Pharmacological agents acting at subtypes of metabotropic glutamate receptors
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Journal Article
Broad spectrum efficacy with LY2969822, an oral prodrug of metabotropic glutamate 2/3 receptor agonist LY2934747, in rodent pain models
Johnson, Michael P, Muhlhauser, Mark A, Nisenbaum, Eric S, Simmons, Rosa M A, Forster, Beth M, Knopp, Kelly L, Yang, Lijuan, Morrow, Denise, Li, Dominic L, Kennedy, Jeffrey D, Swanson, Steven, Monn, James A
Published in British journal of pharmacology (01.05.2017)
Published in British journal of pharmacology (01.05.2017)
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Journal Article
Preclinical predictors that the orthosteric mGlu2/3 receptor antagonist LY3020371 will not engender ketamine-associated neurotoxic, motor, cognitive, subjective, or abuse-liability-related effects
Witkin, J M, Monn, J A, Li, J, Johnson, B, McKinzie, D L, Wang, X-S, Heinz, B A, Li, R, Ornstein, P L, Smith, S C, Mitch, C H, Calligaro, D O, Swanson, S, Allen, D, Phillips, K, Gilmour, G
Published in Pharmacology, biochemistry and behavior (01.04.2017)
Published in Pharmacology, biochemistry and behavior (01.04.2017)
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Journal Article
Discovery of allosteric potentiators for the metabotropic glutamate 2 receptor: Synthesis and subtype selectivity of N-(4-(2-methoxyphenoxy)phenyl)-N-(2,2,2-trifluoroethylsulfonyl)pyrid-3-ylmethyl-amine
Johnson, MP, Baez, M, Jagdmann, GE, Britton, TC, Large, TH, Callagaro, DO, Tizzano, JP, Monn, JA, Schoepp, DD
Published in Journal of medicinal chemistry (17.07.2003)
Published in Journal of medicinal chemistry (17.07.2003)
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Journal Article
The Metabotropic Glutamate 2/3 Receptor Agonists LY354740 and LY379268 Selectively Attenuate Phencyclidine versus d-Amphetamine Motor Behaviors in Rats
Cartmell, J, Monn, J A, Schoepp, D D
Published in The Journal of pharmacology and experimental therapeutics (01.10.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.10.1999)
Journal Article
Physiological antagonism between 5-hydroxytryptamine(2A) and group II metabotropic glutamate receptors in prefrontal cortex
Marek, G J, Wright, R A, Schoepp, D D, Monn, J A, Aghajanian, G K
Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
Journal Article
Synthesis and Metabotropic Glutamate Receptor Activity of S-Oxidized Variants of (−)-4-Amino-2-thiabicyclo-[3.1.0]hexane-4,6-dicarboxylate: Identification of Potent, Selective, and Orally Bioavailable Agonists for mGlu2/3 Receptors
Monn, James A., Massey, Steven M., Valli, Matthew J., Henry, Steven S., Stephenson, Gregory A., Bures, Mark, Hérin, Marc, Catlow, John, Giera, Deborah, Wright, Rebecca A., Johnson, Bryan G., Andis, Sherri L., Kingston, Ann, Schoepp, Darryle D.
Published in Journal of medicinal chemistry (25.01.2007)
Published in Journal of medicinal chemistry (25.01.2007)
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Journal Article
Analgesic effects of the selective group II (mGlu2/3) metabotropic glutamate receptor agonists LY379268 and LY389795 in persistent and inflammatory pain models after acute and repeated dosing
Jones, Carrie K., Eberle, Elizabeth Lutz, Peters, Stephen C., Monn, James A., Shannon, Harlan E.
Published in Neuropharmacology (2005)
Published in Neuropharmacology (2005)
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Journal Article
Anxiolytic and Side-Effect Profile of LY354740: A Potent, Highly Selective, Orally Active Agonist for Group II Metabotropic Glutamate Receptors
Helton, D R, Tizzano, J P, Monn, J A, Schoepp, D D, Kallman, M J
Published in The Journal of pharmacology and experimental therapeutics (01.02.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1998)
Journal Article
Synthesis, Pharmacological Characterization, and Molecular Modeling of Heterobicyclic Amino Acids Related to (+)-2-Aminobicyclo[3.1.0]hexane- 2,6-dicarboxylic Acid (LY354740): Identification of Two New Potent, Selective, and Systemically Active Agonists for Group II Metabotropic Glutamate Receptors
Monn, James A, Valli, Matthew J, Massey, Steven M, Hansen, Marvin M, Kress, Thomas J, Wepsiec, James P, Harkness, Allen R, Grutsch, John L, Wright, Rebecca A, Johnson, Bryan G, Andis, Sherri L, Kingston, Ann, Tomlinson, Rosemarie, Lewis, Richard, Griffey, Kelly R, Tizzano, Joseph P, Schoepp, Darryle D
Published in Journal of medicinal chemistry (25.03.1999)
Published in Journal of medicinal chemistry (25.03.1999)
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Journal Article
Methyl Substitution of 2-Aminobicyclo[3.1.0]hexane 2,6-Dicarboxylate (LY354740) Determines Functional Activity at Metabotropic Glutamate Receptors: Identification of a Subtype Selective mGlu2 Receptor Agonist
Dominguez, Carmen, Prieto, Lourdes, Valli, Matthew J, Massey, Steven M, Bures, Mark, Wright, Rebecca A, Johnson, Bryan G, Andis, Sherri L, Kingston, Ann, Schoepp, Darryle D, Monn, James A
Published in Journal of medicinal chemistry (19.05.2005)
Published in Journal of medicinal chemistry (19.05.2005)
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Journal Article
Design, Synthesis, and Pharmacological Characterization of (+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid (LY354740): A Potent, Selective, and Orally Active Group 2 Metabotropic Glutamate Receptor Agonist Possessing Anticonvulsant and Anxiolytic Properties
Monn, James A, Valli, Matthew J, Massey, Steven M, Wright, Rebecca A, Salhoff, Craig R, Johnson, Bryan G, Howe, Trevor, Alt, Charles A, Rhodes, Gary A, Robey, Roger L, Griffey, Kelly R, Tizzano, Joseph P, Kallman, Mary J, Helton, David R, Schoepp, Darryle D
Published in Journal of medicinal chemistry (14.02.1997)
Published in Journal of medicinal chemistry (14.02.1997)
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Journal Article
Dipeptides as Effective Prodrugs of the Unnatural Amino Acid (+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid (LY354740), a Selective Group II Metabotropic Glutamate Receptor Agonist
Bueno, Ana Belén, Collado, Iván, de Dios, Alfonso, Domínguez, Carmen, Martín, José Alfredo, Martín, Luisa M, Martínez-Grau, María Angeles, Montero, Carlos, Pedregal, Concepción, Catlow, John, Coffey, D. Scott, Clay, Michael P, Dantzig, Anne H, Lindstrom, Terry, Monn, James A, Jiang, Haiyan, Schoepp, Darryle D, Stratford, Robert E, Tabas, Linda B, Tizzano, Joseph P, Wright, Rebecca A, Herin, Marc F
Published in Journal of medicinal chemistry (11.08.2005)
Published in Journal of medicinal chemistry (11.08.2005)
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Journal Article
Neuroprotective Effects of LY379268, a Selective mGlu2/3 Receptor Agonist: Investigations into Possible Mechanism of Action In Vivo
Bond, A, Jones, N M, Hicks, C A, Whiffin, G M, Ward, M A, O'Neill, M F, Kingston, A E, Monn, J A, Ornstein, P L, Schoepp, D D, Lodge, D, O'Neill, M J
Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
Journal Article
LY354740 is a potent and highly selective group II metabotropic glutamate receptor agonist in cells expressing human glutamate receptors
SCHOEPP, D. D, JOHNSON, B. G, MONN, J. A, WRIGHT, R. A, SALHOFF, C. R, MAYNE, N. G, WU, S, COCKERHAM, S. L, BURNETT, J. P, BELEGAJE, R, BLEAKMAN, D
Published in Neuropharmacology (1997)
Published in Neuropharmacology (1997)
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Journal Article