Synthesis and Pharmacological Evaluation of Novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole Derivatives as Promising Anxiolytic and Analgesic Agents
Maltsev, Dmitriy V., Spasov, Alexander A., Vassiliev, Pavel M., Skripka, Maria O., Miroshnikov, Mikhail V., Kochetkov, Andrey N., Eliseeva, Nataliya V., Lifanova, Yuliya V., Kuzmenko, Tatyana A., Divaeva, Lyudmila N., Morkovnik, Anatolii S.
Published in Molecules (Basel, Switzerland) (06.10.2021)
Published in Molecules (Basel, Switzerland) (06.10.2021)
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Design, Synthesis and Pharmacological Evaluation of Novel C2,C3-Quinoxaline Derivatives as Promising Anxiolytic Agents
Maltsev, Dmitriy V., Skripka, Maria O., Spasov, Alexander A., Vassiliev, Pavel M., Perfiliev, Maxim A., Divaeva, Lyudmila N., Zubenko, Alexander A., Morkovnik, Anatolii S., Klimenko, Alexander I., Miroshnikov, Mikhail V., Klochkov, Vladlen G., Ianalieva, Laura R.
Published in International journal of molecular sciences (19.11.2022)
Published in International journal of molecular sciences (19.11.2022)
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Towards multi-target antidiabetic agents: Discovery of biphenyl-benzimidazole conjugates as AMPK activators
Babkov, Denis A., Zhukowskaya, Olga N., Borisov, Alexander V., Babkova, Valentina A., Sokolova, Elena V., Brigadirova, Anastasia A., Litvinov, Roman A., Kolodina, Alexandra A., Morkovnik, Anatolii S., Sochnev, Vadim S., Borodkin, Gennady S., Spasov, Alexander A.
Published in Bioorganic & medicinal chemistry letters (01.09.2019)
Published in Bioorganic & medicinal chemistry letters (01.09.2019)
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Discovery and evaluation of biphenyl derivatives of 2‐iminobenzimidazoles as prototype dual PTP1B inhibitors and AMPK activators with in vivo antidiabetic activity
Babkov, Denis A., Zhukovskaya, Olga N., Brigadirova, Anastasia A., Prilepskaya, Diana R., Kolodina, Alexandra A., Abbas, Abbas Haider S., Morkovnik, Anatolii S., Sobhia, M. Elizabeth, Ghosh, Ketan, Spasov, Alexander A.
Published in Chemical biology & drug design (01.04.2023)
Published in Chemical biology & drug design (01.04.2023)
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Searching for new anxiolytic agents among derivatives of 11-dialkylaminoethyl-2,3,4,5-tetrahydrodiazepino[1,2-a]benzimidazole
Maltsev, Dmitriy V., Spasov, Alexander A., Yakovlev, Dmitriy S., Vassiliev, Pavel M., Skripka, Maria O., Miroshnikov, Mikhail V., Sultanova, Kira T., Kochetkov, Andrey N., Divaeva, Lyudmila N., Kuzmenko, Tatyana A., Morkovnik, Anatolii S.
Published in European journal of pharmaceutical sciences (01.06.2021)
Published in European journal of pharmaceutical sciences (01.06.2021)
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Tautomeric and non-tautomeric N-substituted 2-iminobenzimidazolines as new lead compounds for the design of anti-influenza drugs: An in vitro study
Zarubaev, Vladimir V., Morkovnik, Anatolii S., Divaeva, Liudmila N., Karpinskaya, Liubov' A., Borodkin, Gennadii S.
Published in Bioorganic & medicinal chemistry (15.11.2016)
Published in Bioorganic & medicinal chemistry (15.11.2016)
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Hypoglycemic potential of cyclic guanidine derivatives
Spasov, Alexander A., Vassiliev, Pavel M., Lenskaya, Karina V., Anisimova, Vera A., Kuzmenko, Tatyana A., Morkovnik, Anatolii S., Kosolapov, Vadim A., Babkov, Denis A.
Published in Pure and applied chemistry (01.08.2017)
Published in Pure and applied chemistry (01.08.2017)
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Design, Synthesis and Pharmacological Evaluation of Novel C 2 ,C 3 -Quinoxaline Derivatives as Promising Anxiolytic Agents
Maltsev, Dmitriy V, Skripka, Maria O, Spasov, Alexander A, Vassiliev, Pavel M, Perfiliev, Maxim A, Divaeva, Lyudmila N, Zubenko, Alexander A, Morkovnik, Anatolii S, Klimenko, Alexander I, Miroshnikov, Mikhail V, Klochkov, Vladlen G, Ianalieva, Laura R
Published in International journal of molecular sciences (19.11.2022)
Published in International journal of molecular sciences (19.11.2022)
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Journal Article
An efficient, one-pot synthesis of N-isatinylmethylthioacetic acid and its derivatives as potential anticancer agents
Ukhin, Lev Yu, Akopova, Arina R., Morkovnik, Anatolii S., Suponitzky, Kirill Yu, Shepelenko, Evgenii N., Bicherov, Alexander V., Popov, Leonid D.
Published in Tetrahedron letters (19.11.2014)
Published in Tetrahedron letters (19.11.2014)
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A facile, one pot method for the synthesis of 4-acyl-1,2-dihydro-3-benzazepines, based on the ring expansion of natural and synthetic 3,4-dihydroisoquinoline pseudo bases
Kartsev, Viktor G., Zubenko, Alexander A., Morkovnik, Anatolii S., Divaeva, Ludmila N.
Published in Tetrahedron letters (16.12.2015)
Published in Tetrahedron letters (16.12.2015)
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β-Carbolines as intermediates in indirect heteroarylation of tryptamines exemplified by the synthesis of 2-pyrazolyltryptamines
Zubenko, Alexander A., Divaeva, Lyudmila N., Morkovnik, Anatolii S., Sochnev, Vadim S., Demidov, Oleg P., Chekrysheva, Viktorya V., Klimenko, Alexander I., Svyatogorova, Alexandra E.
Published in Mendeleev communications (01.09.2023)
Published in Mendeleev communications (01.09.2023)
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New β-[o-(5-oxopyrazol-3-yl)aryl]ethylamines and their unusual metastable betaine form
Zubenko, Alexander A., Morkovnik, Anatolii S., Divaeva, Lyudmila N., Sochnev, Vadim S., Demidov, Oleg P., Fetisov, Leonid N., Andros, Natal'ya O., Svyatogorova, Alexandra E., Klimenko, Alexander I.
Published in Mendeleev communications (01.03.2023)
Published in Mendeleev communications (01.03.2023)
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Journal Article
One-pot synthesis of 4-heteroaryl-1,2-dihydro-3-benzazepines from 3,4-dihydroisoquinolinium salts or pseudo bases
Zubenko, Alexander A., Kartsev, Viktor G., Morkovnik, Anatolii S., Divaeva, Ludmila N., Alexeenko, Danil V., Suponitsky, Kyrill Yu, Borodkin, Gennadii S., Klimenko, Alexander I.
Published in Tetrahedron letters (22.03.2017)
Published in Tetrahedron letters (22.03.2017)
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ChemInform Abstract: A Facile, One Pot Method for the Synthesis of 4‐Acyl‐1,2‐dihydro‐3‐benzazepines, Based on the Ring Expansion of Natural and Synthetic 3,4‐Dihydroisoquinoline Pseudo Bases
Kartsev, Viktor G., Zubenko, Alexander A., Morkovnik, Anatolii S., Divaeva, Ludmila N.
Published in ChemInform (01.03.2016)
Published in ChemInform (01.03.2016)
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ChemInform Abstract: Unexpected Domino Reaction of 3‐Alkyl‐1,2,4‐triazolo[1,5‐a]benzimidazoles with Butylmagnesium Bromide Leading to Benzimidazolyl Guanidines
Koshchienko, Yurii V., Kuz'menko, Tatyana A., Morkovnik, Anatolii S., Kiskin, Mikhail A., Alexandrov, Grigorii G.
Published in ChemInform (01.12.2016)
Published in ChemInform (01.12.2016)
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Novel recyclization of 3,4-dihydroisoquinolines as an efficient route to a new type of heteroarylated derivatives of β-arylethylamines
Sochnev, Vadim S., Morkovnik, Anatolii S., Zubenko, Alexander A., Divaeva, Lyudmila N., Demidov, Oleg P., Gribanova, Tatyana N., Fetisov, Leonid N., Chekrysheva, Viktorya V., Kononenko, Kristina N., Bodryakova, Marya A., Klimenko, Alexander I., Borodkin, Gennadii S., Estrin, Igor A.
Published in Mendeleev communications (01.11.2022)
Published in Mendeleev communications (01.11.2022)
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New route to bioactive 2-(hetero)arylethylamines via nucleophilic ring opening in fused 7-acyl-2,3-dihydroazepines
Zubenko, Alexander A., Morkovnik, Anatolii S., Divaeva, Lyudmila N., Demidov, Oleg P., Sochnev, Vadim S., Borodkina, Inna G., Drobin, Yuriy D., Spasov, Alexander A.
Published in Mendeleev communications (01.01.2020)
Published in Mendeleev communications (01.01.2020)
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Nitration of 2,3-dihydroimidazo[1,2-a]benzimidazole and its N 9-substituted derivatives
Sochnev, Vadim S., Kuz'menko, Tatyana A., Morkovnik, Anatolii S., Divaeva, Lyudmila N., Podobina, Anastasia S., Zubenko, Alexander A., Chepurnoy, Pavel B., Borodkin, Gennadii S., Klimenko, Alexander I.
Published in Mendeleev communications (01.07.2021)
Published in Mendeleev communications (01.07.2021)
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New type of recyclization in 3,4-dihydroisoquinolines in the synthesis of β-(o-indazolylaryl)ethylamines and their 7-azaindazolyl analogues
Zubenko, Aleksandr A., Morkovnik, Anatolii S., Divaeva, Lyudmila N., Sochnev, Vadim S., Demidov, Oleg P., Klimenko, Aleksandr I., Fetisov, Leonid N., Bodryakov, Anatolii N., Bodryakova, Mariya A., Borodkin, Gennadii S.
Published in Mendeleev communications (01.03.2022)
Published in Mendeleev communications (01.03.2022)
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The novel structural modification of pyridoxal via its cyclization into 2-acyl- and 2-heteroarylfuro[2,3-c]pyridines
Morkovnik, Anatolii S., Zubenko, Alexander A., Divaeva, Ludmila N., Kartsev, Victor G., Borodkin, Gennadii S., Klimenko, Alexander I.
Published in Mendeleev communications (01.01.2019)
Published in Mendeleev communications (01.01.2019)
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