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Chantigny, Yves A, Murray, John C, Kleinman, Edward F, Robinson, Ralph P, Plotkin, Michael A, Reese, Matthew R, Buckbinder, Leonard, McNiff, Patricia A, Millham, Michele L, Schaefer, Jean F, Abramov, Yuriy A, Bordner, Jon
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Published in Journal of medicinal chemistry (26.03.2015)
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Discovery of triazolopyrimidine-based PDE8B inhibitors: Exceptionally ligand-efficient and lipophilic ligand-efficient compounds for the treatment of diabetes
DeNinno, Michael P., Wright, Stephen W., Etienne, John B., Olson, Thanh V., Rocke, Benjamin N., Corbett, Jeffrey W., Kung, Daniel W., DiRico, Kenneth J., Andrews, Kim M., Millham, Michele L., Parker, Janice C., Esler, William, van Volkenburg, Maria, Boyer, David D., Houseknecht, Karen L., Doran, Shawn D.
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Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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1,5-Substituted nipecotic amides: Selective PDE8 inhibitors displaying diastereomer-dependent microsomal stability
DeNinno, Michael P., Wright, Stephen W., Visser, Michael S., Etienne, John B., Moore, Dianna E., Olson, Thanh V., Rocke, Benjamin N., Andrews, Melissa P., Zarbo, Cynthia, Millham, Michele L., Boscoe, Brian P., Boyer, David D., Doran, Shawn D., Houseknecht, Karen L.
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Robinson, Ralph P, Buckbinder, Leonard, Haugeto, Amber I, McNiff, Patricia A, Millham, Michele L, Reese, Matthew R, Schaefer, Jean F, Abramov, Yuriy A, Bordner, Jon, Chantigny, Yves A, Kleinman, Edward F, Laird, Ellen R, Morgan, Bradley P, Murray, John C, Salter, Eben D, Wessel, Matthew D, Yocum, Sue A
Published in Journal of medicinal chemistry (26.03.2009)
Published in Journal of medicinal chemistry (26.03.2009)
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