Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: Design, synthesis, and microbiological evaluation
Schiaffella, Fausto, Macchiarulo, Antonio, Milanese, Lara, Vecchiarelli, Anna, Fringuelli, Renata
Published in Bioorganic & medicinal chemistry (01.08.2006)
Published in Bioorganic & medicinal chemistry (01.08.2006)
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Journal Article
Design, Synthesis, and Microbiological Evaluation of New Candida albicans CYP51 Inhibitors
Schiaffella, Fausto, Macchiarulo, Antonio, Milanese, Lara, Vecchiarelli, Anna, Costantino, Gabriele, Pietrella, Donatella, Fringuelli, Renata
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
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Journal Article
Oxime and Oxime Ether Derivatives of 1,4-Benzothiazine Related to Oxiconazole
Milanese, Lara, Giacchè, Nicola, Schiaffella, Fausto, Vecchiarelli, Anna, Macchiarulo, Antonio, Fringuelli, Renata
Published in ChemMedChem (13.08.2007)
Published in ChemMedChem (13.08.2007)
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Journal Article
1,4-Benzothiazine analogues and apoptosis: structure–activity relationship
Fringuelli, Renata, Schiaffella, Fausto, Utrilla Navarro, M.Pilar, Milanese, Lara, Santini, Cristina, Rapucci, Michela, Marchetti, Cristina, Riccardi, Carlo
Published in Bioorganic & medicinal chemistry (31.07.2003)
Published in Bioorganic & medicinal chemistry (31.07.2003)
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Journal Article
1,4-Benzothiazine analogues and apoptosis
Fringuelli, Renata, Schiaffella, Fausto, Utrilla Navarro, M.Pilar, Milanese, Lara, Santini, Cristina, Rapucci, Michela, Marchetti, Cristina, Riccardi, Carlo
Published in Bioorganic & medicinal chemistry (01.07.2003)
Published in Bioorganic & medicinal chemistry (01.07.2003)
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Journal Article
Synthesis and evaluation of anti-apoptotic activity of L-carnitine cyclic analogues and amino acid derivatives
Fringuelli, Renata, Utrilla Navarro, M.Pilar, Milanese, Lara, Bruscoli, Stefano, Schiaffella, Fausto, Riccardi, Carlo, De Simone, Claudio
Published in Farmaco (Società chimica italiana : 1989) (01.04.2004)
Published in Farmaco (Società chimica italiana : 1989) (01.04.2004)
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Synthesis and Evaluation of anti-Apoptotic Activity of L-Carnitine Cyclic Analogues and Amino Acid Derivatives
Fringuelli, Renata, Utrilla Navarro, M. Pilar, Milanese, Lara, Bruscoli, Stefano, Schiaffella, Fausto, Riccardi, Carlo, De Simone, Claudio
Published in ChemInform (24.08.2004)
Published in ChemInform (24.08.2004)
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