Copper-Mediated Radiofluorination of Arylstannanes with [18F]KF
Makaravage, Katarina J, Brooks, Allen F, Mossine, Andrew V, Sanford, Melanie S, Scott, Peter J. H
Published in Organic letters (21.10.2016)
Published in Organic letters (21.10.2016)
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Journal Article
Solution‐Phase Magnetic Mechanistic Study of Ni‐Seamed Pyrogallol[4]arene Nanocapsules Reveal Presence of Novel Cylindrical and Spherical Species
Kumari, Harshita, Dennis, Cindi L., Kline, Steven R., Mossine, Andrew V., Deakyne, Carol A., Atwood, Jerry L.
Published in Angewandte Chemie International Edition (25.07.2022)
Published in Angewandte Chemie International Edition (25.07.2022)
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Journal Article
Synthesis of high-molar-activity [ 18 F]6-fluoro-L-DOPA suitable for human use via Cu-mediated fluorination of a BPin precursor
Mossine, Andrew V, Tanzey, Sean S, Brooks, Allen F, Makaravage, Katarina J, Ichiishi, Naoko, Miller, Jason M, Henderson, Bradford D, Erhard, Thomas, Bruetting, Christian, Skaddan, Marc B, Sanford, Melanie S, Scott, Peter J H
Published in Nature protocols (01.05.2020)
Published in Nature protocols (01.05.2020)
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Journal Article
Development of Customized [ 18 F]Fluoride Elution Techniques for the Enhancement of Copper-Mediated Late-Stage Radiofluorination
Mossine, Andrew V, Brooks, Allen F, Ichiishi, Naoko, Makaravage, Katarina J, Sanford, Melanie S, Scott, Peter J H
Published in Scientific reports (22.03.2017)
Published in Scientific reports (22.03.2017)
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Journal Article
Identification of AV-1451 as a Weak, Nonselective Inhibitor of Monoamine Oxidase
Drake, Lindsey R, Pham, Jonathan M, Desmond, Timothy J, Mossine, Andrew V, Lee, So Jeong, Kilbourn, Michael R, Koeppe, Robert A, Brooks, Allen F, Scott, Peter J.H
Published in ACS chemical neuroscience (21.08.2019)
Published in ACS chemical neuroscience (21.08.2019)
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Journal Article
Preliminary Evaluations of [11C]Verubulin: Implications for Microtubule Imaging With PET
Lindberg, Anton, Mossine, Andrew V., Aliaga, Arturo, Hopewell, Robert, Massarweh, Gassan, Rosa-Neto, Pedro, Shao, Xia, Bernard-Gauthier, Vadim, Scott, Peter J. H., Vasdev, Neil
Published in Frontiers in neuroscience (08.09.2021)
Published in Frontiers in neuroscience (08.09.2021)
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Journal Article
Synthesis and Initial In Vivo Evaluation of [ 11 C]AZ683-A Novel PET Radiotracer for Colony Stimulating Factor 1 Receptor (CSF1R)
Tanzey, Sean S, Shao, Xia, Stauff, Jenelle, Arteaga, Janna, Sherman, Phillip, Scott, Peter J H, Mossine, Andrew V
Published in Pharmaceuticals (Basel, Switzerland) (13.12.2018)
Published in Pharmaceuticals (Basel, Switzerland) (13.12.2018)
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Journal Article
One-pot synthesis of high molar activity 6-[F-18]fluoro-l-DOPA by Cu-mediated fluorination of a BPin precursor
Mossine, Andrew V., Tanzey, Sean S., Brooks, Allen F., Makaravage, Katarina J., Ichiishi, Naoko, Miller, Jason M., Henderson, Bradford D., Skaddan, Marc B., Sanford, Melanie S., Scott, Peter J. H.
Published in Organic & biomolecular chemistry (2019)
Published in Organic & biomolecular chemistry (2019)
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Journal Article
Identification of [18F]TRACK, a Fluorine-18-Labeled Tropomyosin Receptor Kinase (Trk) Inhibitor for PET Imaging
Bernard-Gauthier, Vadim, Mossine, Andrew V, Mahringer, Anne, Aliaga, Arturo, Bailey, Justin J, Shao, Xia, Stauff, Jenelle, Arteaga, Janna, Sherman, Phillip, Grand’Maison, Marilyn, Rochon, Pierre-Luc, Wängler, Björn, Wängler, Carmen, Bartenstein, Peter, Kostikov, Alexey, Kaplan, David R, Fricker, Gert, Rosa-Neto, Pedro, Scott, Peter J. H, Schirrmacher, Ralf
Published in Journal of medicinal chemistry (22.02.2018)
Published in Journal of medicinal chemistry (22.02.2018)
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Journal Article
Controlling the Self-Assembly of Metal-Seamed Organic Nanocapsules
Kumari, Harshita, Mossine, Andrew V., Kline, Steven R., Dennis, Cindi L., Fowler, Drew A., Teat, Simon J., Barnes, Charles L., Deakyne, Carol A., Atwood, Jerry L.
Published in Angewandte Chemie (International ed.) (06.02.2012)
Published in Angewandte Chemie (International ed.) (06.02.2012)
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Journal Article
Structural Basis for Achieving GSK-3β Inhibition with High Potency, Selectivity, and Brain Exposure for Positron Emission Tomography Imaging and Drug Discovery
Bernard-Gauthier, Vadim, Mossine, Andrew V, Knight, Ashley, Patnaik, Debasis, Zhao, Wen-Ning, Cheng, Chialin, Krishnan, Hema S, Xuan, Lucius L, Chindavong, Peter S, Reis, Surya A, Chen, Jinshan Michael, Shao, Xia, Stauff, Jenelle, Arteaga, Janna, Sherman, Phillip, Salem, Nicolas, Bonsall, David, Amaral, Brenda, Varlow, Cassis, Wells, Lisa, Martarello, Laurent, Patel, Shil, Liang, Steven H, Kurumbail, Ravi G, Haggarty, Stephen J, Scott, Peter J. H, Vasdev, Neil
Published in Journal of medicinal chemistry (14.11.2019)
Published in Journal of medicinal chemistry (14.11.2019)
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Journal Article
Engineering Void Space Enclosed within Resorcin[4]arene-Based Supramolecular Frameworks
Patil, Rahul S, Mossine, Andrew V, Kumari, Harshita, Barnes, Charles L, Atwood, Jerry L
Published in Crystal growth & design (01.10.2014)
Published in Crystal growth & design (01.10.2014)
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Journal Article
Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2
Mossine, Andrew V, Brooks, Allen F, Jackson, Isaac M, Quesada, Carole A, Sherman, Phillip, Cole, Erin L, Donnelly, David J, Scott, Peter J H, Shao, Xia
Published in Bioconjugate chemistry (18.05.2016)
Published in Bioconjugate chemistry (18.05.2016)
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Journal Article
Coordination Polymer Chains of Dimeric Pyrogallol[4]arene Capsules
Fowler, Drew A, Mossine, Andrew V, Beavers, Christine M, Teat, Simon J, Dalgarno, Scott J, Atwood, Jerry L
Published in Journal of the American Chemical Society (27.07.2011)
Published in Journal of the American Chemical Society (27.07.2011)
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Journal Article
A Kinome-Wide Selective Radiolabeled TrkB/C Inhibitor for in Vitro and in Vivo Neuroimaging: Synthesis, Preclinical Evaluation, and First-in-Human
Bernard-Gauthier, Vadim, Bailey, Justin J, Mossine, Andrew V, Lindner, Simon, Vomacka, Lena, Aliaga, Arturo, Shao, Xia, Quesada, Carole A, Sherman, Phillip, Mahringer, Anne, Kostikov, Alexey, Grand’Maison, Marilyn, Rosa-Neto, Pedro, Soucy, Jean-Paul, Thiel, Alexander, Kaplan, David R, Fricker, Gert, Wängler, Björn, Bartenstein, Peter, Schirrmacher, Ralf, Scott, Peter J. H
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article