN HEROLD, XU XIANGDONG, GRIER A WALLACE, WANG LU, HEATHER M DAVIS, MICHAEL Z HOEMANN, GEORGE SHEPPARD, DOMINIQUE BONAFOUX, KRISTINE E FRANK, JENNIFER VAN CAMP
Year of Publication 25.07.2019
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Year of Publication 25.07.2019
Patent
MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF
NOEL S WILSON, ALAN F GASIECKI, ZHAO HONGYU, ANA-LUCIA RELO, CHRISTINA M THOMPSON, BRAJE WILFRIED, ALBERT W KRUGER, DENNIE S WELCH, TURNER SEAN C, LI HUANQIU, ZHANG MIN, IRINI AKRITOPOULOU-ZANZE, SHASHANK SHEKHAR, GANDARILLA JORGE, STEVAN W DJURIC
Year of Publication 14.01.2016
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Year of Publication 14.01.2016
Patent
ChemInform Abstract: A Scalable Approach to Diaminopyrazoles Using Flow Chemistry
Wilson, Noel S., Osuma, Augustine T., Van Camp, Jennifer A., Xu, Xiangdong
Published in ChemInform (27.11.2012)
Published in ChemInform (27.11.2012)
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Journal Article
Recent trends in microwave-assisted synthesis
Wilson, Noel S, Roth, Gregory P
Published in Current opinion in drug discovery & development (01.07.2002)
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Published in Current opinion in drug discovery & development (01.07.2002)
Journal Article