Transient receptor potential cation channel, subfamily V, member 4 and airway sensory afferent activation: Role of adenosine triphosphate
Bonvini, Sara J., PhD, Birrell, Mark A., PhD, Grace, Megan S., PhD, Maher, Sarah A., PhD, Adcock, John J., PhD, Wortley, Michael A., PhD, Dubuis, Eric, PhD, Ching, Yee-Man, MRes, Ford, Anthony P., PhD, Shala, Fisnik, MD, Miralpeix, Montserrat, PhD, Tarrason, Gema, PhD, Smith, Jaclyn A., PhD, Belvisi, Maria G., PhD
Published in Journal of allergy and clinical immunology (01.07.2016)
Published in Journal of allergy and clinical immunology (01.07.2016)
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Journal Article
The pan-JAK inhibitor LAS194046 reduces neutrophil activation from severe asthma and COPD patients in vitro
Milara, Javier, Ballester, Beatriz, de Diego, Alfredo, Calbet, Marta, Ramis, Isabel, Miralpeix, Montserrat, Cortijo, Julio
Published in Scientific reports (24.03.2022)
Published in Scientific reports (24.03.2022)
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Journal Article
In vitro anti-inflammatory effects of AZD8999, a novel bifunctional muscarinic acetylcholine receptor antagonist /β2-adrenoceptor agonist (MABA) compound in neutrophils from COPD patients
Milara, Javier, Contreras, Sonia, de Diego, Alfredo, Calbet, Marta, Aparici, Mònica, Morcillo, Esteban, Miralpeix, Montserrat, Cortijo, Julio
Published in PloS one (01.01.2019)
Published in PloS one (01.01.2019)
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Journal Article
Characterization of Aclidinium Bromide, a Novel Inhaled Muscarinic Antagonist, with Long Duration of Action and a Favorable Pharmacological Profile
Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Otal, Raquel, Carreño, Cristina, Viñals, Marisa, Doménech, Teresa, Carcasona, Carla, Reyes, Blanca, Vilella, Dolors, Gras, Jordi, Cortijo, Julio, Morcillo, Esteban, Llenas, Jesús, Ryder, Hamish, Beleta, Jorge
Published in The Journal of pharmacology and experimental therapeutics (01.11.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2009)
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Journal Article
Non-neuronal cholinergic system contributes to corticosteroid resistance in chronic obstructive pulmonary disease patients
Milara, Javier, Cervera, Angela, de Diego, Alfredo, Sanz, Celia, Juan, Gustavo, Gavaldà, Amadeu, Miralpeix, Montserrat, Morcillo, Esteban, Cortijo, Julio
Published in Respiratory research (08.11.2016)
Published in Respiratory research (08.11.2016)
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Journal Article
Application of a phenotypic drug discovery strategy to identify biological and chemical starting points for inhibition of TSLP production in lung epithelial cells
Orellana, Adelina, García-González, Vicente, López, Rosa, Pascual-Guiral, Sonia, Lozoya, Estrella, Díaz, Julia, Casals, Daniel, Barrena, Antolín, Paris, Stephane, Andrés, Miriam, Segarra, Victor, Vilella, Dolors, Malhotra, Rajneesh, Eastwood, Paul, Planagumà, Anna, Miralpeix, Montserrat, Nueda, Arsenio
Published in PloS one (01.01.2018)
Published in PloS one (01.01.2018)
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Journal Article
Effects of aclidinium bromide in a cigarette smoke-exposed Guinea pig model of chronic obstructive pulmonary disease
Domínguez-Fandos, David, Ferrer, Elisabet, Puig-Pey, Raquel, Carreño, Cristina, Prats, Neus, Aparici, Mònica, Musri, Melina Mara, Gavaldà, Amadeu, Peinado, Víctor I, Miralpeix, Montserrat, Barberà, Joan A
Published in American journal of respiratory cell and molecular biology (01.02.2014)
Published in American journal of respiratory cell and molecular biology (01.02.2014)
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Journal Article
PI3K, p38 and JAK/STAT signalling in bronchial tissue from patients with asthma following allergen challenge
Southworth, Thomas, Mason, Sarah, Bell, Alan, Ramis, Isabel, Calbet, Marta, Domenech, Anna, Prats, Neus, Miralpeix, Montserrat, Singh, Dave
Published in Biomarker research (11.04.2018)
Published in Biomarker research (11.04.2018)
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Journal Article
Synthesis and Biological Activity of Pyrido[3′,2′:4,5]thieno[3,2-d]pyrimidines as Phosphodiesterase Type 4 Inhibitors
Taltavull, Joan, Serrat, Jordi, Gràcia, Jordi, Gavaldà, Amadeu, Andrés, Míriam, Córdoba, Mònica, Miralpeix, Montserrat, Vilella, Dolors, Beleta, Jorge, Ryder, Hamish, Pagès, Lluís
Published in Journal of medicinal chemistry (14.10.2010)
Published in Journal of medicinal chemistry (14.10.2010)
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Journal Article
Discovery of novel quaternary ammonium derivatives of (3 R)-quinuclidinyl carbamates as potent and long acting muscarinic antagonists
Prat, Maria, Buil, María Antonia, Fernández, Maria Dolors, Castro, Jordi, Monleón, Juan Manuel, Tort, Laia, Casals, Gaspar, Ferrer, Manuel, Huerta, Josep Maria, Espinosa, Sònia, López, Manuel, Segarra, Victor, Gavaldà, Amadeu, Miralpeix, Montserrat, Ramos, Israel, Vilella, Dolors, González, Marisa, Córdoba, Mònica, Cárdenas, Alvaro, Antón, Francisca, Beleta, Jorge, Ryder, Hamish
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Journal Article
Synthesis and Biological Evaluation of 3,4-Diaryloxazolones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors
Puig, Carles, Crespo, María I, Godessart, Núria, Feixas, Joan, Ibarzo, Javier, Jiménez, Juan-Miguel, Soca, Lídia, Cardelús, Ignasi, Heredia, Ascensión, Miralpeix, Montserrat, Puig, Jaume, Beleta, Jordi, Huerta, Josep M, López, Manel, Segarra, Victor, Ryder, Hamish, Palacios, José M
Published in Journal of medicinal chemistry (27.01.2000)
Published in Journal of medicinal chemistry (27.01.2000)
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Journal Article
Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist
Eastwood, Paul, Esteve, Cristina, González, Jacob, Fonquerna, Silvia, Aiguadé, Josep, Carranco, Inés, Doménech, Teresa, Aparici, Mònica, Miralpeix, Montserrat, Albertí, Joan, Córdoba, Mónica, Fernández, Raquel, Pont, Mercè, Godessart, Núria, Prats, Neus, Loza, María Isabel, Cadavid, María Isabel, Nueda, Arsenio, Vidal, Bernat
Published in ACS medicinal chemistry letters (10.03.2011)
Published in ACS medicinal chemistry letters (10.03.2011)
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Journal Article
Novel Inhaled Pan-JAK Inhibitor, LAS194046, Reduces Allergen-Induced Airway Inflammation, Late Asthmatic Response, and pSTAT Activation in Brown Norway Rats
Calbet, Marta, Ramis, Isabel, Calama, Elena, Carreño, Cristina, Paris, Stephane, Maldonado, Monica, Orellana, Adelina, Calaf, Elena, Pauta, Montse, De Alba, Jorge, Bach, Jordi, Miralpeix, Montserrat
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
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Journal Article
Design, synthesis and biological activity of a targeted library of potential tryptase inhibitors
Garcia, M, del Rio, Silvestre, S, Rubiralta, M, Lozoya, E, Segarra, Fernandez, D, Miralpeix, M, Aparici, M, Diez, A
Published in Organic & biomolecular chemistry (07.06.2004)
Published in Organic & biomolecular chemistry (07.06.2004)
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Journal Article
Anti-inflammatory potential of PI3Kδ and JAK inhibitors in asthma patients
Southworth, Thomas, Plumb, Jonathan, Gupta, Vandana, Pearson, James, Ramis, Isabel, Lehner, Martin D, Miralpeix, Montserrat, Singh, Dave
Published in Respiratory research (04.10.2016)
Published in Respiratory research (04.10.2016)
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Journal Article
Selective induction of cyclo‐oxygenase‐2 activity in the permanent human endothelial cell line HUV‐EC‐C: biochemical and pharmacological characterization
Miralpeix, Montserrat, Camacho, Mercedes, López‐Belmonte, Jesús, Canalías, Francesca, Beleta, Jordi, Ma Palacios, José, Vila, Luis
Published in British journal of pharmacology (01.05.1997)
Published in British journal of pharmacology (01.05.1997)
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Journal Article
Abediterol (LAS100977), an inhaled long-acting β2-adrenoceptor agonist, has a fast association rate and long residence time at receptor
Ramos, Israel, Aparici, Mònica, Letosa, Maria, Puig, Carlos, Gavaldà, Amadeu, Huerta, Josep Maria, Espinosa, Sonia, Vilella, Dolors, Miralpeix, Montserrat
Published in European journal of pharmacology (15.01.2018)
Published in European journal of pharmacology (15.01.2018)
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Journal Article
In vitro anti-inflammatory effects of AZD8999, a novel bifunctional muscarinic acetylcholine receptor antagonist /[beta]2-adrenoceptor agonist compound in neutrophils from COPD patients
Milara, Javier, Contreras, Sonia, de Diego, Alfredo, Calbet, Marta, Aparici, Mònica, Morcillo, Esteban, Miralpeix, Montserrat, Co
Published in PloS one (04.01.2019)
Published in PloS one (04.01.2019)
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Journal Article
In vitro anti-inflammatory effects of AZD8999, a novel bifunctional muscarinic acetylcholine receptor antagonist /[beta]2-adrenoceptor agonist
Milara, Javier, Contreras, Sonia, de Diego, Alfredo, Calbet, Marta, Aparici, Mònica, Morcillo, Esteban, Miralpeix, Montserrat, Cortijo, Julio
Published in PloS one (04.01.2019)
Published in PloS one (04.01.2019)
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