Facile synthesis of indole 3-acetic acid and azaindole 3-acetic acid derivatives
Yamada, Koji, Ohta, Mariko, Kitamura, Go, Tsutsumiguchi, Suzuka, Nishi, Takahide
Published in Tetrahedron (06.04.2023)
Published in Tetrahedron (06.04.2023)
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Syntheses of Oxazolidinone-2,3-Fused Indoline and Azaindoline Derivatives
Yamada, Koji, Ishizawa, Kaho, Oonishi, Yoshihiro, Sato, Yoshihiro, Nishi, Takahide
Published in Synlett (23.02.2023)
Published in Synlett (23.02.2023)
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Silver-Mediated Intramolecular Friedel-Crafts-Type Cyclizations of 2-Benzyloxy-3-bromoindolines: Synthesis of Isochromeno[3,4-b] indolines and 3-Arylindoles
Yamashiro, Toshiki, Yamada, Koji, Yoshida, Haruka, Tomisaka, Yutaro, Nishi, Takahide, Abe, Takumi
Published in Synlett (17.12.2019)
Published in Synlett (17.12.2019)
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Journal Article
Syntheses and antimicrobial activities of ogipeptin derivatives
Takiguchi, Shingo, Homma, Hidehito, Fujisawa, Tetsunori, Hirota-Takahata, Yuki, Ono, Yasunori, Kizuka, Masaaki, Ishii, Yuki, Yoshimura, Satomichi, Nishi, Takahide
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
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Structure-based drug design of tricyclic 8H-indeno[1,2-d][1,3]thiazoles as potent FBPase inhibitors
Tsukada, Tomoharu, Takahashi, Mizuki, Takemoto, Toshiyasu, Kanno, Osamu, Yamane, Takahiro, Kawamura, Sayako, Nishi, Takahide
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Design and optimization of novel (2S,4S,5S)-5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxy-2-isopropylhexanamides as renin inhibitors
Nakamura, Yuji, Sugita, Chie, Meguro, Masaki, Miyazaki, Shojiro, Tamaki, Kazuhiko, Takahashi, Mizuki, Nagai, Yoko, Nagayama, Takahiro, Kato, Mikio, Suemune, Hiroshi, Nishi, Takahide
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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Journal Article
Discovery of CS-2100, a potent, orally active and S1P3-sparing S1P1 agonist
Nakamura, Tsuyoshi, Asano, Masayoshi, Sekiguchi, Yukiko, Mizuno, Yumiko, Tamaki, Kazuhiko, Kimura, Takako, Nara, Futoshi, Kawase, Yumi, Shimozato, Takaichi, Doi, Hiromi, Kagari, Takashi, Tomisato, Wataru, Inoue, Ryotaku, Nagasaki, Miyuki, Yuita, Hiroshi, Oguchi-Oshima, Keiko, Kaneko, Reina, Watanabe, Nobuaki, Abe, Yasuyuki, Nishi, Takahide
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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Journal Article
Discovery of DS-8108b, a Novel Orally Bioavailable Renin Inhibitor
Nakamura, Yuji, Fujimoto, Teppei, Ogawa, Yasuyuki, Sugita, Chie, Miyazaki, Shojiro, Tamaki, Kazuhiko, Takahashi, Mizuki, Matsui, Yumi, Nagayama, Takahiro, Manabe, Kenichi, Mizuno, Makoto, Masubuchi, Noriko, Chiba, Katsuyoshi, Nishi, Takahide
Published in ACS medicinal chemistry letters (13.09.2012)
Published in ACS medicinal chemistry letters (13.09.2012)
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Journal Article
EFFICIENT SYNTHESIS OF 5-AMINO-6-DIALKYLAMINO-4-HYDROXYPENTANAMIDE DERIVATIVES FOR RENIN INHIBITORS
Nakamura, Yuji, Ogawa, Yasuyuki, Suzuki, Chie, Fujimoto, Teppei, Miyazaki, Shojiro, Tamaki, Kazuhiko, Nishi, Takahide, Suemune, Hiroshi
Published in Heterocycles (01.07.2011)
Published in Heterocycles (01.07.2011)
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Journal Article
Synthesis and SAR of 1,3-thiazolyl thiophene and pyridine derivatives as potent, orally active and S1P3-sparing S1P1 agonists
Asano, Masayoshi, Nakamura, Tsuyoshi, Sekiguchi, Yukiko, Mizuno, Yumiko, Yamaguchi, Takahiro, Tamaki, Kazuhiko, Shimozato, Takaichi, Doi-Komuro, Hiromi, Kagari, Takashi, Tomisato, Wataru, Inoue, Ryotaku, Yuita, Hiroshi, Oguchi-Oshima, Keiko, Kaneko, Reina, Nara, Futoshi, Kawase, Yumi, Masubuchi, Noriko, Nakayama, Shintaro, Koga, Tetsufumi, Namba, Eiko, Nasu, Hatsumi, Nishi, Takahide
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
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Journal Article
Synthesis and evaluation of CS-2100, a potent, orally active and S1P3- sparing S1P1 agonist
Nakamura, Tsuyoshi, Asano, Masayoshi, Sekiguchi, Yukiko, Mizuno, Yumiko, Tamaki, Kazuhiko, Nara, Futoshi, Kawase, Yumi, Yabe, Yoshiyuki, Nakai, Daisuke, Kamiyama, Emi, Urasaki-Kaneno, Yoko, Shimozato, Takaichi, Doi-Komuro, Hiromi, Kagari, Takashi, Tomisato, Wataru, Inoue, Ryotaku, Nagasaki, Miyuki, Yuita, Hiroshi, Oguchi-Oshima, Keiko, Kaneko, Reina, Nishi, Takahide
Published in European journal of medicinal chemistry (01.05.2012)
Published in European journal of medicinal chemistry (01.05.2012)
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Journal Article
[3 + 2] cycloaddition of 1-(4-Methoxybenzyl)indoles and azaindoles with nitrile oxides
Kimura, Reina, Sato, Yoshihiro, Morisaki, Kazuhiro, Nishi, Takahide
Published in Tetrahedron (07.05.2022)
Published in Tetrahedron (07.05.2022)
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Journal Article
Discovery of CS-0777: A Potent, Selective, and Orally Active S1P1 Agonist
Nishi, Takahide, Miyazaki, Shojiro, Takemoto, Toshiyasu, Suzuki, Keisuke, Iio, Yukiko, Nakajima, Katsuyoshi, Ohnuki, Takashi, Kawase, Yumi, Nara, Futoshi, Inaba, Shinichi, Izumi, Takashi, Yuita, Hiroshi, Oshima, Keiko, Doi, Hiromi, Inoue, Ryotaku, Tomisato, Wataru, Kagari, Takashi, Shimozato, Takaichi
Published in ACS medicinal chemistry letters (12.05.2011)
Published in ACS medicinal chemistry letters (12.05.2011)
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