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Design, Synthesis, and Pharmacological Evaluation of a Novel Series of Pyridopyrazine-1,6-dione γ‑Secretase Modulators
Pettersson, Martin, Johnson, Douglas S, Subramanyam, Chakrapani, Bales, Kelly R, am Ende, Christopher W, Fish, Benjamin A, Green, Michael E, Kauffman, Gregory W, Mullins, Patrick B, Navaratnam, Thayalan, Sakya, Subas M, Stiff, Cory M, Tran, Tuan P, Xie, Longfei, Zhang, Liming, Pustilnik, Leslie R, Vetelino, Beth C, Wood, Kathleen M, Pozdnyakov, Nikolay, Verhoest, Patrick R, O’Donnell, Christopher J
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Pettersson, Martin, Johnson, Douglas S., Subramanyam, Chakrapani, Bales, Kelly R., am Ende, Christopher W., Fish, Benjamin A., Green, Michael E., Kauffman, Gregory W., Lira, Ricardo, Mullins, Patrick B., Navaratnam, Thayalan, Sakya, Subas M., Stiff, Cory M., Tran, Tuan P., Vetelino, Beth C., Xie, Longfei, Zhang, Liming, Pustilnik, Leslie R., Wood, Kathleen M., O’Donnell, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active I3-secretase modulators
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Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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NOVEL BICYCLIC PYRIDINONES
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