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Published in Bioorganic & medicinal chemistry letters (21.02.2000)
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Characterization of the allosteric binding pocket of human liver fructose‐1,6‐bisphosphatase by protein crystallography and inhibitor activity studies
Iversen, L. F., Brzozowski, M., Hastrup, S., Hubbard, R., Kastrup, J. S., Larsen, I. K., Nærum, L., Nørskov‐Lauridsen, L., Rasmussen, P. B., Thim, L., Wiberg, F. C., Lundgren, K.
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Virtual Screening for Submicromolar Leads of tRNA-guanine Transglycosylase Based on a New Unexpected Binding Mode Detected by Crystal Structure Analysis
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Published in Journal of medicinal chemistry (27.03.2003)
Published in Journal of medicinal chemistry (27.03.2003)
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Novel semicarbazide-derived inhibitors of human dipeptidyl peptidase I (hDPPI)
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Published in Bioorganic & medicinal chemistry (15.07.2005)
Published in Bioorganic & medicinal chemistry (15.07.2005)
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Synthesis and estrogen receptor binding affinities of novel pyrrolo[2,1,5- cd]indolizine derivatives
Jørgensen, Anker Steen, Jacobsen, Poul, Christiansen, Lise Brown, Bury, Paul S., Kanstrup, Anders, Thorpe, Susan M., Nærum, Lars, Wassermann, Karsten
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents
Knutsen, Lars J. S, Andersen, Knud Erik, Lau, Jesper, Lundt, Behrend F, Henry, Rodger F, Morton, Howard E, Nærum, Lars, Petersen, Hans, Stephensen, Henrik, Suzdak, Peter D, Swedberg, Michael D. B, Thomsen, Christian, Sørensen, Per O
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Published in Journal of medicinal chemistry (09.09.1999)
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Synthesis and pharmacological evaluation of novel cis-3,4-Diaryl-hydroxychromanes as high affinity partial agonists for the estrogen receptor
Bury, Paul S., Christiansen, Lise B., Jacobsen, Poul, Jørgensen, Anker S., Kanstrup, Anders, Nærum, Lars, Bain, Steven, Fledelius, Christian, Gissel, Birgitte, Hansen, Birgit S., Korsgaard, Niels, Thorpe, Susan M., Wassermann, Karsten
Published in Bioorganic & medicinal chemistry (2002)
Published in Bioorganic & medicinal chemistry (2002)
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Efficient Generation, Storage, and Manipulation of Fully Flexible Pharmacophore Multiplets and Their Use in 3-D Similarity Searching
Abrahamian, Edmond, Fox, Peter C, Nærum, Lars, Christensen, Inge Thøger, Thøgersen, Henning, Clark, Robert D
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Published in Journal of Chemical Information and Computer Sciences (01.03.2003)
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Synthesis and biological evaluation of novel thio-substituted chromanes as high-affinity partial agonists for the estrogen receptor
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Published in Bioorganic & medicinal chemistry letters (07.01.2002)
Published in Bioorganic & medicinal chemistry letters (07.01.2002)
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The preferential dopamine D 3 receptor agonist cis-8-OH-PBZI induces limbic Fos expression in rat brain
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Published in European journal of pharmacology (27.11.1997)
Published in European journal of pharmacology (27.11.1997)
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The preferential dopamine D3 receptor agonist cis-8-OH-PBZI induces limbic Fos expression in rat brain
SCHEIDELER, M. A, MARTIN, J, CRUSE, S. F, FINK-JENSEN, A, HOHLWEG, R, RASMUSSEN, J. S, NAERUM, L, LUDVIGSEN, T. S, LARSEN, P. J, KORSGAARD, N, CRIDER, A. M, GHOSH, D
Published in European journal of pharmacology (27.11.1997)
Published in European journal of pharmacology (27.11.1997)
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