Diastereotopic and Deuterium Effects in Gemini
Maehr, Hubert, Rochel, Natacha, Lee, Hong Jin, Suh, Nanjoo, Uskokovic, Milan R
Published in Journal of medicinal chemistry (23.05.2013)
Published in Journal of medicinal chemistry (23.05.2013)
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Altered Nuclear Receptor Corepressor Expression Attenuates Vitamin D Receptor Signaling in Breast Cancer Cells
BANWELL, Claire M, MACCARTNEY, Donia P, CAMPBELL, Moray J, GUY, Michelle, MILES, Alice E, USKOKOVIC, Milan R, MANSI, Janine, STEWART, Paul M, O'NEILL, Laura P, TURNER, Bryan M, COLSTON, Kay W
Published in Clinical cancer research (01.04.2006)
Published in Clinical cancer research (01.04.2006)
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Structural Evaluation of the Agonistic Action of a Vitamin D Analog with Two Side Chains Binding to the Nuclear Vitamin D Receptor
Väisänen, Sami, Peräkylä, Mikael, Kärkkäinen, Jouni I, Uskokovic, Milan R, Carlberg, Carsten
Published in Molecular pharmacology (01.06.2003)
Published in Molecular pharmacology (01.06.2003)
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Metabolism of selective 20-epi-vitamin D-3 analogs in rat osteosarcoma UMR-106 cells: Isolation and identification of four novel C-1 fatty acid esters of 1 alpha,25-dihydroxy-16-ene-20-epi-vitamin D-3
Flarakos, Caroline Ceailles, Weiskopf, Andrew, Robinson, Matthew, Wang, Guoshun, Vouros, Paul, Sasso, Gino J., Uskokovic, Milan R., Reddy, G. Satyanarayana
Published in Steroids (01.03.2017)
Published in Steroids (01.03.2017)
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Calcitriol Derivatives with Two Different Side Chains at C-20. V. Potent Inhibitors of Mammary Carcinogenesis and Inducers of Leukemia Differentiation
Maehr, Hubert, Lee, Hong Jin, Perry, Bradford, Suh, Nanjoo, Uskokovic, Milan R
Published in Journal of medicinal chemistry (10.09.2009)
Published in Journal of medicinal chemistry (10.09.2009)
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Journal Article
Novel Gemini vitamin D3 analogs: Large structure/function analysis and ability to induce antimicrobial peptide
Okamoto, Ryoko, Gery, Sigal, Kuwayama, Yoshio, Borregaard, Niels, Ho, Quoc, Alvarez, Rocio, Akagi, Tadayuki, Liu, George Y., Uskokovic, Milan R., Koeffler, H. Phillip
Published in International journal of cancer (01.01.2014)
Published in International journal of cancer (01.01.2014)
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Journal Article
Metabolism of selective 20-epi-vitamin D3 analogs in rat osteosarcoma UMR-106 cells: Isolation and identification of four novel C-1 fatty acid esters of 1α,25-dihydroxy-16-ene-20-epi-vitamin D3
Flarakos, Caroline Ceailles, Weiskopf, Andrew, Robinson, Matthew, Wang, Guoshun, Vouros, Paul, Sasso, Gino J., Uskokovic, Milan R., Reddy, G. Satyanarayana
Published in Steroids (01.03.2017)
Published in Steroids (01.03.2017)
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Journal Article
Synergistic Antileukemic Activity of Carnosic Acid-Rich Rosemary Extract and the 19-nor Gemini Vitamin D Analogue in a Mouse Model of Systemic Acute Myeloid Leukemia
Shabtay, Ayelet, Sharabani, Hagar, Barvish, Zeev, Kafka, Michael, Amichay, Doron, Levy, Joseph, Sharoni, Yoav, Uskokovic, Milan R., Studzinski, George P., Danilenko, Michael
Published in Oncology (01.10.2008)
Published in Oncology (01.10.2008)
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Journal Article
Potent Antiproliferative Effects of 25-Hydroxy-16-ene-23-yne-vitamin D3 That Resists the Catalytic Activity of Both CYP27B1 and CYP24A1
Rhieu, Steve Y., Annalora, Andrew J., LaPorta, Erika, Welsh, JoEllen, Itoh, Toshimasa, Yamamoto, Keiko, Sakaki, Toshiyuki, Chen, Tai C., Uskokovic, Milan R., Reddy, G. Satyanarayana
Published in Journal of cellular biochemistry (01.08.2014)
Published in Journal of cellular biochemistry (01.08.2014)
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Journal Article
Synergistic growth inhibition of prostate cancer cells by 1α, 25 dihydroxyvitamin D3 and its 19-nor-hexafluoride analogs in combination with either sodium butyrate or trichostatin A
RASHID, Samantha F, MOORE, Jasbir S, WALKER, Elizabeth, DRIVER, Philip M, ENGEL, Jaqueline, EDWARDS, Ceri E, BROWN, Geoffrey, USKOKOVIC, Milan R, CAMPBELL, Moray J
Published in Oncogene (05.04.2001)
Published in Oncogene (05.04.2001)
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Journal Article
Novel vitamin D3 analog, 21-(3-methyl-3-hydroxy-butyl)-19-nor D3, that modulates cell growth, differentiation, apoptosis, cell cycle, and induction of PTEN in leukemic cells
Hisatake, Jun-ichi, O'Kelly, James, Uskokovic, Milan R., Tomoyasu, Shigeru, Koeffler, H. Phillip
Published in Blood (15.04.2001)
Published in Blood (15.04.2001)
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Journal Article
Calcitriol derivatives with two different side-chains at C-20. Part 4: Further chain modifications that alter VDR-dependent monocytic differentiation potency in human leukemia cells
Garay, Edward, Jankowski, Pawel, Lizano, Paulo, Marczak, Stanislaw, Maehr, Hubert, Adorini, Luciano, Uskokovic, Milan R., Studzinski, George P.
Published in Bioorganic & medicinal chemistry (01.07.2007)
Published in Bioorganic & medicinal chemistry (01.07.2007)
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Journal Article
Targeting 1α, 25-dihydroxyvitamin D3 antiproliferative insensitivity in breast cancer cells by co-treatment with histone deacetylation inhibitors
BANWELL, Claire M, O'NEILL, Laura P, USKOKOVIC, Milan R, CAMPBELL, Moray J
Published in Journal of steroid biochemistry and molecular biology (01.05.2004)
Published in Journal of steroid biochemistry and molecular biology (01.05.2004)
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Conference Proceeding
Journal Article
The Biological Activities of 1α,25-Dihydroxyvitamin D3 and Its Synthetic Analog 1α,25-Dihydroxy-16-ene-vitamin D3 in Normal Human Osteoblastic Cells and Human Osteosarcoma SaOS-2 Cells Are Modulated by 17-β Estradiol and Dependent on Stage of Differentiation
RAO, Leticia G., LIU, Lily J.-F., RAWLINS, Myrna R., MCBROOM, Robert J., MURRAY, Timothy M., REDDY, G. Satyanarayama, USKOKOVIC, Milan R., RAO, D. Sunita, SUTHERLAND, May Kung
Published in Biological and Pharmaceutical Bulletin (2001)
Published in Biological and Pharmaceutical Bulletin (2001)
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Journal Article
Response Element and Coactivator-Mediated Conformational Change of the Vitamin D3 Receptor Permits Sensitive Interaction with Agonists
Michaela Herdick, Yvonne Bury, Marcus Quack, Milan R. Uskokovic, Patsie Polly, Carsten Carlberg
Published in Molecular pharmacology (01.06.2000)
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Published in Molecular pharmacology (01.06.2000)
Journal Article
Characterization of a Novel Analogue of 1α,25(OH)2-Vitamin D3 with Two Side Chains: Interaction with Its Nuclear Receptor and Cellular Actions
Norman, Anthony W, Manchand, Percy S, Uskokovic, Milan R, Okamura, William H, Takeuchi, Janet A, Bishop, June E, Hisatake, Jun-Iichi, Koeffler, H. Phillip, Peleg, Sara
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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Journal Article
23-carboxy-24,25,26,27-tetranorvitamin D3 (calcioic acid) and 24-carboxy-25,26,27-trinorvitamin D3 (cholacalcioic acid): end products of 25-hydroxyvitamin D3 metabolism in rat kidney through C-24 oxidation pathway
Reddy, G Satyanarayana, Omdahl, John L, Robinson, Matthew, Wang, Guochun, Palmore, G Tayhas R, Vicchio, Domenick, Yergey, Alfred L, Tserng, Kou-Yi, Uskokovic, Milan R
Published in Archives of biochemistry and biophysics (01.11.2006)
Published in Archives of biochemistry and biophysics (01.11.2006)
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Journal Article