Novel Inhibition of Porcine Pepsin by a Substituted Piperidine
Marcinkeviciene, Jovita, Kopcho, Lisa M., Yang, Tao, Copeland, Robert A., Glass, Brian M., Combs, Andrew P., Falahatpisheh, Nikoo, Thompson, Lorin
Published in The Journal of biological chemistry (09.08.2002)
Published in The Journal of biological chemistry (09.08.2002)
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Journal Article
The Novel Bromodomain and Extraterminal Domain Inhibitor INCB054329 Induces Vulnerabilities in Myeloma Cells That Inform Rational Combination Strategies
Stubbs, Matthew C, Burn, Timothy C, Sparks, Richard, Maduskuie, Thomas, Diamond, Sharon, Rupar, Mark, Wen, Xiaoming, Volgina, Alla, Zolotarjova, Nina, Waeltz, Paul, Favata, Margaret, Jalluri, Ravi, Liu, Huiqing, Liu, Xuesong Mike, Li, Jun, Collins, Robert, Falahatpisheh, Nikoo, Polam, Padmaja, DiMatteo, Darlise, Feldman, Patricia, Dostalik, Valerie, Thekkat, Pramod, Gardiner, Christine, He, Xin, Li, Yanlong, Covington, Maryanne, Wynn, Richard, Ruggeri, Bruce, Yeleswaram, Swamy, Xue, Chu-Biao, Yao, Wenqing, Combs, Andrew P, Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip C C
Published in Clinical cancer research (01.01.2019)
Published in Clinical cancer research (01.01.2019)
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INCB050465 (Parsaclisib), a Novel Next-Generation Inhibitor of Phosphoinositide 3‑Kinase Delta (PI3Kδ)
Yue, Eddy W, Li, Yun-Long, Douty, Brent, He, Chunhong, Mei, Song, Wayland, Brian, Maduskuie, Thomas, Falahatpisheh, Nikoo, Sparks, Richard B, Polam, Padmaja, Zhu, Wenyu, Glenn, Joseph, Feng, Hao, Zhang, Ke, Li, Yanlong, He, Xin, Katiyar, Kamna, Covington, Maryanne, Feldman, Patricia, Shin, Niu, Wang, Kathy He, Diamond, Sharon, Li, Yu, Koblish, Holly K, Hall, Leslie, Scherle, Peggy, Yeleswaram, Swamy, Xue, Chu-Biao, Metcalf, Brian, Combs, Andrew P, Yao, Wenqing
Published in ACS medicinal chemistry letters (14.11.2019)
Published in ACS medicinal chemistry letters (14.11.2019)
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Abstract 5071: Preclinical characterization of the potent and selective BET inhibitor INCB057643 in models of hematologic malignancies
Stubbs, Matthew C., Maduskuie, Thomas, Burn, Timothy, Diamond-Fosbenner, Sharon, Falahatpisheh, Nikoo, Volgina, Alla, Zolotarjova, Nina, Wen, Xiaoming, Feldman, Patricia, Rupar, Mark, Collins, Robert, Marando, Cindy, Ruggeri, Bruce, Covington, Maryanne, Liu, Xuesong Mike, Wynn, Richard, Yeleswaram, Swamy, Yao, Wenqing, Huber, Reid, Hollis, Gregory, Scherle, Peggy, Combs, Andrew P., Liu, Phillip C.
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Abstract 3525: The BET inhibitor INCB054329 is efficacious as a single agent or in combination with targeted agents in colorectal cancer models
Liu, Xuesong, Li, Jun, He, Xin, Stubbs, Matthew, Favata, Margaret, Wen, Xiaoming, Chang, Hong, Rumberger, Beth R., Li, Yanlong, Maduskuie, Thomas, Sparks, Richard, Falahatpisheh, Nikoo, Polam, Padmaja, Combs, Andrew P., Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip C.
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Abstract C103: The combination of PI3kδ-selective inhibition and immunomodulation shows efficacy in solid tumor models
Koblish, Holly K., Wang, Liang-Chuan, Hansbury, Michael, Zhang, Yue, Yang, Gengjie, Burn, Timothy, Waeltz, Paul, Rupar, Mark, Yue, Eddy, Douty, Brent, Maduskuie, Thomas, Falahatpisheh, Nikoo, Li, Yun-long, Combs, Andrew, Hollis, Gregory, Huber, Reid, Scherle, Peggy
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Abstract 691: Activity of the BET inhibitor INCB054329 in models of multiple myeloma
Stubbs, Matthew, Wen, Xiaoming, Dostalik, Valerie, O'Connor, Sybil, Caulder, Eian, Vogina, Alla, Maduskuie, Thomas, Sparks, Richard, Huang, Taisheng, Falahatpisheh, Nikoo, Polam, Padmaja, Xue, Chu-Biao, Liu, Xuesong M., Burn, Timothy, Vaddi, Kris, Combs, Andrew P., Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip CC
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
Abstract 3523: Discovery of a novel BET inhibitor INCB054329
Liu, Phillip CC, Liu, Xuesong Mike, Stubbs, Matthew C., Maduskuie, Thomas, Sparks, Richard, Zolotarjova, Nina, Li, Jun, Wen, Xiaoming, Favata, Margaret, Feldman, Patricia, Volgina, Alla, DiMatteo, Darlise, Collins, Robert, Falahatpisheh, Nikoo, Polam, Padmaja, Li, Yu, Covington, Maryanne, Diamond-Fosbenner, Sharon, Wynn, Richard, Burn, Timothy, Vaddi, Kris, Yeleswaram, Swamy, Combs, Andrew P., Yao, Wenqing, Huber, Reid, Scherle, Peggy, Hollis, Gregory
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Abstract 692: The BET inhibitor INCB054329 is synergistic with JAK1 inhibition in models of multiple myeloma
Stubbs, Matthew C., Liu, Xuesong M., Wen, Xiaoming, Li, Jun, Dostalik, Valerie, O'Connor, Sybil, Caulder, Eian, Favata, Margaret, Rupar, Mark, Li, Yu, Rumberger, Beth, Maduskuie, Thomas, Sparks, Richard, Falahatpisheh, Nikoo, Polam, Padmaja, Vaddi, Kris, Burn, Timothy, Combs, Andrew P., Yao, Wenqing, Huber, Reid, Hollis, Gregory, Scherle, Peggy, Liu, Phillip CC
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Photochemically Enhanced Binding of Small Molecules to the Tumor Necrosis Factor Receptor-1 Inhibits the Binding of TNF-α
Carter, Percy H., Scherle, Peggy A., Muckelbauer, Jodi A., Voss, Matthew E., Liu, Rui-Qin, Thompson, Lorin A., Tebben, Andrew J., Solomon, Kimberly A., Lo, Yvonne C., Li, Zhong, Strzemienski, Paul, Yang, Gengjie, Falahatpisheh, Nikoo, Xu, Meizhong, Wu, Zhongren, Farrow, Neil A., Ramnarayan, Kal, Wang, Jing, Rideout, Darryl, Yalamoori, Venkatachalapathi, Domaille, Peter, Underwood, Dennis J., Trzaskos, James M., Friedman, Steven M., Newton, Robert C., Decicco, Carl P.
Published in Proceedings of the National Academy of Sciences - PNAS (09.10.2001)
Published in Proceedings of the National Academy of Sciences - PNAS (09.10.2001)
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Pharmacological inactivation of PI3Kδ in the tumor microenvironment enhances efficacy of other immunotherapeutic agents
Wang, Liang-Chuan S, Koblish, Holly, Hansbury, Michael, Zhang, Yue, Yang, Gengjie, Burn, Timothy, Waeltz, Paul, Rupar, Mark, Yue, Eddy, Douty, Brent, Maduskuie, Thomas, Falahatpisheh, Nikoo, Li, Yun-Long, Combs, Andrew P, Hollis, Gregory, Huber, Reid, Scherle, Peggy
Published in Journal for immunotherapy of cancer (04.11.2015)
Published in Journal for immunotherapy of cancer (04.11.2015)
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