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Year of Publication 12.11.2014
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Year of Publication 12.11.2014
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LOKE PUI LENG, MONTALBETTI CHRISTIAN A.G.N, FENG JIANWEN, STABEN STEVEN
Year of Publication 05.12.2013
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Discovery of a Novel Hsp90 Inhibitor by Fragment Linking
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Design, synthesis and structure-activity relationships of a novel class of sulfonylpyridine inhibitors of Interleukin-2 inducible T-cell kinase (ITK)
Trani, Giancarlo, Barker, John J., Bromidge, Steven M., Brookfield, Frederick A., Burch, Jason D., Chen, Yuan, Eigenbrot, Charles, Heifetz, Alexander, Ismaili, M. Hicham A., Johnson, Adam, Krulle, Thomas M., MacKinnon, Colin H., Maghames, Rosemary, McEwan, Paul A., Montalbetti, Christian A. G. N., Ortwine, Daniel F., Perez-Fuertes, Yolanda, Vaidya, Darshan G., Wang, Xiaolu, Zarrin, Ali A., Pei, Zhonghua
Published in Bioorganic & medicinal chemistry letters (15.12.2014)
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Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2-Amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one Oxime
Amici, Raffaella, Bigogno, Chiara, Boggio, Roberto, Colombo, Andrea, Courtney, Stephen M., Dal Zuffo, Roberto, Dondio, Giulio, Fusar, Fulvia, Gagliardi, Stefania, Minucci, Saverio, Molteni, Marco, Montalbetti, Christian A. G. N., Mortoni, Annalisa, Varasi, Mario, Vultaggio, Stefania, Mercurio, Ciro
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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Fragment‐based Identification of Hsp90 Inhibitors
Barker, John J., Barker, Oliver, Boggio, Roberto, Chauhan, Viddhata, Cheng, Robert K. Y., Corden, Vincent, Courtney, Stephen M., Edwards, Neil, Falque, Virginie M., Fusar, Fulvia, Gardiner, Mihaly, Hamelin, Estelle M. N., Hesterkamp, Thomas, Ichihara, Osamu, Jones, Richard S., Mather, Owen, Mercurio, Ciro, Minucci, Saverio, Montalbetti, Christian A. G. N., Müller, Annett, Patel, Deepti, Phillips, Banu G., Varasi, Mario, Whittaker, Mark, Winkler, Dirk, Yarnold, Christopher J.
Published in ChemMedChem (08.06.2009)
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HCV NS5B polymerase inhibitors 2: Synthesis and in vitro activity of (1,1-dioxo-2H-[1,2,4]benzothiadiazin-3-yl) azolo[1,5-a]pyridine and azolo[1,5-a]pyrimidine derivatives
Wang, Guangyi, Lei, Huoxing, Wang, Xiaofang, Das, Debasis, Hong, Jian, Mackinnon, Colin H., Coulter, Thomas S., Montalbetti, Christian A.G.N., Mears, Richard, Gai, Xinjie, Bailey, Sarah E., Ruhrmund, Donald, Hooi, Lisa, Misialek, Shawn, Rajagopalan, P.T. Ravi, Cheng, Robert K.Y., Barker, John J., Felicetti, Brunella, Schönfeld, Dorian L., Stoycheva, Antitsa, Buckman, Brad O., Kossen, Karl, Seiwert, Scott D., Beigelman, Leonid
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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compostos de álcool propargílico 6,5-heterocíclico e uso dos mesmos
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Year of Publication 13.12.2016
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Year of Publication 13.12.2016
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TRICYCLIC COMPOUNDS AND METHODS OF USE THEREFOR
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Year of Publication 31.12.2015
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