Design, Synthesis, and Investigation of Novel Nitric Oxide (NO)-Releasing Aromatic Aldehydes as Drug Candidates for the Treatment of Sickle Cell Disease
Huang, Boshi, Ghatge, Mohini S., Donkor, Akua K., Musayev, Faik N., Deshpande, Tanvi M., Al-Awadh, Mohammed, Alhashimi, Rana T., Zhu, Hongmei, Omar, Abdelsattar M., Telen, Marilyn J., Zhang, Yan, McMahon, Tim J., Abdulmalik, Osheiza, Safo, Martin K.
Published in Molecules (Basel, Switzerland) (01.10.2022)
Published in Molecules (Basel, Switzerland) (01.10.2022)
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Journal Article
Characterization of the Staphylococcus aureus rRNA Methyltransferase Encoded by orfX, the Gene Containing the Staphylococcal Chromosome Cassette mec (SCCmec) Insertion Site
Boundy, Sam, Safo, Martin K., Wang, Lei, Musayev, Faik N., O'Farrell, Heather C., Rife, Jason P., Archer, Gordon L.
Published in The Journal of biological chemistry (04.01.2013)
Published in The Journal of biological chemistry (04.01.2013)
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Journal Article
Crystal structures of influenza A virus matrix protein M1: variations on a theme
Safo, Martin K, Musayev, Faik N, Mosier, Philip D, Zhou, Qibing, Xie, Hang, Desai, Umesh R
Published in PloS one (08.10.2014)
Published in PloS one (08.10.2014)
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Journal Article
A Triazole Disulfide Compound Increases the Affinity of Hemoglobin for Oxygen and Reduces the Sickling of Human Sickle Cells
Nakagawa, Akito, Ferrari, Michele, Schleifer, Grigorij, Cooper, Marissa K, Liu, Chen, Yu, Binglan, Berra, Lorenzo, Klings, Elizabeth S, Safo, Ronni S, Chen, Qiukan, Musayev, Faik N, Safo, Martin K, Abdulmalik, Osheiza, Bloch, Donald B, Zapol, Warren M
Published in Molecular pharmaceutics (07.05.2018)
Published in Molecular pharmaceutics (07.05.2018)
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Journal Article
Design, Synthesis, and Antisickling Investigation of a Nitric Oxide-Releasing Prodrug of 5HMF for the Treatment of Sickle Cell Disease
Alhashimi, Rana T, Ghatge, Mohini S, Donkor, Akua K, Deshpande, Tanvi M, Anabaraonye, Nancy, Alramadhani, Dina, Danso-Danquah, Richmond, Huang, Boshi, Zhang, Yan, Musayev, Faik N, Abdulmalik, Osheiza, Safo, Martin K
Published in Biomolecules (Basel, Switzerland) (12.05.2022)
Published in Biomolecules (Basel, Switzerland) (12.05.2022)
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Journal Article
Crystal structures of human pyridoxal kinase in complex with the neurotoxins, ginkgotoxin and theophylline: insights into pyridoxal kinase inhibition
Gandhi, Amit K, Desai, Jigar V, Ghatge, Mohini S, di Salvo, Martino L, Di Biase, Stefano, Danso-Danquah, Richmond, Musayev, Faik N, Contestabile, Roberto, Schirch, Verne, Safo, Martin K
Published in PloS one (18.07.2012)
Published in PloS one (18.07.2012)
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Journal Article
Molecular Basis of Reduced Pyridoxine 5′-Phosphate Oxidase Catalytic Activity in Neonatal Epileptic Encephalopathy Disorder
Musayev, Faik N., Di Salvo, Martino L., Saavedra, Mario A., Contestabile, Roberto, Ghatge, Mohini S., Haynes, Alexina, Schirch, Verne, Safo, Martin K.
Published in The Journal of biological chemistry (06.11.2009)
Published in The Journal of biological chemistry (06.11.2009)
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Journal Article
Maintaining pH-dependent conformational flexibility of M1 is critical for efficient influenza A virus replication
Chiang, Meng-Jung, Musayev, Faik N, Kosikova, Martina, Lin, Zhengshi, Gao, Yamei, Mosier, Philip D, Althufairi, Bashayer, Ye, Zhiping, Zhou, Qibing, Desai, Umesh R, Xie, Hang, Safo, Martin K
Published in Emerging microbes & infections (2017)
Published in Emerging microbes & infections (2017)
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Journal Article
Kinetic and structural studies of the role of the active site residue Asp235 of human pyridoxal kinase
Gandhi, Amit K., Ghatge, Mohini S., Musayev, Faik N., Sease, Aaron, Aboagye, Samuel O., di Salvo, Martino L., Schirch, Verne, Safo, Martin K.
Published in Biochemical and biophysical research communications (27.03.2009)
Published in Biochemical and biophysical research communications (27.03.2009)
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Journal Article
Crystal Structure of Pyridoxal Kinase from the Escherichia coli pdxK Gene: Implications for the Classification of Pyridoxal Kinases
SAFO, Martin K, MUSAYEV, Faik N, DI SALVO, Martino L, HUNT, Sharyn, CLAUDE, Jean-Baptiste, SCHIRCH, Verne
Published in Journal of Bacteriology (01.06.2006)
Published in Journal of Bacteriology (01.06.2006)
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Journal Article
Structural Basis for the Potent Antisickling Effect of a Novel Class of Five-Membered Heterocyclic Aldehydic Compounds
Safo, Martin K, Abdulmalik, Osheiza, Danso-Danquah, Richmond, Burnett, James C, Nokuri, Samuel, Joshi, Gajanan S, Musayev, Faik N, Asakura, Toshio, Abraham, Donald J
Published in Journal of medicinal chemistry (09.09.2004)
Published in Journal of medicinal chemistry (09.09.2004)
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Journal Article
A novel and unique ATP hydrolysis to AMP by a human Hsp70 Binding immunoglobin protein (BiP)
Li, Hongtao, Musayev, Faik N., Yang, Jiao, Su, Jiayue, Liu, Qingdai, Wang, Wei, Fang, Xianjun, Zhou, Lei, Liu, Qinglian
Published in Protein science (01.04.2022)
Published in Protein science (01.04.2022)
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Journal Article
The Cryo-EM structure of AAV2 Rep68 in complex with ssDNA reveals a malleable AAA+ machine that can switch between oligomeric states
Santosh, Vishaka, Musayev, Faik N, Jaiswal, Rahul, Zárate-Pérez, Francisco, Vandewinkel, Bram, Dierckx, Caroline, Endicott, Molly, Sharifi, Kamyar, Dryden, Kelly, Henckaerts, Els, Escalante, Carlos R
Published in Nucleic acids research (16.12.2020)
Published in Nucleic acids research (16.12.2020)
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Journal Article
Crystal Structures of the BlaI Repressor from Staphylococcus aureus and Its Complex with DNA: Insights into Transcriptional Regulation of the bla and mec Operons
SAFO, Martin K, QIXUN ZHAO, KO, Tzu-Ping, MUSAYEV, Faik N, ROBINSON, Howard, SCARSDALE, Neel, WANG, Andrew H.-J, ARCHER, Gordon L
Published in Journal of Bacteriology (01.03.2005)
Published in Journal of Bacteriology (01.03.2005)
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Journal Article
Functional and structural properties of pyridoxal reductase (PdxI) from Escherichia coli: a pivotal enzyme in the vitamin B6 salvage pathway
Tramonti, Angela, Donkor, Akua K., Parroni, Alessia, Musayev, Faik N., Barile, Anna, Ghatge, Mohini S., Graziani, Claudio, Alkhairi, Mona, AlAwadh, Mohammed, Salvo, Martino Luigi, Safo, Martin K., Contestabile, Roberto
Published in The FEBS journal (01.12.2023)
Published in The FEBS journal (01.12.2023)
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Journal Article
Exploration of Structure–Activity Relationship of Aromatic Aldehydes Bearing Pyridinylmethoxy-Methyl Esters as Novel Antisickling Agents
Pagare, Piyusha P, Ghatge, Mohini S, Chen, Qiukan, Musayev, Faik N, Venitz, Jurgen, Abdulmalik, Osheiza, Zhang, Yan, Safo, Martin K
Published in Journal of medicinal chemistry (10.12.2020)
Published in Journal of medicinal chemistry (10.12.2020)
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Journal Article
Crystal Structure of the PdxY Protein from Escherichia coli
SAFE, Martin K, MUSAYEV, Faik N, HUNT, Sharyn, DI SALVO, Martino L, SCARSDALE, Neel, SCHIRCH, Verne
Published in Journal of Bacteriology (01.12.2004)
Published in Journal of Bacteriology (01.12.2004)
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Journal Article
Characterization of the Escherichia coli pyridoxal 5′‐phosphate homeostasis protein (YggS): Role of lysine residues in PLP binding and protein stability
Tramonti, Angela, Ghatge, Mohini S., Babor, Jill T., Musayev, Faik N., di Salvo, Martino Luigi, Barile, Anna, Colotti, Gianni, Giorgi, Alessandra, Paredes, Steven D., Donkor, Akua K., Al Mughram, Mohammed H., de Crécy‐Lagard, Valérie, Safo, Martin K., Contestabile, Roberto
Published in Protein science (01.11.2022)
Published in Protein science (01.11.2022)
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Journal Article
VZHE-039, a novel antisickling agent that prevents erythrocyte sickling under both hypoxic and anoxic conditions
Abdulmalik, Osheiza, Pagare, Piyusha P, Huang, Boshi, Xu, Guoyan G, Ghatge, Mohini S, Xu, Xiaomeng, Chen, Qiukan, Anabaraonye, Nancy, Musayev, Faik N, Omar, Abdelsattar M, Venitz, Jürgen, Zhang, Yan, Safo, Martin K
Published in Scientific reports (20.11.2020)
Published in Scientific reports (20.11.2020)
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Journal Article
Rational modification of vanillin derivatives to stereospecifically destabilize sickle hemoglobin polymer formation
Deshpande, Tanvi M, Pagare, Piyusha P, Ghatge, Mohini S, Chen, Qiukan, Musayev, Faik N, Venitz, Jurgen, Zhang, Yan, Abdulmalik, Osheiza, Safo, Martin K
Published in Acta crystallographica. Section D, Biological crystallography. (01.10.2018)
Published in Acta crystallographica. Section D, Biological crystallography. (01.10.2018)
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