Search Results - "Mikkelsen, Gitte" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Design and Synthesis of Pyrrolo[2,3‑d]pyrimidine-Derived Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitors Using a Checkpoint Kinase 1 (CHK1)-Derived Crystallographic Surrogate

Design and Synthesis of Pyrrolo[2,3‑d]pyrimidine-Derived Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitors Using a Checkpoint Kinase 1 (CHK1)-Derived Crystallographic Surrogate

by Williamson, Douglas S, Smith, Garrick P, Mikkelsen, Gitte K, Jensen, Thomas, Acheson-Dossang, Pamela, Badolo, Lassina, Bedford, Simon T, Chell, Victoria, Chen, I-Jen, Dokurno, Pawel, Hentzer, Morten, Newland, Samantha, Ray, Stuart C, Shaw, Terry, Surgenor, Allan E, Terry, Lindsey, Wang, Yikang, Christensen, Kenneth V
Published in Journal of medicinal chemistry (22.07.2021)

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Journal Article

Efficacy switching SAR of mGluR5 allosteric modulators: Highly potent positive and negative modulators from one chemotype

Efficacy switching SAR of mGluR5 allosteric modulators: Highly potent positive and negative modulators from one chemotype

by Sams, Anette Graven, Mikkelsen, Gitte Kobberøe, Brodbeck, Robbin M., Pu, Xiaosui, Ritzén, Andreas
Published in Bioorganic & medicinal chemistry letters (01.06.2011)

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Journal Article

The design and SAR of a novel series of 2-aminopyridine based LRRK2 inhibitors

The design and SAR of a novel series of 2-aminopyridine based LRRK2 inhibitors

by Smith, Garrick P., Badolo, Lassina, Chell, Victoria, Chen, I-Jen, Christensen, Kenneth Vielsted, David, Laurent, Daechsel, Justus Alfred, Hentzer, Morten, Herzig, Martin Christian, Mikkelsen, Gitte Kobberøe, Watson, Stephen P., Williamson, Douglas S.
Published in Bioorganic & medicinal chemistry letters (15.09.2017)

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Journal Article

Discovery of Phosphoric Acid Mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluorobenzoylimino]-thiazol-3-ylmethyl} Ester (Lu AA47070): A Phosphonooxymethylene Prodrug of a Potent and Selective hA(2A) Receptor Antagonist

Discovery of Phosphoric Acid Mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluorobenzoylimino]-thiazol-3-ylmethyl} Ester (Lu AA47070): A Phosphonooxymethylene Prodrug of a Potent and Selective hA(2A) Receptor Antagonist

by Sams, Anette G., Mikkelsen, Gitte K., Larsen, Mogens, Langgard, Morten, Howells, Mark E., Schroder, Tenna J., Brennum, Lise T., Torup, Lars, Jorgensen, Erling B., Bundgaard, Christoffer, Kreilgard, Mads, Bang-Andersen, Benny
Published in Journal of medicinal chemistry (10.02.2011)

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Journal Article

The meaning of personal diaries to children and families in the paediatric intensive care unit: A qualitative study

The meaning of personal diaries to children and families in the paediatric intensive care unit: A qualitative study

by Mikkelsen, Gitte
Published in Intensive & critical care nursing (01.04.2018)

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Journal Article

The synthesis and SAR of 2-arylsulfanylphenyl-1-oxyalkylamino acids as GlyT-1 inhibitors

The synthesis and SAR of 2-arylsulfanylphenyl-1-oxyalkylamino acids as GlyT-1 inhibitors

by Smith, Garrick, Mikkelsen, Gitte, Eskildsen, Jørgen, Bundgaard, Christoffer
Published in Bioorganic & medicinal chemistry letters (01.08.2006)

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Journal Article

Hit-to-lead investigation of a series of novel combined dopamine D2 and muscarinic M1 receptor ligands with putative antipsychotic and pro-cognitive potential

Hit-to-lead investigation of a series of novel combined dopamine D2 and muscarinic M1 receptor ligands with putative antipsychotic and pro-cognitive potential

by Sams, Anette Graven, Larsen, Krestian, Mikkelsen, Gitte Kobberøe, Hentzer, Morten, Christoffersen, Claus Tornby, Jensen, Klaus Gjervig, Frederiksen, Kristen, Bang-Andersen, Benny
Published in Bioorganic & medicinal chemistry letters (01.08.2012)

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Journal Article

Family-centred care of children in hospital - a concept analysis

Family-centred care of children in hospital - a concept analysis

by Mikkelsen, Gitte, Frederiksen, Kirsten
Published in Journal of Advanced Nursing (01.05.2011)

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Journal Article Book Review

The synthesis and SAR of 2-arylsulfanyl-phenyl piperazinyl acetic acids as glyT-1 inhibitors

The synthesis and SAR of 2-arylsulfanyl-phenyl piperazinyl acetic acids as glyT-1 inhibitors

by Smith, Garrick, Ruhland, Thomas, Mikkelsen, Gitte, Andersen, Kim, Christoffersen, Claus Tornby, Alifrangis, Lene Hjorth, Mørk, Arne, Wren, Stephen P, Harris, Neil, Wyman, Barry M, Brandt, Guillaume
Published in Bioorganic & medicinal chemistry letters (02.08.2004)

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Journal Article

Family-centred care of children in hospital - a concept analysis: Family-centred care of children in hospital

Family-centred care of children in hospital - a concept analysis: Family-centred care of children in hospital

by Mikkelsen, Gitte, Frederiksen, Kirsten
Published in Journal of advanced nursing (01.05.2011)

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Journal Article

Discovery of N-{1-[3-(3-Oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): An Allosteric Muscarinic M-1 Receptor Agonist with Unprecedented Selectivity and Procognitive Potential

Discovery of N-{1-[3-(3-Oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): An Allosteric Muscarinic M-1 Receptor Agonist with Unprecedented Selectivity and Procognitive Potential

by Sams, Anette G., Hentzer, Morten, Mikkelsen, Gitte K., Larsen, Krestian, Bundgaard, Christoffer, Plath, Niels, Christoffersen, Claus T., Bang-Andersen, Benny
Published in Journal of medicinal chemistry (09.09.2010)

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Journal Article

Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility

Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility

by Mikkelsen, Gitte Kobberøe, Langgård, Morten, Schrøder, Tenna Juul, Kreilgaard, Mads, Jørgensen, Erling B., Brandt, Guillaume, Griffon, Yann, Boffey, Ray, Bang-Andersen, Benny
Published in Bioorganic & medicinal chemistry letters (15.03.2015)

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Journal Article

Synthesis and SAR studies of analogues of 4-(3,3-dimethylbutyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A(2A) receptor ligands with improved aqueous solubility

Synthesis and SAR studies of analogues of 4-(3,3-dimethylbutyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A(2A) receptor ligands with improved aqueous solubility

by Mikkelsen, Gitte Kobberoe, Langgard, Morten, Schroder, Tenna Juul, Kreilgaard, Mads, Jorgensen, Erling B., Brandt, Guillaume, Griffon, Yann, Boffey, Ray, Bang-Andersen, Benny
Published in Bioorganic & medicinal chemistry letters (15.03.2015)

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Journal Article

Discovery of Phosphoric Acid Mono-{2-[( E / Z )-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} Ester (Lu AA47070): A Phosphonooxymethylene Prodrug of a Potent and Selective hA 2A Receptor Antagonist

Discovery of Phosphoric Acid Mono-{2-[( E / Z )-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} Ester (Lu AA47070): A Phosphonooxymethylene Prodrug of a Potent and Selective hA 2A Receptor Antagonist

by Sams, Anette G., Mikkelsen, Gitte K., Larsen, Mogens, Langgård, Morten, Howells, Mark E., Schrøder, Tenna J., Brennum, Lise T., Torup, Lars, Jørgensen, Erling B., Bundgaard, Christoffer, Kreilgård, Mads, Bang-Andersen, Benny
Published in Journal of medicinal chemistry (10.02.2011)

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Journal Article

Hit-to-lead investigation of a series of novel combined dopamine D-2 and muscarinic M-1 receptor ligands with putative antipsychotic and pro-cognitive potential

Hit-to-lead investigation of a series of novel combined dopamine D-2 and muscarinic M-1 receptor ligands with putative antipsychotic and pro-cognitive potential

by Sams, Anette Graven, Larsen, Krestian, Mikkelsen, Gitte Kobberoe, Hentzer, Morten, Christoffersen, Claus Tornby, Jensen, Klaus Gjervig, Frederiksen, Kristen, Bang-Andersen, Benny
Published in Bioorganic & medicinal chemistry letters (01.08.2012)

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Journal Article

Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A2A receptor antagonists

Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A2A receptor antagonists

by GRAVEN SAMS, Anette, MIKKELSEN, Gitte Kobberøe, LARSEN, Mogens, TORUP, Lars, BRENNUM, Lise Tottrup, SCHRØDER, Tenna Juul, BANG-ANDERSEN, Benny
Published in Bioorganic & medicinal chemistry letters (01.09.2010)

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Journal Article

Discovery of N-{1-[3-(3-Oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): An Allosteric Muscarinic M1 Receptor Agonist with Unprecedented Selectivity and Procognitive Potential

Discovery of N-{1-[3-(3-Oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): An Allosteric Muscarinic M1 Receptor Agonist with Unprecedented Selectivity and Procognitive Potential

by Sams, Anette G, Hentzer, Morten, Mikkelsen, Gitte K, Larsen, Krestian, Bundgaard, Christoffer, Plath, Niels, Christoffersen, Claus T, Bang-Andersen, Benny
Published in Journal of medicinal chemistry (09.09.2010)

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Journal Article

STAT3-mediated constitutive expression of SOCS-3 in cutaneous T-cell lymphoma

STAT3-mediated constitutive expression of SOCS-3 in cutaneous T-cell lymphoma

by BRENDER, Christine, NIELSEN, Mette, KALTOFT, Keld, MIKKELSEN, Gitte, ZHANG, Qian, WASIK, Mariusz, BILLESTRUP, Nils, ØDUM, Niels
Published in Blood (15.02.2001)

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Journal Article

Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A 2A receptor antagonists

Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A 2A receptor antagonists

by Sams, Anette Graven, Mikkelsen, Gitte Kobberøe, Larsen, Mogens, Torup, Lars, Brennum, Lise Tøttrup, Schrøder, Tenna Juul, Bang-Andersen, Benny
Published in Bioorganic & medicinal chemistry letters (2010)

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Journal Article

2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME

2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME

by GRENON MICHEL, SAMS ANETTE GRAVEN, HOPPER ALLEN, MIKKELSEN GITTE KOBBEROEE, PACKIARAJAN MATHIVANAN
Year of Publication 08.08.2012

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