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Rinaldi, Laura, Delle Donne, Rossella, Catalanotti, Bruno, Torres-Quesada, Omar, Enzler, Florian, Moraca, Federica, Nisticò, Robert, Chiuso, Francesco, Piccinin, Sonia, Bachmann, Verena, Lindner, Herbert H, Garbi, Corrado, Scorziello, Antonella, Russo, Nicola Antonino, Synofzik, Matthis, Stelzl, Ulrich, Annunziato, Lucio, Stefan, Eduard, Feliciello, Antonio
Published in Nature communications (12.06.2019)
Published in Nature communications (12.06.2019)
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Hijacking SARS-CoV-2/ACE2 Receptor Interaction by Natural and Semi-synthetic Steroidal Agents Acting on Functional Pockets on the Receptor Binding Domain
Carino, Adriana, Moraca, Federica, Fiorillo, Bianca, Marchianò, Silvia, Sepe, Valentina, Biagioli, Michele, Finamore, Claudia, Bozza, Silvia, Francisci, Daniela, Distrutti, Eleonora, Catalanotti, Bruno, Zampella, Angela, Fiorucci, Stefano
Published in Frontiers in chemistry (23.10.2020)
Published in Frontiers in chemistry (23.10.2020)
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Folding intermediate states of the parallel human telomeric G-quadruplex DNA explored using Well-Tempered Metadynamics
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Published in Scientific reports (21.02.2020)
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Author Correction: Feedback inhibition of cAMP effector signaling by a chaperone-assisted ubiquitin system
Rinaldi, Laura, Donne, Rossella Delle, Catalanotti, Bruno, Torres-Quesada, Omar, Enzler, Florian, Moraca, Federica, Nisticò, Robert, Chiuso, Francesco, Piccinin, Sonia, Bachmann, Verena, Lindner, Herbert H, Garbi, Corrado, Scorziello, Antonella, Russo, Nicola Antonino, Synofzik, Matthis, Stelzl, Ulrich, Annunziato, Lucio, Stefan, Eduard, Feliciello, Antonio
Published in Nature communications (29.05.2024)
Published in Nature communications (29.05.2024)
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Molecular Basis for Non-Covalent, Non-Competitive FAAH Inhibition
Morgillo, Carmine Marco, Lupia, Antonio, Deplano, Alessandro, Pirone, Luciano, Fiorillo, Bianca, Pedone, Emilia, Luque, F Javier, Onnis, Valentina, Moraca, Federica, Catalanotti, Bruno
Published in International journal of molecular sciences (07.12.2022)
Published in International journal of molecular sciences (07.12.2022)
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Multi-Targeting Bioactive Compounds Extracted from Essential Oils as Kinase Inhibitors
Maruca, Annalisa, Lanzillotta, Delia, Rocca, Roberta, Lupia, Antonio, Costa, Giosuè, Catalano, Raffaella, Moraca, Federica, Gaudio, Eugenio, Ortuso, Francesco, Artese, Anna, Trapasso, Francesco, Alcaro, Stefano
Published in Molecules (Basel, Switzerland) (06.05.2020)
Published in Molecules (Basel, Switzerland) (06.05.2020)
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Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen
Deplano, Alessandro, Karlsson, Jessica, Svensson, Mona, Moraca, Federica, Catalanotti, Bruno, Fowler, Christopher J., Onnis, Valentina
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Discovery of BAR502, as potent steroidal antagonist of leukemia inhibitory factor receptor for the treatment of pancreatic adenocarcinoma
Di Giorgio, Cristina, Bellini, Rachele, Lupia, Antonio, Massa, Carmen, Bordoni, Martina, Marchianò, Silvia, Rosselli, Rosalinda, Sepe, Valentina, Rapacciuolo, Pasquale, Moraca, Federica, Morretta, Elva, Ricci, Patrizia, Urbani, Ginevra, Monti, Maria Chiara, Biagioli, Michele, Distrutti, Eleonora, Catalanotti, Bruno, Zampella, Angela, Fiorucci, Stefano
Published in Frontiers in oncology (14.03.2023)
Published in Frontiers in oncology (14.03.2023)
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Chemoinformatic Database Building and in Silico Hit-Identification of Potential Multi-Targeting Bioactive Compounds Extracted from Mushroom Species
Maruca, Annalisa, Moraca, Federica, Rocca, Roberta, Molisani, Fulvia, Alcaro, Francesca, Gidaro, Maria, Alcaro, Stefano, Costa, Giosuè, Ortuso, Francesco
Published in Molecules (Basel, Switzerland) (19.09.2017)
Published in Molecules (Basel, Switzerland) (19.09.2017)
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Macrocyclic naphthalene diimides as G-quadruplex binders
Marchetti, Chiara, Minarini, Anna, Tumiatti, Vincenzo, Moraca, Federica, Parrotta, Lucia, Alcaro, Stefano, Rigo, Riccardo, Sissi, Claudia, Gunaratnam, Mekala, Ohnmacht, Stephan A., Neidle, Stephen, Milelli, Andrea
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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Structure-based virtual screening of novel natural alkaloid derivatives as potential binders of h-telo and c-myc DNA G-quadruplex conformations
Rocca, Roberta, Moraca, Federica, Costa, Giosuè, Alcaro, Stefano, Distinto, Simona, Maccioni, Elias, Ortuso, Francesco, Artese, Anna, Parrotta, Lucia
Published in Molecules (Basel, Switzerland) (01.01.2015)
Published in Molecules (Basel, Switzerland) (01.01.2015)
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Molecular and Structural Aspects of Clinically Relevant Mutations of SARS-CoV-2 RNA-Dependent RNA Polymerase in Remdesivir-Treated Patients
Gratteri, Carmen, Ambrosio, Francesca Alessandra, Lupia, Antonio, Moraca, Federica, Catalanotti, Bruno, Costa, Giosuè, Bellocchi, Maria, Carioti, Luca, Salpini, Romina, Ceccherini-Silberstein, Francesca, Frazia, Simone La, Malagnino, Vincenzo, Sarmati, Loredana, Svicher, Valentina, Bryant, Sharon, Artese, Anna, Alcaro, Stefano
Published in Pharmaceuticals (Basel, Switzerland) (01.08.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.08.2023)
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Design, synthesis and in vitro and in vivo biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents
Deplano, Alessandro, Karlsson, Jessica, Moraca, Federica, Svensson, Mona, Cristiano, Claudia, Morgillo, Carmine Marco, Fowler, Christopher J., Russo, Roberto, Catalanotti, Bruno, Onnis, Valentina
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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The leukemia inhibitory factor regulates fibroblast growth factor receptor 4 transcription in gastric cancer
Di Giorgio, Cristina, Bellini, Rachele, Lupia, Antonio, Massa, Carmen, Urbani, Ginevra, Bordoni, Martina, Marchianò, Silvia, Rosselli, Rosalinda, De Gregorio, Rosa, Rapacciuolo, Pasquale, Sepe, Valentina, Morretta, Elva, Monti, Maria Chiara, Moraca, Federica, Cari, Luigi, Ullah, Khan Rana Sami, Natalizi, Nicola, Graziosi, Luigina, Distrutti, Eleonora, Biagioli, Michele, Catalanotti, Bruno, Donini, Annibale, Zampella, Angela, Fiorucci, Stefano
Published in Cellular oncology (Dordrecht) (01.04.2024)
Published in Cellular oncology (Dordrecht) (01.04.2024)
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Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors
Deplano, Alessandro, Cipriano, Mariateresa, Moraca, Federica, Novellino, Ettore, Catalanotti, Bruno, Fowler, Christopher J., Onnis, Valentina
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Chromene Derivatives as Selective TERRA G-Quadruplex RNA Binders with Antiproliferative Properties
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Published in Pharmaceuticals (Basel, Switzerland) (28.04.2022)
Published in Pharmaceuticals (Basel, Switzerland) (28.04.2022)
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Repositioning Mifepristone as a Leukaemia Inhibitory Factor Receptor Antagonist for the Treatment of Pancreatic Adenocarcinoma
Di Giorgio, Cristina, Lupia, Antonio, Marchianò, Silvia, Bordoni, Martina, Bellini, Rachele, Massa, Carmen, Urbani, Ginevra, Roselli, Rosalinda, Moraca, Federica, Sepe, Valentina, Catalanotti, Bruno, Morretta, Elva, Monti, Maria Chiara, Biagioli, Michele, Distrutti, Eleonora, Zampella, Angela, Fiorucci, Stefano
Published in Cells (Basel, Switzerland) (03.11.2022)
Published in Cells (Basel, Switzerland) (03.11.2022)
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Exploring the DNA2-PNA heterotriplex formation in targeting the Bcl-2 gene promoter: A structural insight by physico-chemical and microsecond-scale MD investigation
Falanga, Andrea P., Lupia, Antonio, Tripodi, Lorella, Morgillo, Carmine M., Moraca, Federica, Roviello, Giovanni N., Catalanotti, Bruno, Amato, Jussara, Pastore, Lucio, Cerullo, Vincenzo, D'Errico, Stefano, Piccialli, Gennaro, Oliviero, Giorgia, Borbone, Nicola
Published in Heliyon (15.02.2024)
Published in Heliyon (15.02.2024)
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The polymorphisms of DNA G-quadruplex investigated by docking experiments with telomestatin enantiomers
Alcaro, Stefano, Costa, Giosue, Distinto, Simona, Moraca, Federica, Ortuso, Francesco, Parrotta, Lucia, Artese, Anna
Published in Current pharmaceutical design (01.05.2012)
Published in Current pharmaceutical design (01.05.2012)
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Structure–activity relationships of novel substituted naphthalene diimides as anticancer agents
Milelli, Andrea, Tumiatti, Vincenzo, Micco, Marialuisa, Rosini, Michela, Zuccari, Guendalina, Raffaghello, Lizzia, Bianchi, Giovanna, Pistoia, Vito, Fernando Díaz, J., Pera, Benet, Trigili, Chiara, Barasoain, Isabel, Musetti, Caterina, Toniolo, Marianna, Sissi, Claudia, Alcaro, Stefano, Moraca, Federica, Zini, Maddalena, Stefanelli, Claudio, Minarini, Anna
Published in European journal of medicinal chemistry (01.11.2012)
Published in European journal of medicinal chemistry (01.11.2012)
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