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Kaarsholm, Niels C, Lin, Songnian, Yan, Lin, Kelly, Theresa, van Heek, Margaret, Mu, James, Wu, Margaret, Dai, Ge, Cui, Yan, Zhu, Yonghua, Carballo-Jane, Ester, Reddy, Vijay, Zafian, Peter, Huo, Pei, Shi, Shuai, Antochshuk, Valentyn, Ogawa, Aimie, Liu, Franklin, Souza, Sandra C, Seghezzi, Wolfgang, Duffy, Joseph L, Erion, Mark, Nargund, Ravi P, Kelley, David E
Published in Diabetes (New York, N.Y.) (01.02.2018)
Published in Diabetes (New York, N.Y.) (01.02.2018)
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Huang, Chunhui, Palani, Anandan, Yang, Zhiqiang, Deng, Qiaolin, Reddy, Vijay, Nargund, Ravi P., Lin, Songnian, Altezza, Simona, Bianchi, Elisabetta, Orvieto, Federica, Carrington, Paul
Published in ACS medicinal chemistry letters (11.08.2022)
Published in ACS medicinal chemistry letters (11.08.2022)
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Structure Guided Discovery of Novel Pan Metallo-β-Lactamase Inhibitors with Improved Gram-Negative Bacterial Cell Penetration
Dong, Shuzhi, Zhao, Zhiqiang, Tang, Haiqun, Li, Guoqing, Pan, Jianping, Gu, Xin, Jiang, Jinlong, Xiao, Li, Scapin, Giovanna, Hunter, David N., Yang, Dexi, Huang, Yuhua, Bennett, Frank, Yang, Shu-Wei, Mandal, Mihirbaran, Tang, Haifeng, Su, Jing, Tudge, Clare, deJesus, Reynalda Keh, Ding, Fa-Xiang, Lombardo, Matthew, Hicks, Jacqueline D., Fischmann, Thierry, Mirza, Asra, Dayananth, Priya, Painter, Ronald E., Villafania, Artjohn, Garlisi, Charles G., Zhang, Rumin, Mayhood, Todd W., Si, Qian, Li, Nianyu, Amin, Rupesh P., Bhatt, Bhavana, Chen, Feifei, Regan, Christopher P., Regan, Hillary, Lin, Xinjie, Wu, Jin, Leithead, Andrew, Pollack, Scott R., Scott, Jack D., Nargund, Ravi P., Therien, Alex G., Black, Todd, Young, Katherine, Pasternak, Alexander
Published in Journal of medicinal chemistry (14.03.2024)
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Pissarnitski, Dmitri A, Kekec, Ahmet, Yan, Lin, Zhu, Yuping, Feng, Danqing D, Huo, Pei, Madsen-Duggan, Christina, Moyes, Christopher R, Nargund, Ravi P, Kelly, Terri, Zhang, Xiaoping, Carballo-Jane, Ester, Gorski, Judith, Zafian, Peter, Qatanani, Mo, Kaarsholm, Niels, Meng, Fanyu, Jia, Xiujuan, Lee, Keun-Joong, Wang, Weixun, Xu, Sherrie, Hohn, Michael J, Iammarino, Michael J, McCoy, Mark A, Okoh, Grace A, Liang, Yingkai, Hollingsworth, Scott A, Erion, Mark D, Kelley, David E, Garbaccio, Robert M, Zhang, Amy, Mu, James, Lin, Songnian
Published in Journal of medicinal chemistry (14.04.2022)
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Published in Bioorganic & medicinal chemistry letters (15.12.2019)
Published in Bioorganic & medicinal chemistry letters (15.12.2019)
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Yu, Yang, Wu, Zhicai, Shi, Zhi-Cai, He, Shuwen, Lai, Zhong, Cernak, Timothy A., Vachal, Petr, Liu, Min, Liu, Jian, Hong, Qingmei, Jian, Tianying, Guiadeen, Deodial, Krikorian, Arto, Sperbeck, Donald M., Verras, Andreas, Sonatore, Lisa M., Murphy, Beth A., Wiltsie, Judyann, Chung, Christine C., Gorski, Judith N., Liu, Jinqi, Xiao, Jianying, Wolff, Michael, Tong, Sharon X., Madeira, Maria, Karanam, Bindhu V., Shen, Dong-Ming, Balkovec, James M., De Vita, Robert J., Pinto, Shirly, Nargund, Ravi P.
Published in Bioorganic & medicinal chemistry letters (01.06.2019)
Published in Bioorganic & medicinal chemistry letters (01.06.2019)
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Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Erratum. Engineering Glucose Responsiveness Into Insulin. Diabetes 2018;67:299-308
Kaarsholm, Niels C, Lin, Songnian, Yan, Lin, Kelly, Theresa, van Heek, Margaret, Mu, James, Wu, Margaret, Dai, Ge, Cui, Yan, Zhu, Yonghua, Carballo-Jane, Ester, Reddy, Vijay, Zafian, Peter, Huo, Pei, Shi, Shuai, Antochshuk, Valentyn, Ogawa, Aimie, Liu, Franklin, Souza, Sandra C, Seghezzi, Wolfgang, Duffy, Joseph L, Erion, Mark, Nargund, Ravi P, Kelley, David E
Published in Diabetes (New York, N.Y.) (01.05.2018)
Published in Diabetes (New York, N.Y.) (01.05.2018)
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Published in Journal of medicinal chemistry (13.07.2006)
Published in Journal of medicinal chemistry (13.07.2006)
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Published in Bioorganic & medicinal chemistry letters (15.05.2019)
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Published in Proceedings of the National Academy of Sciences - PNAS (20.08.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (20.08.2002)
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Regulation of Energy Homeostasis by Bombesin Receptor Subtype-3: Selective Receptor Agonists for the Treatment of Obesity
Guan, Xiao-Ming, Chen, Howard, Dobbelaar, Peter H., Dong, Yan, Fong, Tung M., Gagen, Karen, Gorski, Judith, He, Shuwen, Howard, Andrew D., Jian, Tianying, Jiang, Michael, Kan, Yanqing, Kelly, Theresa M., Kosinski, Jennifer, Lin, Linus S., Liu, Jian, Marsh, Donald J., Metzger, Joseph M., Miller, Randy, Nargund, Ravi P., Palyha, Oksana, Shearman, Lauren, Shen, Zhu, Stearns, Ralph, Strack, Alison M., Stribling, Sloan, Tang, Yui Sing, Wang, Sheng-Ping, White, Amanda, Yu, Hong, Reitman, Marc L.
Published in Cell metabolism (03.02.2010)
Published in Cell metabolism (03.02.2010)
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A glucose-responsive insulin therapy protects animals against hypoglycemia
Yang, Ruojing, Wu, Margaret, Lin, Songnian, Nargund, Ravi P, Li, Xinghai, Kelly, Theresa, Yan, Lin, Dai, Ge, Qian, Ying, Dallas-Yang, Qing, Fischer, Paul A, Cui, Yan, Shen, Xiaolan, Huo, Pei, Feng, Danqing Dennis, Erion, Mark D, Kelley, David E, Mu, James
Published in JCI insight (11.01.2018)
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Zhu, Cheng, Wang, Liping, Zhu, Yuping, Guo, Zack Zhiqiang, Liu, Ping, Hu, Zhiyong, Szewczyk, Jason W., Kang, Ling, Chicchi, Gary, Ehrhardt, Anka, Woods, Andrea, Seo, Toru, Woods, Morgan, van Heek, Margaret, Dingley, Karen H., Pang, Jianmei, Salituro, Gino M., Powell, Joyce, Terebetski, Jenna L., Hornak, Viktor, Campeau, Louis-Charles, Orr, Robert K., Ujjainwalla, Feroze, Miller, Michael, Stamford, Andrew, Wood, Harold B., Kowalski, Timothy, Nargund, Ravi P., Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (01.03.2017)
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Howard, Andrew D, McAllister, George, Feighner, Scott D, Liu, Qingyun, Nargund, Ravi P, Van der Ploeg, Lex H.T, Patchett, Arthur A
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Guan, Xiao-Ming, Metzger, Joseph M, Yang, Liming, Raustad, Kate A, Wang, Sheng-Ping, Spann, Stephanie K, Kosinski, Jennifer A, Yu, Hong, Shearman, Lauren P, Faidley, Terry D, Palyha, Oksana, Kan, Yanqing, Kelly, Theresa M, Sebhat, Iyassu, Lin, Linus S, Dragovic, Jasminka, Lyons, Kathy A, Craw, Stephanie, Nargund, Ravi P, Marsh, Donald J, Strack, Alison M, Reitman, Marc L
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He, Shuwen, Dobbelaar, Peter H., Guo, Liangqin, Ye, Zhixiong, Liu, Jian, Jian, Tianying, Truong, Quang, Shah, Shrenik K., Du, Wu, Qi, Hongbo, Bakshi, Raman K., Hong, Qingmei, Dellureficio, James D., Sherer, Edward, Pasternak, Alexander, Feng, Zhe, Reibarkh, Mikhail, Lin, Melissa, Samuel, Koppara, Reddy, Vijay B., Mitelman, Stan, Tong, Sharon X., Chicchi, Gary G., Tsao, Kwei-Lan, Trusca, Dorina, Wu, Margaret, Shao, Qing, Trujillo, Maria E., Fernandez, Guillermo, Nelson, Donald, Bunting, Patricia, Kerr, Janet, Fitzgerald, Patrick, Morissette, Pierre, Volksdorf, Sylvia, Eiermann, George J., Li, Cai, Zhang, Bei B., Howard, Andrew D., Zhou, Yun-Ping, Nargund, Ravi P., Hagmann, William K.
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A general approach to substituted 6H-pyrido[2′,3′:5,6] [1,3]oxazino[3,4-a]indole via cyclization from an indoline precursor followed by re-aromatization
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