Synthesis and biological evaluation of novel hexahydro-pyrido[3',2':4,5]pyrrolo[1,2 -a]pyrazines as potent and selective 5-HT2C receptor agonists
RICHTER, Hans G. F, ADAMS, D. R, KNIGHT, A. R, MALCOLM, C. S, MATTEI, P, MISRA, A, MIZRAHI, J, MONCK, N. J. T, PLANCHER, J.-M, ROEVER, S, ROFFEY, J. R. A, TAYLOR, S, BENARDEAU, A, VICKERS, S. P, BICKERDIKE, M. J, BENTLEY, J. M, BLENCH, T. J, CLIFFE, I. A, DOURISH, C, HEBEISEN, P, KENNETT, G. A
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Indoline derivatives as 5-HT2C receptor agonists
BENTLEY, J. M, ADAMS, D. R, GEORGE, A. R, GILES, P. R, HAMLYN, R. J, KENNETT, G. A, KNIGHT, A. R, MALCOLM, C. S, MANSELL, H. L, MISRA, A, MONCK, N. J. T, PRATT, R. M, BEBBINGTON, D, QUIRK, K, ROFFEY, J. R. A, VICKERS, S. P, CLIFFE, I. A, BENWELL, K. R, BICKERDIKE, M. J, DAVIDSON, J. E. P, DAWSON, C. E, DOURISH, C. T, DUNCTON, M. A. J, GAUR, S
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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3,5-Disubstituted-4-hydroxyphenyls Linked to 3-Hydroxy-2-methyl- 4(1H)-pyridinone: Potent Inhibitors of Lipid Peroxidation and Cell Toxicity
Bebbington, David, Monck, Nathaniel J. T, Gaur, Suneel, Palmer, Alan M, Benwell, Karen, Harvey, Victoria, Malcolm, Craig S, Porter, Richard H. P
Published in Journal of medicinal chemistry (27.07.2000)
Published in Journal of medicinal chemistry (27.07.2000)
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Synthesis and biological evaluation of novel hexahydro- pyrido[3',2':4,5]pyrrolo[1,2-a]pyrazines as potent and selective 5-HT sub(2C) receptor agonists
Richter, Hans GF, Adams, DR, Benardeau, A, Bickerdike, MJ, Bentley, J M, Blench, T J, Cliffe, IA, Dourish, C, Hebeisen, P, Kennett, G A, Knight, A R, Malcolm, C S, Mattei, P, Misra, A, Mizrahi, J, Monck, NJT, Plancher, J-M, Roever, S, Roffey, JRA, Taylor, S, Vickers, S P
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
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Journal Article
3,5-Disubstituted-4-hydroxyphenyls Linked to 3-Hydroxy-2-methyl-4(1H)-pyridinone: Potent Inhibitors of Lipid Peroxidation and Cell Toxicity
Bebbington, David, Monck, Nathaniel J. T, Gaur, Suneel, Palmer, Alan M, Benwell, Karen, Harvey, Victoria, Malcolm, Craig S, Porter, Richard H. P
Published in Journal of medicinal chemistry (30.11.2000)
Published in Journal of medicinal chemistry (30.11.2000)
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