Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging
Fabio, Karine, Guillon, Christophe, Lacey, Carl J., Lu, Shi-fang, Heindel, Ned D., Ferris, Craig F., Placzek, Michael, Jones, Graham, Brownstein, Michael J., Simon, Neal G.
Published in Bioorganic & medicinal chemistry (01.02.2012)
Published in Bioorganic & medicinal chemistry (01.02.2012)
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Doxycycline hydrogels as a potential therapy for ocular vesicant injury
Gordon, Marion K, Desantis, Andrea, Deshmukh, Manjeet, Lacey, Carl Jeffrey, Hahn, Rita A, Beloni, John, Anumolu, Sivanaga S, Schlager, John J, Gallo, Michael A, Gerecke, Donald R, Heindel, Ned D, Svoboda, Kathy K H, Babin, Michael C, Sinko, Patrick J
Published in Journal of ocular pharmacology and therapeutics (01.10.2010)
Published in Journal of ocular pharmacology and therapeutics (01.10.2010)
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SYNTHESIS AND EVALUATION OF WATER-SOLUBLE DIMETHYLAMINOETHYL ETHERS OF METHOXSALEN FOR PROLIFERATIVE SKIN DISORDERS
Guillon, Christophe D, Jan, Yi-Hua, Foster, Natalie, Choudhuri, Mridula, Saxena, Jaya, Mariano, Thomas M, Heck, Diane E, Laskin, Jeffrey D, Heindel, Ned D
Published in Heterocyclic letters (01.08.2018)
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Published in Heterocyclic letters (01.08.2018)
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Azetidinones as vasopressin V1a antagonists
Guillon, Christophe D., Koppel, Gary A., Brownstein, Michael J., Chaney, Michael O., Ferris, Craig F., Lu, Shi-fang, Fabio, Karine M., Miller, Marvin J., Heindel, Ned D., Hunden, David C., Cooper, Robin D.G., Kaldor, Stephen W., Skelton, Jeffrey J., Dressman, Bruce A., Clay, Michael P., Steinberg, Mitchell I., Bruns, Robert F., Simon, Neal G.
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Peripheral site acetylcholinesterase inhibitors targeting both inflammation and cholinergic dysfunction
Young, Sherri, Fabio, Karine, Guillon, Christophe, Mohanta, Pramod, Halton, Timothy A., Heck, Diane E., Flowers, Robert A., Laskin, Jeffrey D., Heindel, Ned D.
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Investigation of anticholinergic and non-steroidal anti-inflammatory prodrugs which reduce chemically induced skin inflammation
Young, Sherri C., Fabio, Karine M., Huang, Mou-Tuan, Saxena, Jaya, Harman, Meredith P., Guillon, Christophe D., Vetrano, Anna M., Heck, Diane E., Flowers II, Robert A., Heindel, Ned D., Laskin, Jeffrey D.
Published in Journal of applied toxicology (01.02.2012)
Published in Journal of applied toxicology (01.02.2012)
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Vasopressin antagonists as anxiolytics and antidepressants: recent developments
Simon, Neal G, Guillon, Christophe, Fabio, Karine, Heindel, Ned D, Lu, Shi-fang, Miller, Marvin, Ferris, Craig F, Brownstein, Michael J, Garripa, Carrie, Koppel, Gary A
Published in Recent patents on CNS drug discovery (01.06.2008)
Published in Recent patents on CNS drug discovery (01.06.2008)
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N ω -NITRO- N ω' -SUBSTITUTED GUANIDINES: A SIMPLE CLASS OF NITRIC OXIDE SYNTHASE INHIBITORS
Guillon, Christophe D, Wisnoski, David D, Saxena, Jaya, Heindel, Ned D, Heck, Diane E, Wolff, Donald J, Laskin, Jeffrey D
Published in Modern research in inflammation (01.05.2014)
Published in Modern research in inflammation (01.05.2014)
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Back-Scattering Interferometry: An Ultrasensitive Method for the Unperturbed Detection of Acetylcholinesterase-Inhibitor Interactions
Haddad, Gabrielle L., Young, Sherri C., Heindel, Ned D., Bornhop, Darryl J., Flowers II, Robert A.
Published in Angewandte Chemie (29.10.2012)
Published in Angewandte Chemie (29.10.2012)
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Inhibition of interferon-γ signaling by a mercurio-substituted dihydropsoralen in murine keratinocytes
Martey, Christine A., Vetrano, Anna M., Whittemore, Marilyn S., Mariano, Thomas M., Heck, Diane E., Laskin, Debra L., Heindel, Ned D., Laskin, Jeffrey D.
Published in Biochemical pharmacology (05.12.2005)
Published in Biochemical pharmacology (05.12.2005)
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Cell-impermeant pyridinium derivatives of psoralens as inhibitors of keratinocyte growth
Mariano, Thomas M., Vetrano, Anna M., Gentile, Shannon L., Heck, Diane E., Whittemore, Marilyn S., Guillon, Christophe D., Jabin, Ivan, Rapp, Robert D., Heindel, Ned D., Laskin, Jeffrey D.
Published in Biochemical pharmacology (2002)
Published in Biochemical pharmacology (2002)
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Mechanisms of growth inhibition in keratinocytes by mercurio-substituted 4′,5′-dihydropsoralens
Martey, Christine A., Vetrano, Anna M., Whittemore, Marilyn S., Mariano, Thomas M., Gentile, Shannon L., Heck, Diane E., Laskin, Debra L., Heindel, Ned D., Laskin, Jeffrey D.
Published in Biochemical pharmacology (01.06.2002)
Published in Biochemical pharmacology (01.06.2002)
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Carboxymethyl dextran lactone: A preactivated polymer for amine conjugations
Heindel, Ned D, Kauffman, Michael A, Akyea, Eric K, Engel, Stephanie A, Frey, Michael F, Lacey, C. Jeffrey, Egolf, Roger A
Published in Bioconjugate chemistry (01.01.1994)
Published in Bioconjugate chemistry (01.01.1994)
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Hydrazide pharmaceuticals as conjugates to polyaldehyde dextran: syntheses, characterization, and stability
Heindel, Ned D, Zhao, Huiru, Leiby, Jeffrey, VanDongen, Jacobus M, Lacey, C. Jeffrey, Lima, Daniel A, Shabsoug, Barakat, Buzby, John H
Published in Bioconjugate chemistry (01.01.1990)
Published in Bioconjugate chemistry (01.01.1990)
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Transfer hydrogenation of furocoumarin derivatives
Heindel, Ned D, Foster, Natalie, Choudhuri, Mridula
Published in Journal of organic chemistry (01.10.1983)
Published in Journal of organic chemistry (01.10.1983)
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A novel heterobifunctional linker for formyl to thiol coupling
Heindel, Ned D, Zhao, Huiru, Egolf, Roger A, Chang, Chien Hsing, Schray, Keith J, Emrich, Jacqueline G, McLaughlin, Joanne P, Woo, David V
Published in Bioconjugate chemistry (01.11.1991)
Published in Bioconjugate chemistry (01.11.1991)
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