Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia
Deshpande, Anil M., Bhuniya, Debnath, De, Siddhartha, Dave, Bhavesh, Vyavahare, Vinod P., Kurhade, Santosh H., Kandalkar, Sachin R., Naik, Keshav P., Kobal, Balasaheb S., Kaduskar, Rahul D., Basu, Sujay, Jain, Vaibhav, Patil, Pratima, Chaturvedi Joshi, Sandhya, Bhat, Ganesh, Raje, Amol A., Reddy, Satyanarayana, Gundu, Jayasagar, Madgula, Vamsi, Tambe, Suhas, Shitole, Prasad, Umrani, Dhananjay, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Journal Article
Design and synthesis of novel spirocyclic carboxylic acids as potent and orally bioavailable DGAT1 inhibitors and their biological evaluation
Koul, Summon, Kurhade, Suresh, Bhosale, Sandeep, Naik, Keshav, Salunkhe, Videsh, Ravula, Sudhir, Punde, Prasad, Velayutham, Ravikumar, Tiwari, Atul, Ahl, Daniela, Malkapuram, Srividya, Mudagala, Vamsi, Raje, Amol, Umrani, Dhananjay, Tambe, Suhas, Patil, Poonam, Singh, Umesh, Bhuniya, Debnath, Hariharan, Narayanan, Mookhtiar, Kasim
Published in Bioorganic & medicinal chemistry letters (15.04.2022)
Published in Bioorganic & medicinal chemistry letters (15.04.2022)
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Journal Article
Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
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Journal Article
Discovery and evaluation of 1 H -pyrrolo[2,3- b ]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
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Journal Article
Synthesis and evaluation of 4,5-dihydro-5-methylisoxazolin-5-carboxamide derivatives as VLA-4 antagonists
Soni, Ajay, Rehman, Abdul, Naik, Keshav, Dastidar, Sunanda, Alam, M.S., Ray, Abhijit, Chaira, Tridib, Shah, Vanya, Palle, Venkata P., Cliffe, Ian A., Sattigeri, Viswajanani J.
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Journal Article
Synthesis and biological activity of N-substituted aminocarbonyl-1,3-dioxolanes as VLA-4 antagonists
Rehman, Abdul, Soni, Ajay, Naik, Keshav, Nair, Sreeji, Palle, Venkata P., Dastidar, Sunanda, Ray, Abhijit, Alam, M.S., Salman, Mohammad, Cliffe, Ian A., Sattigeri, Viswajanani
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Journal Article
FUSED BICYCLIC COMPOUNDS, COMPOSITIONS AND APPLICATIONS THEREOF
BHALERAO, Amit, MOOKHTIAR, Kasim, THAKKAR, Mahesh, NAIK, Keshav, JOSHI, Manoj, SHINDE, Shailesh, KULKARNI, Bheemashankar, BHUNIYA, Debnath, MUKIM, Mayur, SHAIKH, Nadim
Year of Publication 27.04.2022
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Year of Publication 27.04.2022
Patent
Fused bicyclic compounds, compositions and applications thereof
Bhuniya, Debnath, Shaikh, Nadim, Joshi, Manoj, Kulkarni, Bheemashankar, Mukim, Mayur, Thakkar, Mahesh, Naik, Keshav, Shinde, Shailesh, Bhalerao, Amit, Mookhtiar, Kasim
Year of Publication 24.08.2021
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Year of Publication 24.08.2021
Patent