Discovery of a new sialic acid binding region that regulates Siglec-7
Yamakawa, Nao, Yasuda, Yu, Yoshimura, Atsushi, Goshima, Ami, Crocker, Paul R, Vergoten, Gérard, Nishiura, Yuji, Takahashi, Takashi, Hanashima, Shinya, Matsumoto, Kana, Yamaguchi, Yoshiki, Tanaka, Hiroshi, Kitajima, Ken, Sato, Chihiro
Published in Scientific reports (26.05.2020)
Published in Scientific reports (26.05.2020)
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Journal Article
Enantioselective 1,3-Dipolar Cycloadditions of a-Methylene Lactams to Construct Spirocycles
Nishiura, Yuji, Gonzalez, Kevin J., Cusumano, Alexander Q., Stoltz, Brian M.
Published in Organic letters (29.08.2023)
Published in Organic letters (29.08.2023)
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Journal Article
Palladium-Catalyzed Asymmetric Conjugate Addition of Arylboronic Acids to α,β-Unsaturated Lactams: Enantioselective Construction of All-Carbon Quaternary Stereocenters in Saturated Nitrogen-Containing Heterocycles
Zhang, Tianyi, Nishiura, Yuji, Cusumano, Alexander Q., Stoltz, Brian M.
Published in Organic letters (08.09.2023)
Published in Organic letters (08.09.2023)
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Journal Article
Enantioselective 1,3-Dipolar Cycloadditions of α‑Methylene Lactams to Construct Spirocycles
Nishiura, Yuji, Gonzalez, Kevin J., Cusumano, Alexander Q., Stoltz, Brian M.
Published in Organic letters (08.09.2023)
Published in Organic letters (08.09.2023)
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Journal Article
Stereoselective Synthesis of Oligo-α-(2,8)-Sialic Acids
Tanaka, Hiroshi, Nishiura, Yuji, Takahashi, Takashi
Published in Journal of the American Chemical Society (07.06.2006)
Published in Journal of the American Chemical Society (07.06.2006)
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Journal Article
1775-P: Impact of Acetyl-CoA Carboxylase 2 Inhibition on Skeletal Muscle Diacylglycerol and Ceramide Levels and Its Potential Contribution to Improved Glucose Metabolism
TAKAGI, HIROYUKI, IKEHARA, TATSUYA, HASHIMOTO, KUMI, SHIMAZAKI, ATSUYUKI, KASHIWAGI, YUTO, NISHIURA, YUJI, NOTOYA, MITSURU, YUKIOKA, HIDEO
Published in Diabetes (New York, N.Y.) (01.06.2019)
Published in Diabetes (New York, N.Y.) (01.06.2019)
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Journal Article
Discovery of a novel olefin derivative as a highly potent and selective acetyl-CoA carboxylase 2 inhibitor with in vivo efficacy
Nishiura, Yuji, Matsumura, Akira, Kobayashi, Naotake, Shimazaki, Atsuyuki, Sakamoto, Shingo, Kitade, Naohisa, Tonomura, Yutaka, Ino, Akira, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
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Journal Article
FUSED RING COMPOUND HAVING GLP-1 RECEPTOR AGONIST EFFECT
KUSANO, Hiroki, MAENO, Shomitsu, NISHIURA, Yuji, WADA, Toshihiro, KITAMURA FUJIWARA, Misato
Year of Publication 28.03.2024
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Year of Publication 28.03.2024
Patent
An Efficient Convergent Synthesis of GP1c Ganglioside Epitope
Tanaka, Hiroshi, Nishiura, Yuji, Takahashi, Takashi
Published in Journal of the American Chemical Society (24.12.2008)
Published in Journal of the American Chemical Society (24.12.2008)
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Journal Article
MGAT2 저해 활성을 갖는 축합환 유도체
MASUDA KENGO, SASAKI YOSHIKAZU, NODU KOUHEI, TATENO YUSUKE, NISHIURA YUJI
Year of Publication 18.03.2020
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Year of Publication 18.03.2020
Patent
Design, synthesis and identification of novel benzimidazole derivatives as highly potent NPY Y5 receptor antagonists with attractive in vitro ADME profiles
Tamura, Yuusuke, Omori, Naoki, Kouyama, Naoki, Nishiura, Yuji, Hayashi, Kyouhei, Watanabe, Kana, Tanaka, Yukari, Chiba, Takeshi, Yukioka, Hideo, Sato, Hiroki, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Journal Article
Efficient Synthesis of an α(2,9) Trisialic Acid by One-Pot Glycosylation and Polymer-Assisted Deprotection
Tanaka, Hiroshi, Tateno, Yusuke, Nishiura, Yuji, Takahashi, Takashi
Published in Organic letters (18.12.2008)
Published in Organic letters (18.12.2008)
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Journal Article
FUSED-RING DERIVATIVE HAVING MGAT2 INHIBITORY ACTIVITY
NODU Kouhei, TATENO Yusuke, MASUDA Kengo, NISHIURA Yuji, SASAKI Yoshikazu
Year of Publication 17.01.2019
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Year of Publication 17.01.2019
Patent