Next generation GLP-1/GIP/glucagon triple agonists normalize body weight in obese mice
Knerr, Patrick J., Mowery, Stephanie A., Douros, Jonathan D., Premdjee, Bhavesh, Hjøllund, Karina Rahr, He, Yantao, Kruse Hansen, Ann Maria, Olsen, Anette K., Perez-Tilve, Diego, DiMarchi, Richard D., Finan, Brian
Published in Molecular metabolism (Germany) (01.09.2022)
Published in Molecular metabolism (Germany) (01.09.2022)
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ABC and SLC Transporter Expression and Pot Substrate Characterization across the Human CMEC/D3 Blood−Brain Barrier Cell Line
Carl, Stephen M, Lindley, David J, Couraud, Pierre O, Weksler, Babette B, Romero, Ignacio, Mowery, Stephanie A, Knipp, Gregory T
Published in Molecular pharmaceutics (02.08.2010)
Published in Molecular pharmaceutics (02.08.2010)
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The glucose-dependent insulinotropic polypeptide (GIP) regulates body weight and food intake via CNS-GIPR signaling
Zhang, Qian, Delessa, Challa Tenagne, Augustin, Robert, Bakhti, Mostafa, Colldén, Gustav, Drucker, Daniel J., Feuchtinger, Annette, Caceres, Cristina Garcia, Grandl, Gerald, Harger, Alexandra, Herzig, Stephan, Hofmann, Susanna, Holleman, Cassie Lynn, Jastroch, Martin, Keipert, Susanne, Kleinert, Maximilian, Knerr, Patrick J., Kulaj, Konxhe, Legutko, Beata, Lickert, Heiko, Liu, Xue, Luippold, Gerd, Lutter, Dominik, Malogajski, Emilija, Medina, Marta Tarquis, Mowery, Stephanie A., Blutke, Andreas, Perez-Tilve, Diego, Salinno, Ciro, Sehrer, Laura, DiMarchi, Richard D., Tschöp, Matthias H., Stemmer, Kerstin, Finan, Brian, Wolfrum, Christian, Müller, Timo D.
Published in Cell metabolism (06.04.2021)
Published in Cell metabolism (06.04.2021)
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Selection and progression of unimolecular agonists at the GIP, GLP-1, and glucagon receptors as drug candidates
Knerr, Patrick J., Mowery, Stephanie A., Finan, Brian, Perez-Tilve, Diego, Tschöp, Matthias H., DiMarchi, Richard D.
Published in Peptides (New York, N.Y. : 1980) (01.03.2020)
Published in Peptides (New York, N.Y. : 1980) (01.03.2020)
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Characterization of genetic variants of GIPR reveals a contribution of β-arrestin to metabolic phenotypes
Kizilkaya, Hüsün S, Sørensen, Kimmie V, Madsen, Jakob S, Lindquist, Peter, Douros, Jonathan D, Bork-Jensen, Jette, Berghella, Alessandro, Gerlach, Peter A, Gasbjerg, Lærke S, Mokrosiński, Jacek, Mowery, Stephanie A, Knerr, Patrick J, Finan, Brian, Campbell, Jonathan E, D'Alessio, David A, Perez-Tilve, Diego, Faas, Felix, Mathiasen, Signe, Rungby, Jørgen, Sørensen, Henrik T, Vaag, Allan, Nielsen, Jens S, Holm, Jens-Christian, Lauenborg, Jeannet, Damm, Peter, Pedersen, Oluf, Linneberg, Allan, Hartmann, Bolette, Holst, Jens J, Hansen, Torben, Wright, Shane C, Lauschke, Volker M, Grarup, Niels, Hauser, Alexander S, Rosenkilde, Mette M
Published in Nature metabolism (01.07.2024)
Published in Nature metabolism (01.07.2024)
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Correction to “ABC and SLC Transporter Expression and Proton Oligopeptide Transporter (POT) Mediated Permeation across the Human Blood–Brain Barrier Cell Line, hCMEC/D3”
Carl, Stephen M, Lindley, David J, Das, Debanjan, Couraud, Pierre O, Weksler, Babette B, Romero, Ignacio, Mowery, Stephanie A, Knipp, Gregory T
Published in Molecular pharmaceutics (03.12.2012)
Published in Molecular pharmaceutics (03.12.2012)
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THE EVALUATION OF PEPTIDE/HISTIDINE TRANSPORTER 1 (PHT1) FUNCTION: UPTAKE KINETICS UTILIZING A COS-7 STABLY TRANSFECTED CELL LINE
Lindley, David J, Carl, Stephen M, Mowery, Stephanie A, Knipp, Gregory T
Published in Revista mexicana de ciencias farmacéutica (01.10.2011)
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Published in Revista mexicana de ciencias farmacéutica (01.10.2011)
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Evaluation of human peptide/histidine transporter 1 (hPHT1/SLC15A4) function: transport kinetics utilizing a HPHT1 shRNA stably transfected knockdown in the hCMEC/D3 blood-brain barrier cell line
Knipp, Gregory T, Lindley, David J, Carl, Stephen M, Mowery, Stephanie A, Roth, Wyatt J
Published in Pharmacy & Pharmacology International Journal (18.06.2021)
Published in Pharmacy & Pharmacology International Journal (18.06.2021)
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ABC AND SLC TRANSPORTER EXPRESSION AND POT SUBSTRATE CHRACTERIZATION ACROSS THE HUMAN CMEC/D3 BLOOD-BRAIN BARRIER CELL LINE
Carl, Stephen M., Lindley, David J., Couraud, Pierre O., Weksler, Babette B., Romero, Ignacio, Mowery, Stephanie A., Knipp, Gregory T.
Published in Molecular pharmaceutics (02.08.2010)
Published in Molecular pharmaceutics (02.08.2010)
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Journal Article
ABC and SLC transporter expression and proton oligopeptide transporter (POT) mediated permeation across the human blood--brain barrier cell line, hCMEC/D3 [corrected]
Carl, Stephen M, Lindley, David J, Das, Debanjan, Couraud, Pierre O, Weksler, Babette B, Romero, Ignacio, Mowery, Stephanie A, Knipp, Gregory T
Published in Molecular pharmaceutics (02.08.2010)
Published in Molecular pharmaceutics (02.08.2010)
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