Allosteric enhancers for A1 adenosine receptor
Baraldi, Pier Giovanni, Iaconinoto, Maria Antonietta, Moorman, Allan R, Carrion, Maria Dora, Cara, Carlota Lopez, Preti, Delia, López, Olga Cruz, Fruttarolo, Francesca, Tabrizi, Mojgan Aghazade, Romagnoli, Romeo
Published in Mini reviews in medicinal chemistry (01.06.2007)
Published in Mini reviews in medicinal chemistry (01.06.2007)
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7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
Baraldi, Pier Giovanni, Saponaro, Giulia, Moorman, Allan R, Romagnoli, Romeo, Preti, Delia, Baraldi, Stefania, Ruggiero, Emanuela, Varani, Katia, Targa, Martina, Vincenzi, Fabrizio, Borea, Pier Andrea, Aghazadeh Tabrizi, Mojgan
Published in Journal of medicinal chemistry (26.07.2012)
Published in Journal of medicinal chemistry (26.07.2012)
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Journal Article
Current status of A1 adenosine receptor allosteric enhancers
Romagnoli, Romeo, Baraldi, Pier Giovanni, Moorman, Allan R, Borea, Pier Andrea, Varani, Katia
Published in Future medicinal chemistry (2015)
Published in Future medicinal chemistry (2015)
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Journal Article
Pyrrolo- and pyrazolo-[3,4-e][1,2,4]triazolo[1,5-c]pyrimidines as adenosine receptor antagonists
Baraldi, Pier Giovanni, Saponaro, Giulia, Aghazadeh Tabrizi, Mojgan, Baraldi, Stefania, Romagnoli, Romeo, Moorman, Allan R., Varani, Katia, Borea, Pier Andrea, Preti, Delia
Published in Bioorganic & medicinal chemistry (15.01.2012)
Published in Bioorganic & medicinal chemistry (15.01.2012)
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Discovery of 7‑Oxopyrazolo[1,5‑a]pyrimidine-6-carboxamides as Potent and Selective CB2 Cannabinoid Receptor Inverse Agonists
Aghazadeh Tabrizi, Mojgan, Baraldi, Pier Giovanni, Saponaro, Giulia, Moorman, Allan R, Romagnoli, Romeo, Preti, Delia, Baraldi, Stefania, Ruggiero, Emanuela, Tintori, Cristina, Tuccinardi, Tiziano, Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in Journal of medicinal chemistry (13.06.2013)
Published in Journal of medicinal chemistry (13.06.2013)
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Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect study
Romagnoli, Romeo, Baraldi, Pier Giovanni, Lopez-Cara, Carlota, Cruz-Lopez, Olga, Moorman, Allan R., Massink, Arnault, IJzerman, Adriaan P., Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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Journal Article
Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists
Aghazadeh Tabrizi, Mojgan, Baraldi, Pier Giovanni, Saponaro, Giulia, Moorman, Allan R, Romagnoli, Romeo, Preti, Delia, Baraldi, Stefania, Corciulo, Carmen, Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Synthesis and Biological Evaluation of 2‑Amino-3-(4-chlorobenzoyl)-4-[(4-arylpiperazin-1-yl)methyl]-5-substituted-thiophenes. Effect of the 5‑Modification on Allosteric Enhancer Activity at the A1 Adenosine Receptor
Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Cara, Carlota Lopez, Cruz-Lopez, Olga, Salvador, Maria Kimatrai, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Moorman, Allan R, Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in Journal of medicinal chemistry (13.09.2012)
Published in Journal of medicinal chemistry (13.09.2012)
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Journal Article
Synthesis and biological effects of novel 2-amino-3-(4-chlorobenzoyl)-4-substituted thiophenes as allosteric enhancers of the A1 adenosine receptor
Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Lopez Cara, Carlota, Kimatrai Salvador, Maria, Preti, Delia, Aghazadeh Tabrizi, Mojgan, Moorman, Allan R., Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in European journal of medicinal chemistry (01.09.2013)
Published in European journal of medicinal chemistry (01.09.2013)
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Journal Article
Design, Synthesis, and Biological Evaluation of New 8-Heterocyclic Xanthine Derivatives as Highly Potent and Selective Human A2B Adenosine Receptor Antagonists
Baraldi, Pier Giovanni, Tabrizi, Mojgan Aghazadeh, Preti, Delia, Bovero, Andrea, Romagnoli, Romeo, Fruttarolo, Francesca, Zaid, Naser Abdel, Moorman, Allan R, Varani, Katia, Gessi, Stefania, Merighi, Stefania, Borea, Pier Andrea
Published in Journal of medicinal chemistry (11.03.2004)
Published in Journal of medicinal chemistry (11.03.2004)
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Novel 1,3-Dipropyl-8-(3-benzimidazol-2-yl-methoxy-1-methylpyrazol-5-yl)xanthines as Potent and Selective A2B Adenosine Receptor Antagonists
Baraldi, Pier Giovanni, Baraldi, Stefania, Saponaro, Giulia, Preti, Delia, Romagnoli, Romeo, Piccagli, Laura, Cavalli, Andrea, Recanatini, Maurizio, Moorman, Allan R, Zaid, Abdel Naser, Varani, Katia, Borea, Pier Andrea, Tabrizi, Mojgan Aghazadeh
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Journal Article
Synthesis and biological evaluation of novel 2-amino-3-aroyl-4-neopentyl-5-substituted thiophene derivatives as allosteric enhancers of the A1 adenosine receptor
Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Cruz-Lopez, Olga, Cara, Carlota Lopez, Saponaro, Giulia, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Baraldi, Stefania, Moorman, Allan R., Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia
Published in Bioorganic & medicinal chemistry (01.01.2014)
Published in Bioorganic & medicinal chemistry (01.01.2014)
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Journal Article
Synthesis and Biological Evaluation of 2-Amino-3-(4-Chlorobenzoyl)-4-[N-(Substituted) Piperazin-1-yl]Thiophenes as Potent Allosteric Enhancers of the A1 Adenosine Receptor
ROMAGNOLI, Romeo, BARALDI, Pier Giovanni, CARRION, Maria Dora, CARA, Carlota Lopez, CRUZ-LOPEZ, Olga, IACONINOTO, Maria Antonietta, PRETI, Delia, SHRYOCK, John C., MOORMAN, Allan R., VINCENZI, Fabrizio, VARANI, Katia, ANDREA BOREA, Pier
Published in Journal of medicinal chemistry (25.09.2008)
Published in Journal of medicinal chemistry (25.09.2008)
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Journal Article
New Pyrrolo[2,1-f]purine-2,4-dione and Imidazo[2,1-f]purine-2,4-dione Derivatives as Potent and Selective Human A3 Adenosine Receptor Antagonists
Baraldi, Pier Giovanni, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Fruttarolo, Francesca, Romagnoli, Romeo, Zaid, Naser Abdel, Moorman, Allan R, Merighi, Stefania, Varani, Katia, Borea, Pier Andrea
Published in Journal of medicinal chemistry (14.07.2005)
Published in Journal of medicinal chemistry (14.07.2005)
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Journal Article
Structure–activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1-yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A1 adenosine receptor
Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Cara, Carlota Lopez, Cruz-Lopez, Olga, Salvador, Maria Kimatrai, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Shryock, John C., Moorman, Allan R., Vincenzi, Fabrizio, Varani, Katia, Borea, Pier Andrea
Published in Bioorganic & medicinal chemistry (15.01.2012)
Published in Bioorganic & medicinal chemistry (15.01.2012)
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Journal Article
Synthesis and Biological Evaluation of Novel 1-Deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]- 9H-purin-9-yl]-N-ethyl-β-d-ribofuranuronamide Derivatives as Useful Templates for the Development of A2B Adenosine Receptor Agonists
Baraldi, Pier Giovanni, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Fruttarolo, Francesca, Romagnoli, Romeo, Carrion, Maria Dora, Cara, Luisa Carlota Lopez, Moorman, Allan R., Varani, Katia, Borea, Pier Andrea
Published in Journal of medicinal chemistry (25.01.2007)
Published in Journal of medicinal chemistry (25.01.2007)
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Journal Article
New strategies for the synthesis of A3 adenosine receptor antagonists
BARALDI, Pier Giovanni, BOVERO, Andrea, FRUTTAROLO, Francesca, ROMAGNOLI, Romeo, MOJGAN AGHAZADEH TABRIZI, PRETI, Delia, VARANI, Katia, BOREA, Pier Andrea, MOORMAN, Allan R
Published in Bioorganic & medicinal chemistry (15.09.2003)
Published in Bioorganic & medicinal chemistry (15.09.2003)
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Journal Article
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists
Tabrizi, Mojgan Aghazadeh, Baraldi, Pier Giovanni, Preti, Delia, Romagnoli, Romeo, Saponaro, Giulia, Baraldi, Stefania, Moorman, Allan R, Zaid, Abdel Naser, Varani, Katia, Borea, Pier Andrea
Published in Bioorganic & medicinal chemistry (01.03.2008)
Published in Bioorganic & medicinal chemistry (01.03.2008)
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Journal Article
1,3-Dipropyl-8-(1 -phenylacetamide-1Η-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists
AGHAZADEH TABRIZI, Mojgan, GIOVANNI BARALDI, Pier, PRETI, Delia, ROMAGNOLI, Romeo, SAPONARO, Giulia, BARALDI, Stefania, MOORMAN, Allan R, NASER ZAID, Abdel, VARANI, Katia, BOREA, Pier Andrea
Published in Bioorganic & medicinal chemistry (01.03.2008)
Published in Bioorganic & medicinal chemistry (01.03.2008)
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