A novel GIP analogue, ZP4165, enhances glucagon‐like peptide‐1‐induced body weight loss and improves glycaemic control in rodents
Nørregaard, Pia K., Deryabina, Maria A., Tofteng Shelton, Pernille, Fog, Jacob U., Daugaard, Jens R., Eriksson, Per‐Olof, Larsen, Lone F., Jessen, Lene
Published in Diabetes, obesity & metabolism (01.01.2018)
Published in Diabetes, obesity & metabolism (01.01.2018)
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Journal Article
Optimizing and characterizing 4-methyl substituted pyrazol-3-carboxamides leading to the peripheral cannabinoid 1 receptor inverse agonist TM38837
Högberg, Thomas, Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K, Little, Paul B, Cooper, Martin
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
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Journal Article
6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: Structure–activity exploration of eastern and western parts
Ulven, Trond, Little, Paul Brian, Receveur, Jean-Marie, Frimurer, Thomas M., Rist, Øystein, Nørregaard, Pia K., Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Journal Article
Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood–brain-barrier
Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K., Cooper, Martin, Bjurling, Emelie, Nielsen, Peter Aadal, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
6-Acylamino-2-aminoquinolines as Potent Melanin-Concentrating Hormone 1 Receptor Antagonists. Identification, Structure−Activity Relationship, and Investigation of Binding Mode
Ulven, Trond, Frimurer, Thomas M, Receveur, Jean-Marie, Little, Paul Brian, Rist, Øystein, Nørregaard, Pia K, Högberg, Thomas
Published in Journal of medicinal chemistry (08.09.2005)
Published in Journal of medicinal chemistry (08.09.2005)
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Journal Article
Exploring SAR features in diverse library of 4-cyanomethyl-pyrazole-3-carboxamides suitable for further elaborations as CB1 antagonists
Cooper, Martin, Receveur, Jean-Marie, Bjurling, Emelie, Nørregaard, Pia K., Nielsen, Peter Aadal, Sköld, Niklas, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
4-Acylamino- and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists
RECEVEUR, Jean-Marie, BJURLING, Emelie, ULVEN, Trond, LITTLE, Paul Brian, NØRREGAARD, Pia K, HÖGBERG, Thomas
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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Journal Article
A highly conserved glycine within linker I and the extreme C terminus of G protein alpha subunits interact cooperatively in switching G protein-coupled receptor-to-effector specificity
Kostenis, Evi, Martini, Lene, Ellis, James, Waldhoer, Maria, Heydorn, Arne, Rosenkilde, Mette M, Norregaard, Pia K, Jorgensen, Rasmus, Whistler, Jennifer L, Milligan, Graeme
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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Journal Article
A novel GIP analogue, ZP 4165, enhances glucagon‐like peptide‐1‐induced body weight loss and improves glycaemic control in rodents
Nørregaard, Pia K., Deryabina, Maria A., Tofteng Shelton, Pernille, Fog, Jacob U., Daugaard, Jens R., Eriksson, Per‐Olof, Larsen, Lone F., Jessen, Lene
Published in Diabetes, obesity & metabolism (01.01.2018)
Published in Diabetes, obesity & metabolism (01.01.2018)
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Journal Article
A Highly Conserved Glycine within Linker I and the Extreme C Terminus of G Protein α Subunits Interact Cooperatively in Switching G Protein-Coupled Receptor-to-Effector Specificity
Evi Kostenis, Lene Martini, James Ellis, Maria Waldhoer, Arne Heydorn, Mette M. Rosenkilde, Pia K. Norregaard, Rasmus Jorgensen, Jennifer L. Whistler, Graeme Milligan
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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Journal Article
Quinoline compounds for use in mch receptor related disorders
NORREGAARD PIA K, LITTLE PAUL B, ULVEN TROND, HOGBERG THOMAS, FRIMURER THOMAS M, RECEVEUR JEAN-MARIE
Year of Publication 25.05.2006
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Year of Publication 25.05.2006
Patent
Novel methoxybenzamibe compounds for use in mch receptor related disorders
LITTLE PAUL B, NORREGAARD PIA K, BJURLING EMELIE, HOGBERG THOMAS, ULVEN TROND, ELLING CHRISTIAN E, RECEVEUR JEAN-MARIE
Year of Publication 19.10.2006
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Year of Publication 19.10.2006
Patent