K-Ras(G12D)-selective inhibitory peptides generated by random peptide T7 phage display technology
Sakamoto, Kotaro, Kamada, Yusuke, Sameshima, Tomoya, Yaguchi, Masahiro, Niida, Ayumu, Sasaki, Shigekazu, Miwa, Masanori, Ohkubo, Shoichi, Sakamoto, Jun-ichi, Kamaura, Masahiro, Cho, Nobuo, Tani, Akiyoshi
Published in Biochemical and biophysical research communications (11.03.2017)
Published in Biochemical and biophysical research communications (11.03.2017)
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Investigation of the structural requirements of K-Ras(G12D) selective inhibitory peptide KRpep-2d using alanine scans and cysteine bridging
Niida, Ayumu, Sasaki, Shigekazu, Yonemori, Kazuko, Sameshima, Tomoya, Yaguchi, Masahiro, Asami, Taiji, Sakamoto, Kotaro, Kamaura, Masahiro
Published in Bioorganic & medicinal chemistry letters (15.06.2017)
Published in Bioorganic & medicinal chemistry letters (15.06.2017)
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Unequivocal Synthesis of (Z)-Alkene and (E)-Fluoroalkene Dipeptide Isosteres To Probe Structural Requirements of the Peptide Transporter PEPT1
Niida, Ayumu, Tomita, Kenji, Mizumoto, Makiko, Tanigaki, Hiroaki, Terada, Tomohiro, Oishi, Shinya, Otaka, Akira, Inui, Ken-ichi, Fujii, Nobutaka
Published in Organic letters (16.02.2006)
Published in Organic letters (16.02.2006)
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Transport Characteristics of a Novel Peptide Transporter 1 Substrate, Antihypotensive Drug Midodrine, and Its Amino Acid Derivatives
Tsuda, Masahiro, Terada, Tomohiro, Irie, Megumi, Katsura, Toshiya, Niida, Ayumu, Tomita, Kenji, Fujii, Nobutaka, Inui, Ken-ichi
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
Metastin and its variant forms suppress migration of pancreatic cancer cells
Masui, Toshihiko, Doi, Ryuichiro, Mori, Tomohiko, Toyoda, Eiji, Koizumi, Masayuki, Kami, Kazuhiro, Ito, Daisuke, Peiper, Stephen C, Broach, James R, Oishi, Shinya, Niida, Ayumu, Fujii, Nobutaka, Imamura, Masayuki
Published in Biochemical and biophysical research communications (27.02.2004)
Published in Biochemical and biophysical research communications (27.02.2004)
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A Short-Length Peptide YY Analogue with Anorectic Effect in Mice
Nishizawa, Naoki, Niida, Ayumu, Masuda, Yasushi, Kumano, Satoshi, Yokoyama, Kotaro, Hirabayashi, Hideki, Amano, Nobuyuki, Ohtaki, Tetsuya, Asami, Taiji
Published in ACS omega (31.05.2017)
Published in ACS omega (31.05.2017)
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Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Palladium-Catalyzed Carbonylation of Amino Acid Derived Allylic Carbonates
Inokuchi, Eriko, Narumi, Tetsuo, Niida, Ayumu, Kobayashi, Kazuya, Tomita, Kenji, Oishi, Shinya, Ohno, Hiroaki, Fujii, Nobutaka
Published in Journal of organic chemistry (16.05.2008)
Published in Journal of organic chemistry (16.05.2008)
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Structure–activity relationship study on small peptidic GPR54 agonists
Tomita, Kenji, Niida, Ayumu, Oishi, Shinya, Ohno, Hiroaki, Cluzeau, Jérôme, Navenot, Jean-Marc, Wang, Zi-xuan, Peiper, Stephen C., Fujii, Nobutaka
Published in Bioorganic & medicinal chemistry (15.11.2006)
Published in Bioorganic & medicinal chemistry (15.11.2006)
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Stereoselective Synthesis of (Z)-Alkene-Containing Proline Dipeptide Mimetics
Sasaki, Yoshikazu, Niida, Ayumu, Tsuji, Takashi, Shigenaga, Akira, Fujii, Nobutaka, Otaka, Akira
Published in Journal of organic chemistry (23.06.2006)
Published in Journal of organic chemistry (23.06.2006)
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A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres
Narumi, Tetsuo, Niida, Ayumu, Tomita, Kenji, Oishi, Shinya, Otaka, Akira, Ohno, Hiroaki, Fujii, Nobutaka
Published in Chemical communications (Cambridge, England) (01.01.2006)
Published in Chemical communications (Cambridge, England) (01.01.2006)
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Synthesis of (Z)-Alkene and (E)-Fluoroalkene-Containing Diketopiperazine Mimetics Utilizing Organocopper-Mediated Reduction−Alkylation and Diastereoselectivity Examination Using DFT Calculations
Niida, Ayumu, Mizumoto, Makiko, Narumi, Tetsuo, Inokuchi, Eriko, Oishi, Shinya, Ohno, Hiroaki, Otaka, Akira, Kitaura, Kazuo, Fujii, Nobutaka
Published in Journal of organic chemistry (26.05.2006)
Published in Journal of organic chemistry (26.05.2006)
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Application of tri- and tetrasubstituted alkene dipeptide mimetics to conformational studies of cyclic RGD peptides
Oishi, Shinya, Miyamoto, Kazuhide, Niida, Ayumu, Yamamoto, Mikio, Ajito, Keiichi, Tamamura, Hirokazu, Otaka, Akira, Kuroda, Yoshihiro, Asai, Akira, Fujii, Nobutaka
Published in Tetrahedron (13.02.2006)
Published in Tetrahedron (13.02.2006)
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Facile access to (Z)-alkene-containing diketopiperazine mimetics utilizing organocopper-mediated anti-SN2′ reactions
Niida, Ayumu, Oishi, Shinya, Sasaki, Yoshikazu, Mizumoto, Makiko, Tamamura, Hirokazu, Fujii, Nobutaka, Otaka, Akira
Published in Tetrahedron letters (01.06.2005)
Published in Tetrahedron letters (01.06.2005)
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Journal Article
Crystal Structure of a Human K‑Ras G12D Mutant in Complex with GDP and the Cyclic Inhibitory Peptide KRpep-2d
Sogabe, Satoshi, Kamada, Yusuke, Miwa, Masanori, Niida, Ayumu, Sameshima, Tomoya, Kamaura, Masahiro, Yonemori, Kazuko, Sasaki, Shigekazu, Sakamoto, Jun-ichi, Sakamoto, Kotaro
Published in ACS medicinal chemistry letters (13.07.2017)
Published in ACS medicinal chemistry letters (13.07.2017)
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Potent antiobesity effect of a short-length peptide YY-analogue continuously administered in mice
Nishizawa, Naoki, Niida, Ayumu, Adachi, Yusuke, Masuda, Yasushi, Kumano, Satoshi, Yokoyama, Kotaro, Asakawa, Tomoko, Hirabayashi, Hideki, Amano, Nobuyuki, Takekawa, Shiro, Ohtaki, Tetsuya, Asami, Taiji
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
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