New imide 5-HT1A receptor ligands - modification of terminal fragment geometry
Bojarski, Andrzej J, Mokrosz, Maria J, Duszyńska, Beata, Kozioł, Aneta, Bugno, Ryszard
Published in Molecules (Basel, Switzerland) (28.02.2004)
Published in Molecules (Basel, Switzerland) (28.02.2004)
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Biologically Active 1-Arylpiperazines. Synthesis of New N-(4-Aryl-1-piperazinyl)alkyl Derivatives of Quinazolidin-4(3H)-one, 2,3-Dihydrophthalazine-1,4-dione and 1,2-Dihydropyridazine-3,6-dione as Potential Serotonin Receptor Ligands
Kowalski, Piotr, Kowalska, Teresa, Mokrosz, Maria J., Bojarski, Andrzej J., Charakchieva-Minol, Sijka
Published in Molecules (Basel, Switzerland) (01.09.2001)
Published in Molecules (Basel, Switzerland) (01.09.2001)
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On the Bioactive Conformation of NAN-190 (1) and MP3022 (2), 5-HT1A Receptor Antagonists
Paluchowska, Maria H, Mokrosz, Maria J, Bojarski, Andrzej, Wesołowska, Anna, Borycz, Jolanta, Charakchieva-Minol, Sijka, Chojnacka-Wójcik, Ewa
Published in Journal of medicinal chemistry (02.12.1999)
Published in Journal of medicinal chemistry (02.12.1999)
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The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT1A/5-HT2A receptor activities of its 1-adamantoyloaminoalkyl derivatives
BOJARSKI, Andrzej J, MOKROSZ, Maria J, MINOL, Sijka Charakchieva, KOZIOŁ, Aneta, WESOŁOWSKA, Anna, TATARCZYNSKA, Ewa, KŁODZINSKA, Aleksandra, CHOJNACKA-WOJCIK, Ewa
Published in Bioorganic & medicinal chemistry (2002)
Published in Bioorganic & medicinal chemistry (2002)
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Application of Similarity Matrices and Genetic Neural Networks in Quantitative Structure−Activity Relationships of 2- or 4-(4-Methylpiperazino)pyrimidines: 5-HT2A Receptor Antagonists
Borowski, Tomasz, Król, Marcin, Brocławik, Ewa, Baranowski, Timothy C, Strekowski, Lucjan, Mokrosz, Maria J
Published in Journal of medicinal chemistry (18.05.2000)
Published in Journal of medicinal chemistry (18.05.2000)
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Influence of the terminal amide fragment geometry in some 3-arylideneindolin-2(1H)-ones on their 5-HT1A/5-HT2A receptor activity
MOKROSZ, Maria J, CHARAKCHIEVA-MINOL, Sijka, KOZIOŁ, Aneta, KŁODZINSKA, Aleksandra, CHOJNACKA-WOJCIK, Ewa
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
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8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl)]butyl]-8-azaspiro[4.5]decane-7,9-dione: A New 5-HT1A Receptor Ligand with the Same Activity Profile as Buspirone
Mokrosz, Jerzy L, Dereń-Wesołek, Anna, Tatarczyńska, Ewa, Duszyńska, Beata, Bojarski, Andrzej J, Mokrosz, Maria J, Chojnacka-Wójcik, Ewa
Published in Journal of medicinal chemistry (01.03.1996)
Published in Journal of medicinal chemistry (01.03.1996)
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Stereoelectronic factors in the interaction with DNA of small aromatic molecules substituted with a short cationic chain: Importance of the polarity of the aromatic system of the molecule
Strekowski, Lucjan, Mokrosz, Jerzy L, Wilson, W. David, Mokrosz, Maria J, Strekowski, Alewtina
Published in Biochemistry (Easton) (10.11.1992)
Published in Biochemistry (Easton) (10.11.1992)
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Addition and substitution reactions of chloropyrimidines with lithium reagents
Harden, Donald B, Mokrosz, Maria J, Strekowski, Lucjan
Published in Journal of organic chemistry (01.08.1988)
Published in Journal of organic chemistry (01.08.1988)
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Structure-Activity Relationship Studies of Central Nervous System Agents. 13.4-[3-(Benzotriazol-1-yl)propyl]-1-(2-methoxyphenyl)piperazine, a New Putative 5-HT1A Receptor Antagonist, and Its Analogs
Mokrosz, Jerzy L, Paluchowska, Maria H, Chojnacka-Wojcik, Ewa, Filip, Malgorzata, Charakchieva-Minol, Sijka, Deren-Wesolek, Anna, Mokrosz, Maria J
Published in Journal of medicinal chemistry (01.08.1994)
Published in Journal of medicinal chemistry (01.08.1994)
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Quantitative structure-activity relationship analysis of cation-substituted polyaromatic compounds as potentiators (amplifiers) of bleomycin-mediated degradation of DNA
Strekowski, Lucjan, Wilson, W. David, Mokrosz, Jerzy L, Mokrosz, Maria J, Harden, Donald B, Tanious, Farial A, Wydra, Roman L, Crow, Sidney A
Published in Journal of medicinal chemistry (01.02.1991)
Published in Journal of medicinal chemistry (01.02.1991)
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Novel 4-alkyl-1-arylpiperazines and 1,2,3,4-tetrahydroisoquinolines containing diphenylmethylamino or diphenylmethoxy fragment with differentiated 5-HT1A/5-HT2A/D2 receptor activity
Paluchowska, Maria H, Mokrosz, Maria J, Charakchieva-Minol, Sijka, Duszyńska, Beata, Kozioł, Aneta, Wesołowska, Anna, Stachowicz, Katarzyna, Chojnacka-Wójcik, Ewa
Published in Polish journal of pharmacology (01.07.2003)
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Published in Polish journal of pharmacology (01.07.2003)
Journal Article
The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT 1A/5-HT 2A receptor activities of its 1-adamantoyloaminoalkyl derivatives
Bojarski, Andrzej J, Mokrosz, Maria J, Minol, Sijka Charakchieva, Kozioł, Aneta, Wesołowska, Anna, Tatarczyńska, Ewa, Kłodzińska, Aleksandra, Chojnacka-Wójcik, Ewa
Published in Bioorganic & medicinal chemistry (2002)
Published in Bioorganic & medicinal chemistry (2002)
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Journal Article
The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT(1A)/5-HT(2A) receptor activities of its 1-adamantoyloaminoalkyl derivatives
Bojarski, Andrzej J, Mokrosz, Maria J, Minol, Sijka Charakchieva, Kozioł, Aneta, Wesołowska, Anna, Tatarczyńska, Ewa, Kłodzińska, Aleksandra, Chojnacka-Wójcik, Ewa
Published in Bioorganic & medicinal chemistry (01.01.2002)
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Published in Bioorganic & medicinal chemistry (01.01.2002)
Journal Article
Application of Similarity Matrices and Genetic Neural Networks in Quantitative Structure−Activity Relationships of 2- or 4-(4-Methylpiperazino)pyrimidines: 5-HT 2A Receptor Antagonists
Borowski, Tomasz, Król, Marcin, Brocławik, Ewa, Baranowski, Timothy C., Strekowski, Lucjan, Mokrosz, Maria J.
Published in Journal of medicinal chemistry (01.05.2000)
Published in Journal of medicinal chemistry (01.05.2000)
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Journal Article
Influence of the Terminal Amide Fragment Geometry in Some 3-Arylideneindolin-2(1 H)-ones on Their 5-HT 1A/5-HT 2A Receptor Activity
Mokrosz, Maria J, Charakchieva-Minol, Sijka, Kozioł, Aneta, Kłodzińska, Aleksandra, Chojnacka-Wójcik, Ewa
Published in Bioorganic & medicinal chemistry letters (2001)
Published in Bioorganic & medicinal chemistry letters (2001)
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STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF CENTRAL-NERVOUS-SYSTEM AGENTS .13. 4-[3-(BENZOTRIAZOL-1-YL)PROPYL]-1-(2-METHOXYPHENYL)PIPERAZINE, A NEW PUTATIVE 5-HT1A RECEPTOR ANTAGONIST, AND ITS ANALOGS
MOKROSZ, JL, PALUCHOWSKA, MH, CHOJNACKAWOJCIK, E, FILIP, M, CHARAKCHIEVAMINOL, S, DERENWESOLEK, A, MOKROSZ, MJ
Published in Journal of medicinal chemistry (19.08.1994)
Published in Journal of medicinal chemistry (19.08.1994)
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Structure-activity relationship analysis of substituted 4-quinolinamines, antagonists of immunostimulatory CpG-oligodeoxynucleotides
Strekowski, Lucjan, Zegrocka, Oliwia, Henary, Maged, Say, Martial, Mokrosz, Maria J., Kotecka, Barbara M., Manzel, Lori, Macfarlane, Donald E.
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
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