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Published in Chembiochem : a European journal of chemical biology (02.11.2017)
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Molecular mechanism of positive allosteric modulation of the metabotropic glutamate receptor 2 by JNJ‐46281222
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Published in British journal of pharmacology (01.02.2016)
Published in British journal of pharmacology (01.02.2016)
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A New Class of Fluorinated A 2A Adenosine Receptor Agonist with Application to Last-Step Enzymatic [ 18 F]Fluorination for PET Imaging
Lowe, Phillip T, Dall'Angelo, Sergio, Mulder-Krieger, Thea, IJzerman, Adriaan P, Zanda, Matteo, O'Hagan, David
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Published in Chembiochem : a European journal of chemical biology (02.11.2017)
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Predicting Binding Affinities for GPCR Ligands Using Free-Energy Perturbation
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Published in ACS omega (31.08.2016)
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Substructure‐Based Virtual Screening for Adenosine A 2A Receptor Ligands
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Published in ChemMedChem (09.12.2011)
Published in ChemMedChem (09.12.2011)
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Allosteric modulation, thermodynamics and binding to wild‐type and mutant (T277A) adenosine A 1 receptors of LUF5831, a novel nonadenosine‐like agonist
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Published in British journal of pharmacology (29.01.2009)
Published in British journal of pharmacology (29.01.2009)
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Substructure-Based Virtual Screening for Adenosine A2A Receptor Ligands
van der Horst, Eelke, van der Pijl, Rianne, Mulder-Krieger, Thea, Bender, Andreas, IJzerman, Adriaan P.
Published in ChemMedChem (09.12.2011)
Published in ChemMedChem (09.12.2011)
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Allosteric modulation, thermodynamics and binding to wild‐type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine‐like agonist
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Published in British journal of pharmacology (01.03.2006)
Published in British journal of pharmacology (01.03.2006)
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A New Class of Fluorinated A(2A) Adenosine Receptor Agonist with Application to Last-Step Enzymatic [F-18]Fluorination for PET Imaging
Lowe, Phillip T., Dall'Angelo, Sergio, Mulder-Krieger, Thea, IJzerman, Adriaan P., Zanda, Matteo, O'Hagan, David
Published in Chembiochem : a European journal of chemical biology (02.11.2017)
Published in Chembiochem : a European journal of chemical biology (02.11.2017)
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Synthesis and evaluation of N-substituted 2-amino-4,5-diarylpyrimidines as selective adenosine A(1) receptor antagonists
Alachouzos, Georgios, Lenselink, Eelke B., Mulder-Krieger, Thea, de Vries, Henk, IJzerman, Adriaan P., Louvel, Julien
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Structure-kinetics relationships of Capadenoson derivatives as adenosine A(1) receptor agonists
Louvel, Julien, Guo, Dong, Soethoudt, Marjolein, Mocking, Tamara A. M., Lenselink, Eelke B., Mulder-Krieger, Thea, Heitman, Laura H., Ijzerman, Adriaan P.
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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2-amino-6-furan-2-yl-4-substituted nicotinonitriles as A(2A) adenosine receptor antagonists
Mantri, Monica, de Graaf, Olivier, van Veldhoven, Jacobus, Goblyos, Aniko, von Frijtag, Jacobien K., Kuenzel, Drabbe, Mulder-Krieger, Thea, Link, Regina, de Vries, Henk, Beukers, Margot W., Brussee, Johannes, Ijzerman, Adriaan P.
Published in Journal of medicinal chemistry (14.08.2008)
Published in Journal of medicinal chemistry (14.08.2008)
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Discovery and Kinetic Profiling of 7‑Aryl-1,2,4-triazolo[4,3‑a]pyridines: Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 2
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Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonists
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Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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2-Amino-6-furan-2-yl-4-substituted Nicotinonitriles as A2A Adenosine Receptor Antagonists
Mantri, Monica, de Graaf, Olivier, van Veldhoven, Jacobus, Göblyös, Anikó, von Frijtag Drabbe Künzel, Jacobien K, Mulder-Krieger, Thea, Link, Regina, de Vries, Henk, Beukers, Margot W, Brussee, Johannes, IJzerman, Adriaan P
Published in Journal of medicinal chemistry (14.08.2008)
Published in Journal of medicinal chemistry (14.08.2008)
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Synthesis and evaluation of N-substituted 2-amino-4,5-diarylpyrimidines as selective adenosine A1 receptor antagonists
Alachouzos, Georgios, Lenselink, Eelke B., Mulder-Krieger, Thea, de Vries, Henk, IJzerman, Adriaan P., Louvel, Julien
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A(3) Receptor
Heitman, Laura H., Goblyos, Aniko, Zweemer, Annelien M., Bakker, Renee, Mulder-Krieger, Thea, van Veldhover, Jacobus P. D., de Vries, Henk, Brussee, Johannes, Ijzerman, Adriaan P.
Published in Journal of medicinal chemistry (26.02.2009)
Published in Journal of medicinal chemistry (26.02.2009)
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