Naphthyridines as Novel BET Family Bromodomain Inhibitors
Mirguet, Olivier, Lamotte, Yann, Chung, Chun-wa, Bamborough, Paul, Delannée, Delphine, Bouillot, Anne, Gellibert, Françoise, Krysa, Gael, Lewis, Antonia, Witherington, Jason, Huet, Pascal, Dudit, Yann, Trottet, Lionel, Nicodeme, Edwige
Published in ChemMedChem (01.03.2014)
Published in ChemMedChem (01.03.2014)
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The discovery of potent and selective kynurenine 3-monooxygenase inhibitors for the treatment of acute pancreatitis
Liddle, John, Beaufils, Benjamin, Binnie, Margaret, Bouillot, Anne, Denis, Alexis A., Hann, Michael M., Haslam, Carl P., Holmes, Duncan S., Hutchinson, Jon P., Kranz, Michael, McBride, Andrew, Mirguet, Olivier, Mole, Damian J., Mowat, Christopher G., Pal, Sandeep, Rowland, Paul, Trottet, Lionel, Uings, Iain J., Walker, Ann L., Webster, Scott P.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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3-(6-클로로-3-옥소-3,4-디히드로-(2H)-1,4-벤조옥사진-4-일) 프로판산 유도체 및 그의 KMO 억제제로서의 용도
DENIS ALEXIS, BOUILLOT ANNE MARIE JEANNE, LIDDLE JOHN, WALKER ANN LOUISE, MIRGUET OLIVIER
Year of Publication 15.01.2018
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Year of Publication 15.01.2018
Patent
Comparison of soluble guanylate cyclase stimulators and activators in models of cardiovascular disease associated with oxidative stress
Costell, Melissa H, Ancellin, Nicolas, Bernard, Roberta E, Zhao, Shufang, Upson, John J, Morgan, Lisa A, Maniscalco, Kristeen, Olzinski, Alan R, Ballard, Victoria L T, Herry, Kenny, Grondin, Pascal, Dodic, Nerina, Mirguet, Olivier, Bouillot, Anne, Gellibert, Francoise, Coatney, Robert W, Lepore, John J, Jucker, Beat M, Jolivette, Larry J, Willette, Robert N, Schnackenberg, Christine G, Behm, David J
Published in Frontiers in pharmacology (01.01.2012)
Published in Frontiers in pharmacology (01.01.2012)
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Journal Article
Rearrangement of β-amino alcohols and application to the synthesis of biologically active compounds
Cossy, Janine, Pardo, Domingo Gomez, Dumas, Cécile, Mirguet, Olivier, Déchamps, Ingrid, Métro, Thomas-Xavier, Burger, Benjamin, Roudeau, Rémi, Appenzeller, Jérôme, Cochi, Anne
Published in Chirality (New York, N.Y.) (01.10.2009)
Published in Chirality (New York, N.Y.) (01.10.2009)
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3-(5-CHLORO-2-OXOBENZO[D]OXAZOL-3(2H)-YL)PROPANOIC ACID DERIVATIVES AS KMO INHIBITORS
BOUILLOT ANNE MARIE JEANNE, LIDDLE JOHN, WALKER ANN LOUISE, MIRGUET OLIVIER
Year of Publication 18.08.2016
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Year of Publication 18.08.2016
Patent
Cover Picture: A Diverted Total Synthesis of Mycolactone Analogues: An Insight into Buruli Ulcer Toxins (Chem. Eur. J. 51/2011)
Chany, Anne-Caroline, Casarotto, Virginie, Schmitt, Marjorie, Tarnus, Céline, Guenin-Macé, Laure, Demangel, Caroline, Mirguet, Olivier, Eustache, Jacques, Blanchard, Nicolas
Published in Chemistry : a European journal (16.12.2011)
Published in Chemistry : a European journal (16.12.2011)
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Journal Article
Discovery of Pyridones As Oral AMPK Direct Activators
Mirguet, Olivier, Sautet, Stéphane, Clément, Catherine-Anne, Toum, Jérôme, Donche, Frédéric, Marques, Celine, Rondet, Emilie, Pizzonero, Mathieu, Beaufils, Benjamin, Dudit, Yann, Huet, Pascal, Trottet, Lionel, Grondin, Pascal, Brusq, Jean-Marie, Boursier, Eric, Saintillan, Yannick, Nicodeme, Edwige
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Journal Article
Inhibition of BET Recruitment to Chromatin As An Effective Treatment for MLL-Fusion Leukaemia
Dawson, Mark A, Prinjha, Rab, Dittman, Antje, Giotopoulos, George, Bantscheff, Marcus, Chan, Wai-In, Robson, Samuel, Chung, Chun-wa, Hopf, Carsten, Savitski, Mikhail, Döhner, Konstanze, Burnett, Alan K, Delwel, Ruud, Carola, Huthmacher, Gudgin, Emma, Lugo, Dave, Beinke, Soren, Soden, Peter, Auger, Kurt R., Mirguet, Olivier, Jeffrey, Phillip, Drewes, Gerard, Lee, Kevin, Kouzarides, Tony, Huntly, Brian J.P.
Published in Blood (18.11.2011)
Published in Blood (18.11.2011)
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Journal Article
Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia
Dawson, Mark A, Prinjha, Rab K, Dittmann, Antje, Giotopoulos, George, Bantscheff, Marcus, Chan, Wai-In, Robson, Samuel C, Chung, Chun-wa, Hopf, Carsten, Savitski, Mikhail M, Huthmacher, Carola, Gudgin, Emma, Lugo, Dave, Beinke, Soren, Chapman, Trevor D, Roberts, Emma J, Soden, Peter E, Auger, Kurt R, Mirguet, Olivier, Doehner, Konstanze, Delwel, Ruud, Burnett, Alan K, Jeffrey, Phillip, Drewes, Gerard, Lee, Kevin, Huntly, Brian J.P, Kouzarides, Tony
Published in Nature (London) (27.10.2011)
Published in Nature (London) (27.10.2011)
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Journal Article
BENZODIAZEPINE BROMODOMAIN INHIBITOR
BAILEY JAMES, WITHERINGTON JASON, GOSMINI ROMAIN LUC MARIE, MIRGUET OLIVIER
Year of Publication 04.09.2012
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Year of Publication 04.09.2012
Patent
Ring expansion: formal total synthesis of (−)-paroxetine
Cossy, Janine, Mirguet, Olivier, Gomez Pardo, Domingo, Desmurs, Jean-Roger
Published in Tetrahedron letters (13.08.2001)
Published in Tetrahedron letters (13.08.2001)
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Journal Article
PHENOL RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF
MAUGER, Jacques, TOUM, Jérôme, MIRGUET, Olivier, PINKERTON, Anthony B, REMEUR, Camille, TRUONG, Yen Pham Hong
Year of Publication 29.08.2024
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Year of Publication 29.08.2024
Patent