Identification of the binding site for a novel class of CCR2b chemokine receptor antagonists: binding to a common chemokine receptor motif within the helical bundle
Mirzadegan, T, Diehl, F, Ebi, B, Bhakta, S, Polsky, I, McCarley, D, Mulkins, M, Weatherhead, G S, Lapierre, J M, Dankwardt, J, Morgans, Jr, D, Wilhelm, R, Jarnagin, K
Published in The Journal of biological chemistry (18.08.2000)
Published in The Journal of biological chemistry (18.08.2000)
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Novel inhibitors of poly(ADP-ribose) polymerase/PARP1 and PARP2 identified using a cell-based screen in yeast
PERKINS, Ed, DONGXU SUN, YEH, Elaine, THODE, Silke, JARNAGIN, Kurt, JAIN, Ajay, MORGANS, David, MELESE, Teri, NGUYEN, Allen, TULAC, Suzana, FRANCESCO, Michelle, TAVANA, Homa, NGUYEN, Hieu, TUGENDREICH, Stuart, BARTHMAIER, Peter, COUTO, Joe
Published in Cancer research (Chicago, Ill.) (15.05.2001)
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Published in Cancer research (Chicago, Ill.) (15.05.2001)
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Synthesis, pharmacology and pharmacokinetics of 3-(4-aryl-piperazin-1-ylalkyl)-uracils as uroselective α1A-antagonists
LOPEZ, F. J, ARIAS, L, PADILLA, F, PEREZ-MEDRANO, A, QUINTERO, C, ROMERO, M, SANDOVAL, L, SMITH, S. A, WILLIAMS, T. J, BLUE, D. R, CHAN, R, CLARKE, D. E, ELWORTHY, T. R, FORD, A. P. D. W, GUZMAN, A, JAIME-FIGUEROA, S, JASPER, J. R, MORGANS, D. J
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Synthesis, pharmacology and pharmacokinetics of 3-(4-aryl-piperazin-1-ylalkyl)-uracils as uroselective alpha1A-antagonists
Lopez, F J, Arias, L, Chan, R, Clarke, D E, Elworthy, T R, Ford, A P D W, Guzman, A, Jaime-Figueroa, S, Jasper, J R, Morgans, Jr, D J, Padilla, F, Perez-Medrano, A, Quintero, C, Romero, M, Sandoval, L, Smith, S A, Williams, T J, Blue, D R
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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In vitroα1‐adrenoceptor pharmacology of Ro 70–0004 and RS‐100329, novel α1A‐adrenoceptor selective antagonists
Williams, T J, Blue, D R, Daniels, D V, Davis, B, Elworthy, T, Gever, J R, Kava, M S, Morgans, D, Padilla, F, Tassa, S, Vimont, R L, Chapple, C R, Chess‐Williams, R, Eglen, R M, Clarke, D E, Ford, A P D W
Published in British journal of pharmacology (01.05.1999)
Published in British journal of pharmacology (01.05.1999)
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Synthesis of N-allylhydroxamic acids via [3,3]-sigmatropic rearrangement
De la Torre, J.A., Fernandez, M., Morgans, D., Smith, David B., Talamas, F.X., Trejo, A.
Published in Tetrahedron letters (03.01.1994)
Published in Tetrahedron letters (03.01.1994)
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Improved methodology for the enantiospecific synthesis of polyunsaturated phospholipids
MORGANS, D. JR, RAMESHA, C, ROMERO, M, TALAMAS, F. X
Published in Bioorganic & medicinal chemistry letters (24.03.1994)
Published in Bioorganic & medicinal chemistry letters (24.03.1994)
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Epoxy alcohol rearrangements: hydroxyl-mediated delivery of Lewis acid promoters
Morgans, D. J, Sharpless, K. B, Traynor, Sean G
Published in Journal of the American Chemical Society (01.01.1981)
Published in Journal of the American Chemical Society (01.01.1981)
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Thrombocytopenia and platelet functional defects in pre-eclampsia : implications for regional anaesthesia
SCHINDLER, M, GATT, S, ISERT, P, MORGANS, D, CHEUNG, A
Published in Anaesthesia and intensive care (01.05.1990)
Published in Anaesthesia and intensive care (01.05.1990)
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TEMPORARY SERINE PROTECTION IN SOLID-PHASE SYNTHESIS OF LH-RH ANALOGS
ARZENO, HB, BINGENHEIMER, W, BLANCHETTE, R, MORGANS, DJ, ROBINSON, J
Published in International journal of peptide and protein research (01.04.1993)
Published in International journal of peptide and protein research (01.04.1993)
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Asymmetric Synthesis and Stereochemical Assignment of RS-97613, a Potent Immunosuppressive and Antiinflammatory Agent
Smith, David B, Waltos, Ann Marie, Loughhead, David G, Weikert, Robert J, Morgans, David J, Rohloff, John C, Link, John O, Zhu, Rong-rong
Published in Journal of organic chemistry (22.03.1996)
Published in Journal of organic chemistry (22.03.1996)
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