Discovery and biochemical characterization of selective ATP competitive inhibitors of the human mitotic kinesin KSP
Rickert, Keith W., Schaber, Michael, Torrent, Maricel, Neilson, Lou Anne, Tasber, Edward S., Garbaccio, Robert, Coleman, Paul J., Harvey, Diane, Zhang, Yun, Yang, Yi, Marshall, Gary, Lee, Ling, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A.
Published in Archives of biochemistry and biophysics (15.01.2008)
Published in Archives of biochemistry and biophysics (15.01.2008)
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Kinesin spindle protein (KSP) inhibitors. Part 7: Design and synthesis of 3,3-disubstituted dihydropyrazolobenzoxazines as potent inhibitors of the mitotic kinesin KSP
Garbaccio, Robert M., Tasber, Edward S., Neilson, Lou Anne, Coleman, Paul J., Fraley, Mark E., Olson, Christy, Bergman, Jeff, Torrent, Maricel, Buser, Carolyn A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Lobell, Robert B., Tao, Weikang, South, Vicki J., Diehl, Ronald E., Davide, Joseph P., Yan, Youwei, Kuo, Lawrence C., Li, Chunze, Prueksaritanont, Thomayant, Fernandez-Metzler, Carmen, Mahan, Elizabeth A., Slaughter, Donald E., Salata, Joseph J., Kohl, Nancy E., Huber, Hans E., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
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N-Alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, μ and δ opioid agonists: a μ address
CARSON, John R, COATS, Steven J, ZHANG, Sui-Po, CODD, Ellen E, DAX, Scott L, JUNG LEE, MARTINEZ, Rebecca P, MCKOWN, Linda A, NEILSON, Lou Anne, PITIS, Philip M, WU, Wu-Nan
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Methyl-substitution of an iminohydantoin spiropiperidine β-secretase (BACE-1) inhibitor has a profound effect on its potency
Egbertson, Melissa, McGaughey, Georgia B., Pitzenberger, Steven M., Stauffer, Shaun R., Coburn, Craig A., Stachel, Shawn J., Yang, Wenjin, Barrow, James C., Neilson, Lou Anne, McWherter, Melody, Perlow, Debra, Fahr, Bruce, Munshi, Sanjeev, Allison, Timothy J., Holloway, Katharine, Selnick, Harold G., Yang, ZhiQiang, Swestock, John, Simon, Adam J., Sankaranarayanan, Sethu, Colussi, Dennis, Tugusheva, Katherine, Lai, Ming-Tain, Pietrak, Beth, Haugabook, Shari, Jin, Lixia, Chen, I.-W., Holahan, Marie, Stranieri-Michener, Maria, Cook, Jacquelynn J., Vacca, Joseph, Graham, Samuel L.
Published in Bioorganic & medicinal chemistry letters (01.11.2015)
Published in Bioorganic & medicinal chemistry letters (01.11.2015)
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Development of Pyridopyrimidines as Potent Akt1/2 Inhibitors
Wu, Zhicai, Hartnett, John C., Neilson, Lou Anne, Robinson, Ronald G., Fu, Sheng, Barnett, Stanley F., Defeo-Jones, Deborah, Jones, Raymond E., Kral, Astrid M., Huber, Hans E., Hartman, George D., Bilodeau, Mark T.
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Development of Pyridopyrimidines as Potent Aktl/2 Inhibitors
ZHICAI WU, HARTNETT, John C, HARTMAN, George D, BILODEAU, Mark T, NEILSON, Lou Anne, ROBINSON, Ronald G, SHENG FU, BARRETT, Stanley F, DEFEO-JONES, Deborah, JONES, Raymond E, KRAL, Astrid M, HUBER, Hans E
Published in Bioorganic & medicinal chemistry letters (2008)
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Published in Bioorganic & medicinal chemistry letters (2008)
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N, N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, potent, selective δ opioid agonists
CARSON, John R, COATS, Steven J, CODD, Ellen E, DAX, Scott L, JUNG LEE, MARTINEZ, Rebecca P, NEILSON, Lou Anne, PITIS, Philip M, ZHANG, Sui-Po
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Journal Article
N-alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]benzamides, micro and delta opioid agonists: a micro address
Carson, John R, Coats, Steven J, Codd, Ellen E, Dax, Scott L, Lee, Jung, Martinez, Rebecca P, McKown, Linda A, Anne Neilson, Lou, Pitis, Philip M, Wu, Wu-Nan, Zhang, Sui-Po
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Synthesis and binding affinities of 4-diarylaminotropanes, a new class of delta opioid agonists
Boyd, R E, Carson, J R, Codd, E E, Gauthier, A D, Neilson, L A, Zhang, S P
Published in Bioorganic & medicinal chemistry letters (15.05.2000)
Published in Bioorganic & medicinal chemistry letters (15.05.2000)
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