An oral antisense oligonucleotide for PCSK9 inhibition
Gennemark, Peter, Walter, Katrin, Clemmensen, Niclas, Rekić, Dinko, Nilsson, Catarina A M, Knöchel, Jane, Hölttä, Mikko, Wernevik, Linda, Rosengren, Birgitta, Kakol-Palm, Dorota, Wang, Yanfeng, Yu, Rosie Z, Geary, Richard S, Riney, Stan J, Monia, Brett P, Isaksson, Rikard, Jansson-Löfmark, Rasmus, Rocha, Cristina S J, Lindén, Daniel, Hurt-Camejo, Eva, Crooke, Rosanne, Tillman, Lloyd, Rydén-Bergsten, Tina, Carlsson, Björn, Andersson, Ulf, Elebring, Marie, Tivesten, Anna, Davies, Nigel
Published in Science translational medicine (12.05.2021)
Published in Science translational medicine (12.05.2021)
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Predicting Intestinal Precipitation—A Case Example for a Basic BCS Class II Drug
Carlert, Sara, Pålsson, Anna, Hanisch, Gunilla, von Corswant, Christian, Nilsson, Catarina, Lindfors, Lennart, Lennernäs, Hans, Abrahamsson, Bertil
Published in Pharmaceutical research (01.10.2010)
Published in Pharmaceutical research (01.10.2010)
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Type 2 Diabetes and Pancreatic Exocrine Function: Associations Between Fecal Elastase-1 Levels and Gastrointestinal Symptoms, Plasma Nutritional Markers, and Uptake of Free Versus Esterified Omega-3 Fatty Acids in a Randomized, Open-Label, Crossover Study
Oscarsson, Jan, Nilsson, Catarina A, Kvarnström, Mats, Lindkvist, Bjorn
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2017)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2017)
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Comparative quantitative systems pharmacology modeling of anti-PCSK9 therapeutic modalities in hypercholesterolemia[S]
Sokolov, Victor, Helmlinger, Gabriel, Nilsson, Catarina, Zhudenkov, Kirill, Skrtic, Stanko, Hamrén, Bengt, Peskov, Kirill, Hurt-Camejo, Eva, Jansson-Löfmark, Rasmus
Published in Journal of lipid research (01.09.2019)
Published in Journal of lipid research (01.09.2019)
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Journal Article
Effects of Food on the Pharmacokinetics of Omega-3-Carboxylic Acids in Healthy Japanese Male Subjects: A Phase I, Randomized, Open-label, Three-period, Crossover Trial
Shimada, Hitoshi, Nilsson, Catarina, Noda, Yoshinori, Kim, Hyosung, Lundström, Torbjörn, Yajima, Toshitaka
Published in Journal of Atherosclerosis and Thrombosis (01.01.2017)
Published in Journal of Atherosclerosis and Thrombosis (01.01.2017)
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Abstract 13307: An Oral Antisense Oligonucleotide for PCSK9 Inhibition in Humans
Gennemark, Peter, Walter, Katrin, Clemmensen, Niclas, Rekic, Dinko, Nilsson, Catarina, Knoechel, Jane, Holtta, Mikko, Wang, Yanfeng, Yu, Rosie, riney, stanley, Monia, Brett P, Andersson, Ulf, Jansson-Lofmark, Rasmus, Rocha, Cristina S, Linden, Daniel, Ryden-Bergsten, Kristina, Hurt-Camejo, Eva, CROOKE, Rosanne M, Tillman, Lloyd, Carlsson, Bjorn, Elebring, Marie, Tivesten, Anna, Davies, Nigel
Published in Circulation (New York, N.Y.) (17.11.2020)
Published in Circulation (New York, N.Y.) (17.11.2020)
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Omega-3 fatty acid exposure with a low-fat diet in patients with past hypertriglyceridemia-induced acute pancreatitis; an exploratory, randomized, open-label crossover study
Dunbar, Richard L, Gaudet, Daniel, Davidson, Michael, Rensfeldt, Martin, Yang, Hong, Nilsson, Catarina, Kvarnström, Mats, Oscarsson, Jan
Published in Lipids in health and disease (30.05.2020)
Published in Lipids in health and disease (30.05.2020)
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A case‐study of model‐informed drug development of a novel PCSK9 anti sense oligonucleotide. Part 1: First time in man to phase II
Knöchel, Jane, Nilsson, Catarina, Carlsson, Björn, Wernevik, Linda, Hofherr, Alexis, Gennemark, Peter, Jansson‐Löfmark, Rasmus, Isaksson, Rikard, Rydén‐Bergsten, Tina, Hamrén, Bengt, Rekić, Dinko
Published in CPT: pharmacometrics and systems pharmacology (01.12.2022)
Published in CPT: pharmacometrics and systems pharmacology (01.12.2022)
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Assessment of pharmacokinetic interaction between omega-3 carboxylic acids and the statins rosuvastatin and simvastatin: Results of 2 phase I studies in healthy volunteers
Offman, Elliot, PhD, Davidson, Michael, MD, Nilsson, Catarina, MSc
Published in Journal of clinical lipidology (01.05.2017)
Published in Journal of clinical lipidology (01.05.2017)
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Tu1372 - Type 2 Diabetes and Pancreatic Exocrine Function: Associations Between Fecal Elastase-1 Levels and Gastrointestinal Symptoms, Plasma Nutritional Markers, and Uptake of Free Versus Esterified Omega-3 Fatty Acids in a Randomized, Open-Label, Crossover Study
Oscarsson, Jan, Nilsson, Catarina A., Kvarnström, Mats, Lindkvist, Bjorn
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2017)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2017)
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ETESIAN: A PHASE 2B STUDY OF THE EFFICACY, SAFETY AND TOLERABILITY OF AZD8233, A PCSK9-TARGETED ANTISENSE OLIGONUCLEOTIDE, IN PATIENTS WITH DYSLIPIDEMIA
Koren, Michael J., Hofherr, Alexis, Schumi, Jennifer, Rekic, Dinko, Knochel, Jane, Nilsson, Catarina A.M., Rudvik, Anna, Wernevik, Linda, Ryden-Bergsten, Tina, Carlsson, Bjorn C.L.
Published in Journal of the American College of Cardiology (01.03.2022)
Published in Journal of the American College of Cardiology (01.03.2022)
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AZD8233 antisense oligonucleotide targeting PCSK9 does not prolong QT interval
Rekić, Dinko, Azarov, Ivan, Knöchel, Jane, Sokolov, Victor, Nilsson, Catarina, Wernevik, Linda, Han, David, Rydén‐Bergsten, Tina, Ebrahimi, Ahmad, Dota, Corina, Carlsson, Björn
Published in British journal of clinical pharmacology (01.11.2022)
Published in British journal of clinical pharmacology (01.11.2022)
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Journal Article
Population pharmacokinetics of a novel PCSK9 antisense oligonucleotide
Clewe, Oskar, Rekić, Dinko, Quartino, Angelica L., Carlsson, Björn, Higashimori, Mitsuo, Wernevik, Linda, Hofherr, Alexis, Rydén‐Bergsten, Tina, Nilsson, Catarina, Knöchel, Jane
Published in British journal of clinical pharmacology (01.06.2024)
Published in British journal of clinical pharmacology (01.06.2024)
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No Effect of Omega-3 Carboxylic Acids on Pharmacokinetics/Pharmacodynamics of Warfarin or on Platelet Function When Co-administered with Acetylsalicylic Acid: Results of Two Phase I Studies in Healthy Volunteers
Offman, Elliot, Davidson, Michael, Nilsson, Catarina
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.06.2017)
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.06.2017)
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Journal Article
Delayed Density-Dependence in a Small-Rodent Population
Agrell, Jep, Erlinge, Sam, Nelson, Johan, Nilsson, Catarina, Persson, Irene
Published in Proceedings of the Royal Society. B, Biological sciences (23.10.1995)
Published in Proceedings of the Royal Society. B, Biological sciences (23.10.1995)
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Abstract 9747: Safety, Pharmacokinetics and Pharmacodynamics of Multiple Ascending Doses of AZD8233, Targeting PCSK9, in Patients with Dyslipidemia
Hofherr, Alexis, Nilsson, Catarina A, Rekic, Dinko, Knoechel, Jane, Goldwater, Ronald, Han, David, Kusnir, Jorge, Overcash, J. Scott, Waters, Michael, White, Alexander, Hurt-Camejo, Eva, Wernevik, Linda, Isaksson, Rikard, Wang, Yanfeng, Bhanot, Sanjay, Ryden-Bergsten, Kristina, Koren, Michael, Carlsson, Bjorn C
Published in Circulation (New York, N.Y.) (16.11.2021)
Published in Circulation (New York, N.Y.) (16.11.2021)
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Journal Article
Importance of pancreatic exocrine dysfunction in patients with type 2 diabetes: A randomized crossover study
Lindkvist, Björn, Nilsson, Catarina, Kvarnström, Mats, Oscarsson, Jan
Published in Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.] (01.07.2018)
Published in Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.] (01.07.2018)
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Abstract 13913: Single Dose Safety, Pharmacokinetics, and Pharmacodynamics of a Potent PCSK9 Synthesis Inhibitor, AZD8233, in Subjects With Elevated Ldl Cholesterol
Nilsson, Catarina, Monia, Brett P, Ryden-Bergsten, Kristina, Rekic, Dinko, Hurt-Camejo, Eva, Bhanot, Sanjay, Tsimikas, Sotirios, Geary, Richard, Hofherr, Alexis, Crooke, Rosanne M, knöchel, jane, Wernevik, Linda, Arfvidsson, Cecilia, Isaksson, Rikard, Carlsson, Bjorn, Han, David, henry, scott
Published in Circulation (New York, N.Y.) (17.11.2020)
Published in Circulation (New York, N.Y.) (17.11.2020)
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