INTERLEUKIN-10 AND THE INTERLEUKIN-10 RECEPTOR
Moore, Kevin W, de Waal Malefyt, Rene, Coffman, Robert L, O'Garra, Anne
Published in Annual review of immunology (01.01.2001)
Published in Annual review of immunology (01.01.2001)
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IL-10 acts on the antigen-presenting cell to inhibit cytokine production by Th1 cells
Fiorentino, DF, Zlotnik, A, Vieira, P, Mosmann, TR, Howard, M, Moore, KW, O'Garra, A
Published in The Journal of immunology (1950) (15.05.1991)
Published in The Journal of immunology (1950) (15.05.1991)
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Interleukin 10 : a novel stimulatory factor for mast cells and their progenitors
THOMPSON-SNIPES, L, DHAR, V, BOND, M. W, MOSMANN, T. R, MOORE, K. W, RENNICK, D. M
Published in The Journal of experimental medicine (01.02.1991)
Published in The Journal of experimental medicine (01.02.1991)
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Isolation and Expression of Human Cytokine Synthesis Inhibitory Factor cDNA Clones: Homology to Epstein-Barr Virus Open Reading Frame BCRFI
Vieira, P., de Waal-Malefyt, R., M.-N. Dang, Johnson, K. E., Kastelein, R., Fiorention, D. F., de Vries, J. E., M.-G. Roncarolo, Mosmann, T. R., Moore, K. W.
Published in Proceedings of the National Academy of Sciences - PNAS (15.02.1991)
Published in Proceedings of the National Academy of Sciences - PNAS (15.02.1991)
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4-Amido-2-carboxytetrahydroquinolines. Structure-activity relationships for antagonism at the glycine site of the NMDA receptor
Leeson, Paul D, Carling, Robert W, Moore, Kevin W, Moseley, Angela M, Smith, Julian D, Stevenson, Graeme, Chan, Tony, Baker, Raymond, Foster, Alan C
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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A Receptor for the Heterodimeric Cytokine IL-23 Is Composed of IL-12R beta 1 and a Novel Cytokine Receptor Subunit, IL-23R
Parham, C, Chirica, M, Timans, J, Vaisberg, E, Travis, M, Cheung, J, Pflanz, S, Zhang, R, Singh, K P, Vega, F, To, W, Wagner, J, O'Farrell, A, McClanahan, T, Zurawski, S, Hannum, C, Gorman, D, Rennick, D M, Kastelein, R A, de Waal Malefyt, R, Moore, K W
Published in The Journal of immunology (1950) (01.06.2002)
Published in The Journal of immunology (1950) (01.06.2002)
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Novel p19 Protein Engages IL-12p40 to Form a Cytokine, IL-23, with Biological Activities Similar as Well as Distinct from IL-12
Oppmann, Birgit, Lesley, Robin, Blom, Bianca, Timans, Jackie C, Xu, Yuming, Hunte, Brisdell, Vega, Felix, Yu, Nancy, Wang, Jing, Singh, Komal, Zonin, Francesca, Vaisberg, Elena, Churakova, Tatyana, Liu, Man-ru, Gorman, Daniel, Wagner, Janet, Zurawski, Sandra, Liu, Yong-Jun, Abrams, John S, Moore, Kevin W, Rennick, Donna, de Waal-Malefyt, Rene, Hannum, Charles, Bazan, J.Fernando, Kastelein, Robert A
Published in Immunity (Cambridge, Mass.) (01.11.2000)
Published in Immunity (Cambridge, Mass.) (01.11.2000)
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3-phenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[3,4-alpha]phthalazines and analogues: High-affinity gamma-aminobutyric acid-A benzodiazepine receptor ligands with alpha 2, alpha 3, and alpha 5-subtype binding selectivity over alpha 1
Carling, RW, Moore, KW, Street, LJ, Wild, D, Isted, C, Leeson, PD, Thomas, S, O'Connor, D, McKernan, RM, Quirk, K, Cook, SM, Atack, Wafford, KA, Thompson, SA, Dawson, GR, Ferris, P, Castro, JL
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
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Selective, orally active gamma-aminobutyric acid(A) alpha 5 receptor inverse agonists as cognition enhancers
Sternfeld, F, Carling, RW, Jelley, RA, Ladduwahetty, T, Merchant, KJ, Moore, KW, Reeve, AJ, Street, LJ, O'Connor, D, Sohal, B, Atack, Cook, S, Seabrook, G, Wafford, K, Tattersall, FD, Collinson, N, Dawson, GR, Castro, JL, MacLeod, AM
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Synthesis and biological evaluation of 3-heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4-a]phthalazines and analogues as subtype-selective inverse agonists for the GABA(A)alpha 5 benzodiazepine binding site
Street, LJ, Sternfeld, F, Jelley, RA, Reeve, AJ, Carling, RW, Moore, KW, McKernan, RM, Sohal, B, Cook, S, Pike, A, Dawson, GR, Bromidge, FA, Wafford, KA, Seabrook, GR, Thompson, SA, Marshall, G, Pillai, GV, Castro, JL, Atack, MacLeod, AM
Published in Journal of medicinal chemistry (01.07.2004)
Published in Journal of medicinal chemistry (01.07.2004)
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7-(1,1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine: A functionally selective gamma-aminobutyric acid(A) (GABA(A)) alpha 2/alpha 3-subtype selective agonist that exhibits potent anxiolytic activity but is not sedating in animal models
Carling, RW, Madin, A, Guiblin, A, Russell, MGN, Moore, KW, Mitchinson, A, Sohal, B, Pike, A, Cook, SM, Ragan, IC, McKernan, RM, Quirk, K, Ferris, P, Marshall, G, Thompson, SA, Wafford, KA, Dawson, GR, Atack, Harrison, T, Castro, JL, Street, LJ
Published in Journal of medicinal chemistry (17.11.2005)
Published in Journal of medicinal chemistry (17.11.2005)
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Multivalent avimer proteins evolved by exon shuffling of a family of human receptor domains
Silverman, Joshua, Stemmer, Willem Pim C, Lu, Qiang, Bakker, Alice, To, Wayne, Duguay, Amy, Alba, Ben M, Smith, Richard, Rivas, Alberto, Li, Peng, Le, Hon, Whitehorn, Erik, Moore, Kevin W, Swimmer, Candace, Perlroth, Victor, Vogt, Martin, Kolkman, Joost
Published in Nature biotechnology (01.12.2005)
Published in Nature biotechnology (01.12.2005)
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Discovery of functionally selective 7,8,9,10-tetrahydro-7,10-ethano-1,2,4-triazolo[3,4-a]phthalazines as GABA(A) receptor agonists at the alpha(3) subunit
Russell, MGN, Carling, RW, Atack, Bromidge, FA, Cook, SM, Hunt, P, Isted, C, Lucas, M, McKernan, RM, Mitchinson, A, Moore, KW, Narquizian, R, Macaulay, AJ, Thomas, D, Thompson, SA, Wafford, KA, Castro, JL
Published in Journal of medicinal chemistry (10.03.2005)
Published in Journal of medicinal chemistry (10.03.2005)
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Lymphotactin: A Cytokine That Represents a New Class of Chemokine
Kelner, Gregory S., Kennedy, Jacqueline, Bacon, Kevin B., Kleyensteuber, Sarah, Largaespada, David A., Jenkins, Nancy A., Copeland, Neal G., Bazan, J. Fernando, Moore, Kevin W., Schall, Thomas J., Zlotnik, Albert
Published in Science (American Association for the Advancement of Science) (25.11.1994)
Published in Science (American Association for the Advancement of Science) (25.11.1994)
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The EBV IL-10 homologue is a selective agonist with impaired binding to the IL-10 receptor
Liu, Y, de Waal Malefyt, R, Briere, F, Parham, C, Bridon, JM, Banchereau, J, Moore, KW, Xu, J
Published in The Journal of immunology (1950) (15.01.1997)
Published in The Journal of immunology (1950) (15.01.1997)
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IL-10, a novel growth cofactor for mature and immature T cells
MacNeil, IA, Suda, T, Moore, KW, Mosmann, TR, Zlotnik, A
Published in The Journal of immunology (1950) (15.12.1990)
Published in The Journal of immunology (1950) (15.12.1990)
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Homology of Cytokine Synthesis Inhibitory Factor (IL-10) to the Epstein-Barr Virus Gene BCRFI
Moore, Kevin W., Vieira, Paulo, Fiorentino, David F., Trounstine, Mary L., Khan, Tariq A., Mosmann, Timothy R.
Published in Science (American Association for the Advancement of Science) (08.06.1990)
Published in Science (American Association for the Advancement of Science) (08.06.1990)
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Expression cloning and characterization of a human IL-10 receptor
Liu, Y, Wei, SH, Ho, AS, de Waal Malefyt, R, Moore, KW
Published in The Journal of immunology (1950) (15.02.1994)
Published in The Journal of immunology (1950) (15.02.1994)
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IL-18 Receptors, Their Role in Ligand Binding and Function: Anti-IL-1RAcPL Antibody, a Potent Antagonist of IL-18
Debets, Reno, Timans, Jackie C, Churakowa, Tatyana, Zurawski, Sandra, de Waal Malefyt, Rene, Moore, Kevin W, Abrams, John S, O'Garra, Anne, Bazan, J. Fernando, Kastelein, Robert A
Published in The Journal of immunology (1950) (01.11.2000)
Published in The Journal of immunology (1950) (01.11.2000)
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