In silico discovery of small-molecule Ras inhibitors that display antitumor activity by blocking the Ras–effector interaction
Shima, Fumi, Yoshikawa, Yoko, Ye, Min, Araki, Mitsugu, Matsumoto, Shigeyuki, Liao, Jingling, Hu, Lizhi, Sugimoto, Takeshi, Ijiri, Yuichi, Takeda, Azusa, Nishiyama, Yuko, Sato, Chie, Muraoka, Shin, Tamura, Atsuo, Osoda, Tsutomu, Tsuda, Ken-ichiro, Miyakawa, Tomoya, Fukunishi, Hiroaki, Shimada, Jiro, Kumasaka, Takashi, Yamamoto, Masaki, Kataoka, Tohru
Published in Proceedings of the National Academy of Sciences - PNAS (14.05.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (14.05.2013)
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Journal Article
Solution Structure of the State 1 Conformer of GTP-bound H-Ras Protein and Distinct Dynamic Properties between the State 1 and State 2 Conformers
Araki, Mitsugu, Shima, Fumi, Yoshikawa, Yoko, Muraoka, Shin, Ijiri, Yuichi, Nagahara, Yuka, Shirono, Tomoya, Kataoka, Tohru, Tamura, Atsuo
Published in The Journal of biological chemistry (11.11.2011)
Published in The Journal of biological chemistry (11.11.2011)
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Journal Article
Structural Basis for Conformational Dynamics of GTP-bound Ras Protein
Shima, Fumi, Ijiri, Yuichi, Muraoka, Shin, Liao, Jingling, Ye, Min, Araki, Mitsugu, Matsumoto, Kousuke, Yamamoto, Naoki, Sugimoto, Takeshi, Yoshikawa, Yoko, Kumasaka, Takashi, Yamamoto, Masaki, Tamura, Atsuo, Kataoka, Tohru
Published in The Journal of biological chemistry (16.07.2010)
Published in The Journal of biological chemistry (16.07.2010)
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Journal Article
Crystal structures of the state 1 conformations of the GTP-bound H-Ras protein and its oncogenic G12V and Q61L mutants
Muraoka, Shin, Shima, Fumi, Araki, Mitsugu, Inoue, Tomoko, Yoshimoto, Akiko, Ijiri, Yuichi, Seki, Nobuaki, Tamura, Atsuo, Kumasaka, Takashi, Yamamoto, Masaki, Kataoka, Tohru
Published in FEBS letters (12.06.2012)
Published in FEBS letters (12.06.2012)
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Journal Article
Crystal Structure of a Full-length LysR-type Transcriptional Regulator, CbnR: Unusual Combination of Two Subunit Forms and Molecular Bases for Causing and Changing DNA Bend
Muraoka, Shin, Okumura, Rumi, Ogawa, Naoto, Nonaka, Takamasa, Miyashita, Kiyotaka, Senda, Toshiya
Published in Journal of molecular biology (02.05.2003)
Published in Journal of molecular biology (02.05.2003)
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Journal Article
Structure Basis for Antitumor Effect of Aplyronine A
Hirata, Kunio, Muraoka, Shin, Suenaga, Kiyotake, Kuroda, Takeshi, Kato, Kenichi, Tanaka, Hiroshi, Yamamoto, Masaki, Takata, Masaki, Yamada, Kiyoyuki, Kigoshi, Hideo
Published in Journal of molecular biology (03.03.2006)
Published in Journal of molecular biology (03.03.2006)
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Journal Article
Biochemical characterization of missense mutations in the Arf/Arl-family small GTPase Arl6 causing Bardet–Biedl syndrome
Kobayashi, Tetsuo, Hori, Yuji, Ueda, Nami, Kajiho, Hiroaki, Muraoka, Shin, Shima, Fumi, Kataoka, Tohru, Kontani, Kenji, Katada, Toshiaki
Published in Biochemical and biophysical research communications (10.04.2009)
Published in Biochemical and biophysical research communications (10.04.2009)
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Journal Article
Crystal Structure of M-Ras Reveals a GTP-bound “Off” State Conformation of Ras Family Small GTPases
Ye, Min, Shima, Fumi, Muraoka, Shin, Liao, Jingling, Okamoto, Hidetsugu, Yamamoto, Masaki, Tamura, Atsuo, Yagi, Naoto, Ueki, Tatzuo, Kataoka, Tohru
Published in The Journal of biological chemistry (02.09.2005)
Published in The Journal of biological chemistry (02.09.2005)
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Journal Article
Prenatal nicotine exposure affects the development of the central serotonergic system as well as the dopaminergic system in rat offspring: involvement of route of drug administrations
Muneoka, Katsumasa, Ogawa, Tetsuo, Kamei, Kenji, Muraoka, Shin-ichiro, Tomiyoshi, Rika, Mimura, Yuichi, Kato, Hitomi, Suzuki, Minoru R, Takigawa, Morikuni
Published in Brain research. Developmental brain research (18.08.1997)
Published in Brain research. Developmental brain research (18.08.1997)
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Journal Article
CYP52 (cytochrome P450alk) multigene family in Candida maltosa: identification and characterization of eight members
Ohkuma, M, Muraoka, S, Tanimoto, T, Fujii, M, Ohta, A, Takagi, M
Published in DNA and cell biology (01.02.1995)
Published in DNA and cell biology (01.02.1995)
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Journal Article
Purification and crystallization of a LysR-type transcriptional regulator CBNR from Ralstonia eutropha NH9
Muraoka, Shin, Okumura, Rumi, Uragami, Yoshitaka, Nonaka, Takamasa, Ogawa, Naoto, Miyashita, Kiyotaka, Senda, Toshiya
Published in Protein and peptide letters (01.06.2003)
Published in Protein and peptide letters (01.06.2003)
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Journal Article
Electrolytes in erythrocytes of patients with depressive disorders
KAMEI, KENJI, TABATA, OSAMU, MUNEOKA, KATSUMASA, MURAOKA, SHIN‐ICHIRO, TOMIYOSHI, RIKA, TAKIGAWA, MORIKUNI
Published in Psychiatry and clinical neurosciences (01.10.1998)
Published in Psychiatry and clinical neurosciences (01.10.1998)
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Journal Article
Conference Proceeding
Homologous desensitization of serotonin 5-HT2 receptor-stimulated intracellular calcium mobilization in C6BU-1 glioma cells via a mechanism involving a calmodulin pathway
Kagaya, A, Mikuni, M, Muraoka, S, Saitoh, K, Ogawa, T, Shinno, H, Yamawaki, S, Takahashi, K
Published in Journal of neurochemistry (01.09.1993)
Published in Journal of neurochemistry (01.09.1993)
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Journal Article
Peroxisome Proliferators Activate Cytochrome P450 Genes in an Alkane-Assimilating Yeast,Candida maltosa
Ohtomo, Ryo, Kobayashi, Keisuke, Muraoka, Shin-ichiro, Ohkuma, Moriya, Ohta, Akinori, Takagi, Masamichi
Published in Biochemical and biophysical research communications (24.05.1996)
Published in Biochemical and biophysical research communications (24.05.1996)
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Journal Article
Critical Roles of Interactions among Switch I-preceding Residues and between Switch II and Its Neighboring α-Helix in Conformational Dynamics of the GTP-bound Ras Family Small GTPases
Matsumoto, Kousuke, Shima, Fumi, Muraoka, Shin, Araki, Mitsugu, Hu, Lizhi, Ijiri, Yuichi, Hirai, Rina, Liao, Jingling, Yoshioka, Takashi, Kumasaka, Takashi, Yamamoto, Masaki, Tamura, Atsuo, Kataoka, Tohru
Published in The Journal of biological chemistry (29.04.2011)
Published in The Journal of biological chemistry (29.04.2011)
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Journal Article
Cloning of the C-URA3 gene and construction of a triple auxotroph (his5, ade1, ura3) as a useful host for the genetic engineering of Candida maltosa
Ohkuma, M. (Tokyo Univ. (Japan). Dept. of Agricultural Chemistry), Muraoka, S, Hwang, C.W, Ohta, A, Takagi, M
Published in Current genetics (01.03.1993)
Published in Current genetics (01.03.1993)
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Journal Article
Effects of methamphetamine on spinophilin gene expression in the neocortex of the rat
Nishikawa, Toru, Muraoka, Shin-ichiro, Kajii, Yasushi, Toda, Shigenobu, Numachi, Yotaro, Yamamoto, Naoki
Published in Neuroscience research (01.09.2011)
Published in Neuroscience research (01.09.2011)
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Journal Article