Architecture of a single membrane spanning cytochrome P450 suggests constraints that orient the catalytic domain relative to a bilayer
Monk, Brian C., Tomasiak, Thomas M., Keniya, Mikhail V., Huschmann, Franziska U., Tyndall, Joel D. A., O'Connell, Joseph D., Cannon, Richard D., McDonald, Jeffrey G., Rodriguez, Andrew, Finer-Moore, Janet S., Stroud, Robert M.
Published in Proceedings of the National Academy of Sciences - PNAS (11.03.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (11.03.2014)
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Journal Article
Efflux-Mediated Antifungal Drug Resistance
CANNON, Richard D, LAMPING, Erwin, HOLMES, Ann R, NIIMI, Kyoko, BARET, Philippe V, KENIYA, Mikhail V, TANABE, Koichi, NIIMI, Masakazu, GOFFEAU, Andre, MONK, Brian C
Published in Clinical Microbiology Reviews (01.04.2009)
Published in Clinical Microbiology Reviews (01.04.2009)
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Journal Article
Outwitting Multidrug Resistance to Antifungals
Monk, Brian C, Goffeau, Andre
Published in Science (American Association for the Advancement of Science) (18.07.2008)
Published in Science (American Association for the Advancement of Science) (18.07.2008)
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Journal Article
Structural and Functional Elucidation of Yeast Lanosterol 14α-Demethylase in Complex with Agrochemical Antifungals
Tyndall, Joel D A, Sabherwal, Manya, Sagatova, Alia A, Keniya, Mikhail V, Negroni, Jacopo, Wilson, Rajni K, Woods, Matthew A, Tietjen, Klaus, Monk, Brian C
Published in PloS one (01.12.2016)
Published in PloS one (01.12.2016)
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Journal Article
The Monoamine Oxidase A Inhibitor Clorgyline Is a Broad-Spectrum Inhibitor of Fungal ABC and MFS Transporter Efflux Pump Activities Which Reverses the Azole Resistance of Candida albicans and Candida glabrata Clinical Isolates
HOLMES, Ann R, KENIYA, Mikhail V, IVNITSKI-STEELE, Irena, MONK, Brian C, LAMPING, Erwin, SKLAR, Larry A, CANNON, Richard D
Published in Antimicrobial Agents and Chemotherapy (01.03.2012)
Published in Antimicrobial Agents and Chemotherapy (01.03.2012)
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Journal Article
Exploring Cryptococcus neoformans CYP51 and Its Cognate Reductase as a Drug Target
Ruma, Yasmeen N, Keniya, Mikhail V, Monk, Brian C
Published in Journal of fungi (Basel) (28.11.2022)
Published in Journal of fungi (Basel) (28.11.2022)
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Journal Article
ABC Transporter Cdr1p Contributes More than Cdr2p Does to Fluconazole Efflux in Fluconazole-Resistant Candida albicans Clinical Isolates
HOLMES, Ann R, LIN, Ya-Hsun, NIIMI, Kyoko, LAMPING, Erwin, KENIYA, Mikhail, NIIMI, Masakazu, TANABE, Koichi, MONK, Brian C, CANNON, Richard D
Published in Antimicrobial Agents and Chemotherapy (01.11.2008)
Published in Antimicrobial Agents and Chemotherapy (01.11.2008)
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Journal Article
Protein content of molar–incisor hypomineralisation enamel
Farah, Rami A, Monk, Brian C, Swain, Michael V, Drummond, Bernadette K
Published in Journal of dentistry (01.07.2010)
Published in Journal of dentistry (01.07.2010)
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Journal Article
Identification of Nile red as a fluorescent substrate of the Candida albicans ATP-binding cassette transporters Cdr1p and Cdr2p and the major facilitator superfamily transporter Mdr1p
Ivnitski-Steele, Irena, Holmes, Ann R., Lamping, Erwin, Monk, Brian C., Cannon, Richard D., Sklar, Larry A.
Published in Analytical biochemistry (01.11.2009)
Published in Analytical biochemistry (01.11.2009)
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Journal Article
Fungal PDR transporters: Phylogeny, topology, motifs and function
Lamping, Erwin, Baret, Philippe V., Holmes, Ann R., Monk, Brian C., Goffeau, Andre, Cannon, Richard D.
Published in Fungal genetics and biology (01.02.2010)
Published in Fungal genetics and biology (01.02.2010)
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Journal Article
Characterization of Three Classes of Membrane Proteins Involved in Fungal Azole Resistance by Functional Hyperexpression in Saccharomyces cerevisiae
Lamping, Erwin, Monk, Brian C, Niimi, Kyoko, Holmes, Ann R, Tsao, Sarah, Tanabe, Koichi, Niimi, Masakazu, Uehara, Yoshimasa, Cannon, Richard D
Published in Eukaryotic Cell (01.07.2007)
Published in Eukaryotic Cell (01.07.2007)
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Journal Article
[Fe₂L₃]⁴⁺ cylinders derived from bis(bidentate) 2-pyridyl-1,2,3-triazole "click" ligands: synthesis, structures and exploration of biological activity
Vellas, Sreedhar K, Lewis, James E M, Shankar, Madhu, Sagatova, Alia, Tyndall, Joel D A, Monk, Brian C, Fitchett, Christopher M, Hanton, Lyall R, Crowley, James D
Published in Molecules (Basel, Switzerland) (29.05.2013)
Published in Molecules (Basel, Switzerland) (29.05.2013)
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Journal Article
Specific interactions between the Candida albicans ABC transporter Cdr1p ectodomain and a d-octapeptide derivative inhibitor
Niimi, Kyoko, Harding, David R. K., Holmes, Ann R., Lamping, Erwin, Niimi, Masakazu, Tyndall, Joel D. A., Cannon, Richard D., Monk, Brian C.
Published in Molecular microbiology (01.08.2012)
Published in Molecular microbiology (01.08.2012)
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Journal Article