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Efficacy of Antiviral Agents against the SARS-CoV-2 Omicron Subvariant BA.2
Takashita, Emi, Kinoshita, Noriko, Yamayoshi, Seiya, Sakai-Tagawa, Yuko, Fujisaki, Seiichiro, Ito, Mutsumi, Iwatsuki-Horimoto, Kiyoko, Halfmann, Peter, Watanabe, Shinji, Maeda, Kenji, Imai, Masaki, Mitsuya, Hiroaki, Ohmagari, Norio, Takeda, Makoto, Hasegawa, Hideki, Kawaoka, Yoshihiro
Published in The New England journal of medicine (14.04.2022)
Published in The New England journal of medicine (14.04.2022)
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Efficacy of Antibodies and Antiviral Drugs against Covid-19 Omicron Variant
Takashita, Emi, Kinoshita, Noriko, Yamayoshi, Seiya, Sakai-Tagawa, Yuko, Fujisaki, Seiichiro, Ito, Mutsumi, Iwatsuki-Horimoto, Kiyoko, Chiba, Shiho, Halfmann, Peter, Nagai, Hiroyuki, Saito, Makoto, Adachi, Eisuke, Sullivan, David, Pekosz, Andrew, Watanabe, Shinji, Maeda, Kenji, Imai, Masaki, Yotsuyanagi, Hiroshi, Mitsuya, Hiroaki, Ohmagari, Norio, Takeda, Makoto, Hasegawa, Hideki, Kawaoka, Yoshihiro
Published in The New England journal of medicine (10.03.2022)
Published in The New England journal of medicine (10.03.2022)
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Syrian hamsters as a small animal model for SARS-CoV-2 infection and countermeasure development
Imai, Masaki, Iwatsuki-Horimoto, Kiyoko, Hatta, Masato, Loeber, Samantha, Halfmann, Peter J., Nakajima, Noriko, Watanabe, Tokiko, Ujie, Michiko, Takahashi, Kenta, Ito, Mutsumi, Yamada, Shinya, Fan, Shufang, Chiba, Shiho, Kuroda, Makoto, Guan, Lizheng, Takada, Kosuke, Armbrust, Tammy, Balogh, Aaron, Furusawa, Yuri, Okuda, Moe, Ueki, Hiroshi, Yasuhara, Atsuhiro, Sakai-Tagawa, Yuko, Lopes, Tiago J. S., Kiso, Maki, Yamayoshi, Seiya, Kinoshita, Noriko, Ohmagari, Norio, Hattori, Shin-ichiro, Takeda, Makoto, Mitsuya, Hiroaki, Krammer, Florian, Suzuki, Tadaki, Kawaoka, Yoshihiro
Published in Proceedings of the National Academy of Sciences - PNAS (14.07.2020)
Published in Proceedings of the National Academy of Sciences - PNAS (14.07.2020)
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Characterization and antiviral susceptibility of SARS-CoV-2 Omicron BA.2
Uraki, Ryuta, Kiso, Maki, Iida, Shun, Imai, Masaki, Takashita, Emi, Kuroda, Makoto, Halfmann, Peter J., Loeber, Samantha, Maemura, Tadashi, Yamayoshi, Seiya, Fujisaki, Seiichiro, Wang, Zhongde, Ito, Mutsumi, Ujie, Michiko, Iwatsuki-Horimoto, Kiyoko, Furusawa, Yuri, Wright, Ryan, Chong, Zhenlu, Ozono, Seiya, Yasuhara, Atsuhiro, Ueki, Hiroshi, Sakai-Tagawa, Yuko, Li, Rong, Liu, Yanan, Larson, Deanna, Koga, Michiko, Tsutsumi, Takeya, Adachi, Eisuke, Saito, Makoto, Yamamoto, Shinya, Hagihara, Masao, Mitamura, Keiko, Sato, Tetsuro, Hojo, Masayuki, Hattori, Shin-ichiro, Maeda, Kenji, Valdez, Riccardo, Okuda, Moe, Murakami, Jurika, Duong, Calvin, Godbole, Sucheta, Douek, Daniel C., Maeda, Ken, Watanabe, Shinji, Gordon, Aubree, Ohmagari, Norio, Yotsuyanagi, Hiroshi, Diamond, Michael S., Hasegawa, Hideki, Mitsuya, Hiroaki, Suzuki, Tadaki, Kawaoka, Yoshihiro
Published in Nature (London) (07.07.2022)
Published in Nature (London) (07.07.2022)
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Recent Drug Development and Medicinal Chemistry Approaches for the Treatment of SARS‐CoV‐2 Infection and COVID‐19
Ghosh, Arun K., Mishevich, Jennifer L., Mesecar, Andrew, Mitsuya, Hiroaki
Published in ChemMedChem (18.11.2022)
Published in ChemMedChem (18.11.2022)
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A novel highly quantitative and reproducible assay for the detection of anti-SARS-CoV-2 IgG and IgM antibodies
Noda, Kenta, Matsuda, Kouki, Yagishita, Shigehiro, Maeda, Kenji, Akiyama, Yutaro, Terada-Hirashima, Junko, Matsushita, Hiromichi, Iwata, Satoshi, Yamashita, Kazuto, Atarashi, Yusuke, Watanabe, Shunsuke, Ide, Nobuyuki, Yoshida, Tomokazu, Ohmagari, Norio, Mitsuya, Hiroaki, Hamada, Akinobu
Published in Scientific reports (04.03.2021)
Published in Scientific reports (04.03.2021)
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Third-Dose BNT162b2 Vaccination Elicits Markedly High-Level SARS-CoV-2–Neutralizing Antibodies in Vaccinees Who Responded Poorly to a Second Dose in Japan
Amano, Masayuki, Maeda, Kenji, Tsuchiya, Kiyoto, Shimada, Shinya, Mitsuya, Hiroaki
Published in The Journal of infectious diseases (28.11.2022)
Published in The Journal of infectious diseases (28.11.2022)
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Indole Chloropyridinyl Ester-Derived SARS-CoV‑2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure–Activity Relationship, and X‑ray Structural Studies
Ghosh, Arun K, Raghavaiah, Jakka, Shahabi, Dana, Yadav, Monika, Anson, Brandon J, Lendy, Emma K, Hattori, Shin-ichiro, Higashi-Kuwata, Nobuyo, Mitsuya, Hiroaki, Mesecar, Andrew D
Published in Journal of Medicinal Chemistry (14.10.2021)
Published in Journal of Medicinal Chemistry (14.10.2021)
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Correlates of neutralizing/SARS-CoV-2-S1-binding antibody response with adverse effects and immune kinetics in BNT162b2-vaccinated individuals
Maeda, Kenji, Amano, Masayuki, Uemura, Yukari, Tsuchiya, Kiyoto, Matsushima, Tomoko, Noda, Kenta, Shimizu, Yosuke, Fujiwara, Asuka, Takamatsu, Yuki, Ichikawa, Yasuko, Nishimura, Hidehiro, Kinoshita, Mari, Matsumoto, Shota, Gatanaga, Hiroyuki, Yoshimura, Kazuhisa, Oka, Shin-ichi, Mikami, Ayako, Sugiura, Wataru, Sato, Toshiyuki, Yoshida, Tomokazu, Shimada, Shinya, Mitsuya, Hiroaki
Published in Scientific reports (24.11.2021)
Published in Scientific reports (24.11.2021)
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A small molecule compound with an indole moiety inhibits the main protease of SARS-CoV-2 and blocks virus replication
Hattori, Shin-ichiro, Higashi-Kuwata, Nobuyo, Hayashi, Hironori, Allu, Srinivasa Rao, Raghavaiah, Jakka, Bulut, Haydar, Das, Debananda, Anson, Brandon J., Lendy, Emma K., Takamatsu, Yuki, Takamune, Nobutoki, Kishimoto, Naoki, Murayama, Kazutaka, Hasegawa, Kazuya, Li, Mi, Davis, David A., Kodama, Eiichi N., Yarchoan, Robert, Wlodawer, Alexander, Misumi, Shogo, Mesecar, Andrew D., Ghosh, Arun K., Mitsuya, Hiroaki
Published in Nature communications (28.01.2021)
Published in Nature communications (28.01.2021)
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Coronavirus Disease 2019 (COVID-19) Breakthrough Infection and Post-Vaccination Neutralizing Antibodies Among Healthcare Workers in a Referral Hospital in Tokyo: A Case-Control Matching Study
Yamamoto, Shohei, Maeda, Kenji, Matsuda, Kouki, Tanaka, Akihito, Horii, Kumi, Okudera, Kaori, Takeuchi, Junko S, Mizoue, Tetsuya, Konishi, Maki, Ozeki, Mitsuru, Sugiyama, Haruhito, Aoyanagi, Nobuyoshi, Mitsuya, Hiroaki, Sugiura, Wataru, Ohmagari, Norio
Published in Clinical infectious diseases (24.08.2022)
Published in Clinical infectious diseases (24.08.2022)
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Tecovirimat is active against various MPXV strains, while cidofovir, brincidofovir, trifluridine, and gemcitabine have no detectable MPXV-specific antiviral activity
Higashi-Kuwata, Nobuyo, Kato, Mariko, Hattori, Shin-ichiro, Takamatsu, Yuki, Mitsuya, Hiroaki
Published in Virus research (01.10.2025)
Published in Virus research (01.10.2025)
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Neutralization of SARS-CoV-2 with IgG from COVID-19-convalescent plasma
Maeda, Kenji, Higashi-Kuwata, Nobuyo, Kinoshita, Noriko, Kutsuna, Satoshi, Tsuchiya, Kiyoto, Hattori, Shin-ichiro, Matsuda, Kouki, Takamatsu, Yuki, Gatanaga, Hiroyuki, Oka, Shinichi, Sugiyama, Haruhito, Ohmagari, Norio, Mitsuya, Hiroaki
Published in Scientific reports (10.03.2021)
Published in Scientific reports (10.03.2021)
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Comparison of Rapid Antigen Tests for COVID-19
Yamayoshi, Seiya, Sakai-Tagawa, Yuko, Koga, Michiko, Akasaka, Osamu, Nakachi, Ichiro, Koh, Hidefumi, Maeda, Kenji, Adachi, Eisuke, Saito, Makoto, Nagai, Hiroyuki, Ikeuchi, Kazuhiko, Ogura, Takayuki, Baba, Rie, Fujita, Kensuke, Fukui, Takahiro, Ito, Fumimaro, Hattori, Shin-ichiro, Yamamoto, Kei, Nakamoto, Takato, Furusawa, Yuri, Yasuhara, Atsuhiro, Ujie, Michiko, Yamada, Shinya, Ito, Mutsumi, Mitsuya, Hiroaki, Omagari, Norio, Yotsuyanagi, Hiroshi, Iwatsuki-Horimoto, Kiyoko, Imai, Masaki, Kawaoka, Yoshihiro
Published in Viruses (10.12.2020)
Published in Viruses (10.12.2020)
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Structure–Activity Relationship Studies of SARS-CoV‑2 Main Protease Inhibitors Containing 4‑Fluorobenzothiazole-2-carbonyl Moieties
Tsuji, Kohei, Ishii, Takahiro, Kobayakawa, Takuya, Higashi-Kuwata, Nobuyo, Shinohara, Kouki, Azuma, Chika, Miura, Yutaro, Nakano, Hiroki, Wada, Naoya, Hattori, Shin-ichiro, Bulut, Haydar, Mitsuya, Hiroaki, Tamamura, Hirokazu
Published in Journal of medicinal chemistry (12.10.2023)
Published in Journal of medicinal chemistry (12.10.2023)
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Regio- and Stereoselective Synthesis of 2′-Deoxy-4′-thioguanine Nucleosides: Evaluation of Anti-Hepatitis B Virus Activity and Cytotoxicity Leading to Improved Selectivity Index by 4′- C -Cyanation
Kumamoto, Hiroki, Imoto, Shuhei, Kuwata-Higashi, Nobuyo, Mitsuya, Hiroaki, Haraguchi, Kazuhiro
Published in Synlett (05.12.2023)
Published in Synlett (05.12.2023)
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Neutralization against Omicron sublineages (BA.2/BA.5/BQ.1.1/XBB/XBB.1.5) in bivalent BNT162b2-vaccinated HCWs with or without risk factors, or following BT infection with Omicron
Amano, Masayuki, Otsu, Sachiko, Uemura, Yukari, Ichikawa, Yasuko, Matsumoto, Shota, Higashi-Kuwata, Nobuyo, Matsushita, Shuzo, Shimada, Shinya, Mitsuya, Hiroaki
Published in Scientific reports (13.10.2023)
Published in Scientific reports (13.10.2023)
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