Protein–Protein Interaction Inhibition (2P2I)-Oriented Chemical Library Accelerates Hit Discovery
Milhas, Sabine, Raux, Brigitt, Betzi, Stéphane, Derviaux, Carine, Roche, Philippe, Restouin, Audrey, Basse, Marie-Jeanne, Rebuffet, Etienne, Lugari, Adrien, Badol, Marion, Kashyap, Rudra, Lissitzky, Jean-Claude, Eydoux, Cécilia, Hamon, Véronique, Gourdel, Marie-Edith, Combes, Sébastien, Zimmermann, Pascale, Aurrand-Lions, Michel, Roux, Thomas, Rogers, Catherine, Müller, Susanne, Knapp, Stefan, Trinquet, Eric, Collette, Yves, Guillemot, Jean-Claude, Morelli, Xavier
Published in ACS chemical biology (19.08.2016)
Published in ACS chemical biology (19.08.2016)
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Journal Article
Competitive SPR using an intracellular anti-LMO2 antibody identifies novel LMO2-interacting compounds
Canning, Peter, Bataille, Carole, Bery, Nicolas, Milhas, Sabine, Hayes, Angela, Raynaud, Florence, Miller, Ami, Rabbitts, Terry
Published in Journal of immunological methods (01.07.2021)
Published in Journal of immunological methods (01.07.2021)
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Journal Article
Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins
Raux, Brigitt, Voitovich, Yuliia, Derviaux, Carine, Lugari, Adrien, Rebuffet, Etienne, Milhas, Sabine, Priet, Stéphane, Roux, Thomas, Trinquet, Eric, Guillemot, Jean-Claude, Knapp, Stefan, Brunel, Jean-Michel, Fedorov, Alexey Yu, Collette, Yves, Roche, Philippe, Betzi, Stéphane, Combes, Sébastien, Morelli, Xavier
Published in Journal of medicinal chemistry (25.02.2016)
Published in Journal of medicinal chemistry (25.02.2016)
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Journal Article
An antibody-drug conjugate with intracellular drug release properties showing specific cytotoxicity against CD7-positive cells
Zhang, Jing, Jain, Arvind, Milhas, Sabine, Williamson, Daniel J., Mysliwy, Justyna, Lodge, Adam, Thirlway, Jenny, Al Nakeeb, Majid, Miller, Ami, Rabbitts, Terry H.
Published in Leukemia research (01.09.2021)
Published in Leukemia research (01.09.2021)
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Journal Article
A cell-based screening method using an intracellular antibody for discovering small molecules targeting the translocation protein LMO2
Bery, Nicolas, Bataille, Carole J R, Russell, Angela, Hayes, Angela, Raynaud, Florence, Milhas, Sabine, Anand, Sneha, Tulmin, Hanna, Miller, Ami, Rabbitts, Terence H
Published in Science advances (09.04.2021)
Published in Science advances (09.04.2021)
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Journal Article
XANTHINE DERIVATIVE INHIBITORS OF BET PROTEINS
COLLETTE, Yves, COMBES, Sébastien, GUILLEMOT, Jean-Claude, ROCHE, Philippe, VOITOVICH, luliia, LUGARI, Adrein, MORELLI, Xavier, MILHAS, Sabine, RAUX, Brigit, BETZI, Stéphanie
Year of Publication 26.09.2019
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Year of Publication 26.09.2019
Patent
XANTHINE DERIVATIVE INHIBITORS OF BET PROTEINS
VOITOVICH, Iuliia, RAUX, Brigitt, COLLETTE, Yves, COMBES, Sébastien, GUILLEMOT, Jean-Claude, ROCHE, Philippe, MORELLI, Xavier, BETZI, Stéphane, LUGARI, Adrien, MILHAS, Sabine
Year of Publication 07.11.2018
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Year of Publication 07.11.2018
Patent
XANTHINE DERIVATIVE INHIBITORS OF BET PROTEINS
VOITOVICH, Iuliia, RAUX, Brigitt, COLLETTE, Yves, COMBES, Sébastien, GUILLEMOT, Jean-Claude, ROCHE, Philippe, MORELLI, Xavier, BETZI, Stéphane, LUGARI, Adrien, MILHAS, Sabine
Year of Publication 06.07.2017
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Year of Publication 06.07.2017
Patent