Direct catalytic asymmetric aldol reactions of aldehydes
Bogevig, A, Kumaragurubaran, N, Jorgensen, KA
Published in Chemical communications (Cambridge, England) (21.03.2002)
Published in Chemical communications (Cambridge, England) (21.03.2002)
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Journal Article
Memapsin 2 (beta-secretase) inhibitors: drug development
Ghosh, Arun K, Kumaragurubaran, Nagaswamy, Hong, Ling, Koelsh, Gerald, Tang, Jordan
Published in Current Alzheimer research (01.04.2008)
Published in Current Alzheimer research (01.04.2008)
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Journal Article
Applications of Baylis–Hillman chemistry: enantioselective synthesis of (−)-methyl 3-aryl-2-methylene-3-(prop-2-yn-1-yloxy)propanoates via chiral leaving group strategy
Basavaiah, Deevi, Kumaragurubaran, Nagaswamy, Sharada, Duddu S, Reddy, Ravi Mallikarjuna
Published in Tetrahedron (17.09.2001)
Published in Tetrahedron (17.09.2001)
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Journal Article
Direct Organo-Catalytic Asymmetric α-Amination of Aldehydes-A Simple Approach to Optically Active α-Amino Aldehydes, α-Amino Alcohols, and α-Amino Acids
Bøgevig, Anders, Juhl, Karsten, Kumaragurubaran, Nagaswamy, Zhuang, Wei, Jørgensen, Karl Anker
Published in Angewandte Chemie (International ed.) (17.05.2002)
Published in Angewandte Chemie (International ed.) (17.05.2002)
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Journal Article
Direct l-Proline-Catalyzed Asymmetric α-Amination of Ketones
Kumaragurubaran, Nagaswamy, Juhl, Karsten, Zhuang, Wei, Bøgevig, Anders, Jørgensen, Karl Anker
Published in Journal of the American Chemical Society (05.06.2002)
Published in Journal of the American Chemical Society (05.06.2002)
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Journal Article
Design, synthesis, X-ray studies, and biological evaluation of novel BACE1 inhibitors with bicyclic isoxazoline carboxamides as the P3 ligand
Ghosh, Arun K., Ghosh, Koena, Brindisi, Margherita, Lendy, Emma K., Yen, Yu-Chen, Kumaragurubaran, Nagaswamy, Huang, Xiangping, Tang, Jordan, Mesecar, Andrew D.
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
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Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Journal Article
Abstract 2643: Discovery and characterization of a selective TrkA inhibitor for the treatment of TrkA-driven cancers
Tirunagaru, Vijaya G., Nagaswamy, Kumaragurubaran, Mitra, Sayan, Maddi, Srinivas, Adluri, Ram Sudheer, Joshi, Hemant, Gupta, Jang B.
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Design, synthesis, X-ray studies, and biological evaluation of novel BACE1 inhibitors with bicyclic isoxazoline carboxamides as the P3 ligand
Ghosh, Arun K., Ghosh, Koena, Brindisi, Margherita, Lendy, Emma K., Yen, Yu-Chen, Kumaragurubaran, Nagaswamy, Huang, Xiangping, Tang, Jordan, Mesecar, Andrew D.
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
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Journal Article
Design, synthesis, and X-ray structural studies of BACE-1 inhibitors containing substituted 2-oxopiperazines as P1′-P2′ ligands
Ghosh, Arun K., Brindisi, Margherita, Yen, Yu-Chen, Cárdenas, Emilio L., Ella-Menye, Jean-Rene, Kumaragurubaran, Nagaswamy, Huang, Xiangping, Tang, Jordan, Mesecar, Andrew D.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
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Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Journal Article
Design, synthesis, and X-ray structural studies of BACE-1 inhibitors containing substituted 2-oxopiperazines as P1′-P2′ ligands
Ghosh, Arun K., Brindisi, Margherita, Yen, Yu-Chen, Cárdenas, Emilio L., Ella-Menye, Jean-Rene, Kumaragurubaran, Nagaswamy, Huang, Xiangping, Tang, Jordan, Mesecar, Andrew D.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
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Journal Article
Design, Synthesis, and X-ray Structure of Potent Memapsin 2 (β-Secretase) Inhibitors with Isophthalamide Derivatives as the P2 -P3-Ligands
Ghosh, Arun K, Kumaragurubaran, Nagaswamy, Hong, Lin, Kulkarni, Sarang S, Xu, Xiaoming, Chang, Wanpin, Weerasena, Vajira, Turner, Robert, Koelsch, Gerald, Bilcer, Geoffrey, Tang, Jordan
Published in Journal of medicinal chemistry (17.05.2007)
Published in Journal of medicinal chemistry (17.05.2007)
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Journal Article
Bis-Tetrahydrofuran: a Privileged Ligand for Darunavir and a New Generation of HIV Protease Inhibitors That Combat Drug Resistance
Ghosh, Arun K., Ramu Sridhar, Perali, Kumaragurubaran, Nagaswamy, Koh, Yasuhiro, Weber, Irene T., Mitsuya, Hiroaki
Published in ChemMedChem (11.09.2006)
Published in ChemMedChem (11.09.2006)
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Journal Article
Design, Synthesis and X-ray Structure of Protein−Ligand Complexes: Important Insight into Selectivity of Memapsin 2 (β-Secretase) Inhibitors
Ghosh, Arun K, Kumaragurubaran, Nagaswamy, Hong, Lin, Lei, Hui, Hussain, Khaja Azhar, Liu, Chun-Feng, Devasamudram, Thippeswamy, Weerasena, Vajira, Turner, Robert, Koelsch, Gerald, Bilcer, Geoffrey, Tang, Jordan
Published in Journal of the American Chemical Society (26.04.2006)
Published in Journal of the American Chemical Society (26.04.2006)
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Journal Article
Potent memapsin 2 (β-secretase) inhibitors: Design, synthesis, protein-ligand X-ray structure, and in vivo evaluation
Ghosh, Arun K., Kumaragurubaran, Nagaswamy, Hong, Lin, Kulkarni, Sarang, Xu, Xiaoming, Miller, Heather B., Srinivasa Reddy, Dandepally, Weerasena, Vajira, Turner, Robert, Chang, Wanpin, Koelsch, Gerald, Tang, Jordan
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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