Stable Pyrrole‐Linked Bioconjugates through Tetrazine‐Triggered Azanorbornadiene Fragmentation
Gil de Montes, Enrique, Istrate, Alena, Navo, Claudio D., Jiménez‐Moreno, Ester, Hoyt, Emily A., Corzana, Francisco, Robina, Inmaculada, Jiménez‐Osés, Gonzalo, Moreno‐Vargas, Antonio J., Bernardes, Gonçalo J. L.
Published in Angewandte Chemie International Edition (06.04.2020)
Published in Angewandte Chemie International Edition (06.04.2020)
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Synthesis and Glycosidase Inhibition Studies of 5-Methyl-Substituted Tetrahydroxyindolizidines and -pyrrolizidines Related to Natural Hyacinthacines B
Martella, Daniele, Cardona, Francesca, Parmeggiani, Camilla, Franco, Francisco, Tamayo, Juan A., Robina, Inmaculada, Moreno-Clavijo, Elena, Moreno-Vargas, Antonio J., Goti, Andrea
Published in European journal of organic chemistry (01.07.2013)
Published in European journal of organic chemistry (01.07.2013)
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Mechanistic Insight into the Binding of Multivalent Pyrrolidines to α‐Mannosidases
Mirabella, Stefania, D'Adamio, Giampiero, Matassini, Camilla, Goti, Andrea, Delgado, Sandra, Gimeno, Ana, Robina, Inmaculada, Moreno‐Vargas, Antonio J., Šesták, Sergej, Jiménez‐Barbero, Jesús, Cardona, Francesca
Published in Chemistry : a European journal (17.10.2017)
Published in Chemistry : a European journal (17.10.2017)
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Discovery of human hexosaminidase inhibitors by in situ screening of a library of mono- and divalent pyrrolidine iminosugars
Pingitore, Valeria, Martínez-Bailén, Macarena, Carmona, Ana T., Mészáros, Zuzana, Kulik, Natalia, Slámová, Kristýna, Křen, Vladimír, Bojarová, Pavla, Robina, Inmaculada, Moreno-Vargas, Antonio J.
Published in Bioorganic chemistry (01.03.2022)
Published in Bioorganic chemistry (01.03.2022)
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Journal Article
Polyhydroxyamino-Piperidine-Type Iminosugars and Pipecolic Acid Analogues from a D-Mannose-Derived Aldehyde
Matassini, Camilla, Mirabella, Stefania, Ferhati, Xhenti, Faggi, Cristina, Robina, Inmaculada, Goti, Andrea, Moreno-Clavijo, Elena, Moreno-Vargas, Antonio J., Cardona, Francesca
Published in European journal of organic chemistry (01.09.2014)
Published in European journal of organic chemistry (01.09.2014)
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Journal Article
Synthesis, Biological Evaluation, WAC and NMR Studies of S-Galactosides and Non-Carbohydrate Ligands of Cholera Toxin Based on Polyhydroxyalkylfuroate Moieties
Ramos-Soriano, Javier, Niss, Ulf, Angulo, Jesús, Angulo, Manuel, Moreno-Vargas, Antonio J., Carmona, Ana T., Ohlson, Sten, Robina, Inmaculada
Published in Chemistry : a European journal (23.12.2013)
Published in Chemistry : a European journal (23.12.2013)
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Journal Article
Exploring architectures displaying multimeric presentations of a trihydroxypiperidine iminosugar
Matassini, Camilla, Mirabella, Stefania, Goti, Andrea, Robina, Inmaculada, Moreno-Vargas, Antonio J, Cardona, Francesca
Published in Beilstein journal of organic chemistry (16.12.2015)
Published in Beilstein journal of organic chemistry (16.12.2015)
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Journal Article
New Methodology for the Stereoselective Synthesis of α-Furfurylamines from Sugars: Application to the Synthesis of Furyl Amino Acids and 3-Furylisoserines
Molina, Lidia, Moreno-Clavijo, Elena, Moreno-Vargas, Antonio J., Carmona, Ana T., Robina, Inmaculada
Published in European Journal of Organic Chemistry (01.06.2010)
Published in European Journal of Organic Chemistry (01.06.2010)
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Book Review
Journal Article
Transferring Substituents from Alkynes to Furans and Pyrroles through Heteronorbornadienes as Intermediates: Synthesis of β‑Substituted Pyrroles/Furans
García-Domínguez, Javier, Carranza, Marina, Jansons, Edijs, Carmona, Ana T., Robina, Inmaculada, Moreno-Vargas, Antonio J.
Published in Journal of organic chemistry (15.09.2023)
Published in Journal of organic chemistry (15.09.2023)
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Synthesis and structure-activity relationship of new nicotinamide phosphoribosyltransferase inhibitors with antitumor activity on solid and haematological cancer
Fratta, Simone, Biniecka, Paulina, Moreno-Vargas, Antonio J., Carmona, Ana T., Nahimana, Aimable, Duchosal, Michel A., Piacente, Francesco, Bruzzone, Santina, Caffa, Irene, Nencioni, Alessio, Robina, Inmaculada
Published in European journal of medicinal chemistry (15.03.2023)
Published in European journal of medicinal chemistry (15.03.2023)
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Journal Article
Experimental and Theoretical Analysis of the Thiol-Promoted Fragmentation of 2‑Halo-3-tosyl-oxanorbornadienes
Carranza, Marina, Carmona, Ana T., Navo, Claudio D., Robina, Inmaculada, Fratta, Simone, Newburn, Carlos, Jiménez-Osés, Gonzalo, Moreno-Vargas, Antonio J.
Published in Organic letters (20.10.2023)
Published in Organic letters (20.10.2023)
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Journal Article
Dual targeting of PTP1B and glucosidases with new bifunctional iminosugar inhibitors to address type 2 diabetes
Ferhati, Xhenti, Matassini, Camilla, Fabbrini, Maria Giulia, Goti, Andrea, Morrone, Amelia, Cardona, Francesca, Moreno-Vargas, Antonio J., Paoli, Paolo
Published in Bioorganic chemistry (01.06.2019)
Published in Bioorganic chemistry (01.06.2019)
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Synthesis of multimeric pyrrolidine iminosugar inhibitors of human β-glucocerebrosidase and α-galactosidase A: First example of a multivalent enzyme activity enhancer for Fabry disease
Martínez-Bailén, Macarena, Carmona, Ana T., Cardona, Francesca, Matassini, Camilla, Goti, Andrea, Kubo, Moemi, Kato, Atsushi, Robina, Inmaculada, Moreno-Vargas, Antonio J.
Published in European journal of medicinal chemistry (15.04.2020)
Published in European journal of medicinal chemistry (15.04.2020)
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Journal Article
Studies on the Regioselective Rearrangement of Azanorbornanic Aminyl Radicals into 2,8-Diazabicyclo[3.2.1]oct-2-ene Systems
de Montes, Enrique Gil, Tallarida, Matteo A., Carmona, Ana T., Navo, Claudio D., Robina, Inmaculada, Elías-Rodríguez, Pilar, Jiménez-Osés, Gonzalo, Moreno-Vargas, Antonio J.
Published in Journal of organic chemistry (16.12.2022)
Published in Journal of organic chemistry (16.12.2022)
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Identification of new FK866 analogues with potent anticancer activity against pancreatic cancer
Bai, Jian-Fei, Majjigapu, Somi Reddy, Sordat, Bernard, Poty, Sophie, Vogel, Pierre, Elías-Rodríguez, Pilar, Moreno-Vargas, Antonio J., Carmona, Ana T., Caffa, Irene, Ghanem, Moustafa, Khalifa, Amr, Monacelli, Fiammetta, Cea, Michele, Robina, Inmaculada, Gajate, Consuelo, Mollinedo, Faustino, Bellotti, Axel, Nahimana, Aimable, Duchosal, Michel, Nencioni, Alessio
Published in European journal of medicinal chemistry (05.09.2022)
Published in European journal of medicinal chemistry (05.09.2022)
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Journal Article
Harnessing pyrrolidine iminosugars into dimeric structures for the rapid discovery of divalent glycosidase inhibitors
Carmona, Ana T., Carrión-Jiménez, Sebastián, Pingitore, Valeria, Moreno-Clavijo, Elena, Robina, Inmaculada, Moreno-Vargas, Antonio J.
Published in European journal of medicinal chemistry (10.05.2018)
Published in European journal of medicinal chemistry (10.05.2018)
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Journal Article
Regioselectivity of the 1,3-Dipolar Cycloaddition of Organic Azides to 7‑Heteronorbornadienes. Synthesis of β‑Substituted Furans/Pyrroles
Gil de Montes, Enrique, Martı́nez-Bailén, Macarena, Carmona, Ana T, Robina, Inmaculada, Moreno-Vargas, Antonio J
Published in Journal of organic chemistry (17.07.2020)
Published in Journal of organic chemistry (17.07.2020)
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Journal Article
Total asymmetric synthesis of monosaccharides and analogues
Robina, Inmaculada, Carmona, Ana T, Moreno-Vargas, Antonio J, Moreno-Clavijo, Elena
Published in Chimia (01.01.2011)
Published in Chimia (01.01.2011)
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Journal Article
Tuning of β-glucosidase and α-galactosidase inhibition by generation and in situ screening of a library of pyrrolidine-triazole hybrid molecules
Martínez-Bailén, Macarena, Carmona, Ana T., Moreno-Clavijo, Elena, Robina, Inmaculada, Ide, Daisuke, Kato, Atsushi, Moreno-Vargas, Antonio J.
Published in European journal of medicinal chemistry (29.09.2017)
Published in European journal of medicinal chemistry (29.09.2017)
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