Molecular Design and Synthesis of Ivermectin Hybrids Targeting Hepatic and Erythrocytic Stages of Plasmodium Parasites
Singh, Lovepreet, Fontinha, Diana, Francisco, Denise, Mendes, Antonio M, Prudêncio, Miguel, Singh, Kamaljit
Published in Journal of medicinal chemistry (27.02.2020)
Published in Journal of medicinal chemistry (27.02.2020)
Get full text
Journal Article
Five decades of clinical assessment of whole-sporozoite malaria vaccines
Nunes-Cabaço, Helena, Moita, Diana, Prudêncio, Miguel
Published in Frontiers in immunology (08.09.2022)
Published in Frontiers in immunology (08.09.2022)
Get full text
Journal Article
Repurposing Drugs to Fight Hepatic Malaria Parasites
Fontinha, Diana, Moules, Isabel, Prudêncio, Miguel
Published in Molecules (Basel, Switzerland) (28.07.2020)
Published in Molecules (Basel, Switzerland) (28.07.2020)
Get full text
Journal Article
The silent path to thousands of merozoites: the Plasmodium liver stage
Mota, Maria M, Prudêncio, Miguel, Rodriguez, Ana
Published in Nature reviews. Microbiology (01.11.2006)
Published in Nature reviews. Microbiology (01.11.2006)
Get full text
Journal Article
Liver-stage malaria parasites vulnerable to diverse chemical scaffolds
Derbyshire, Emily R, Prudêncio, Miguel, Mota, Maria M, Clardy, Jon
Published in Proceedings of the National Academy of Sciences - PNAS (29.05.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (29.05.2012)
Get full text
Journal Article
Targeting the Liver Stage of Malaria Parasites: A Yet Unmet Goal
Rodrigues, Tiago, Prudêncio, Miguel, Moreira, Rui, Mota, Maria M, Lopes, Francisca
Published in Journal of medicinal chemistry (09.02.2012)
Published in Journal of medicinal chemistry (09.02.2012)
Get full text
Journal Article
Novel Harmicines with Improved Potency against Plasmodium
Marinović, Marina, Perković, Ivana, Fontinha, Diana, Prudêncio, Miguel, Held, Jana, Pessanha de Carvalho, Lais, Tandarić, Tana, Vianello, Robert, Zorc, Branka, Rajić, Zrinka
Published in Molecules (Basel, Switzerland) (23.09.2020)
Published in Molecules (Basel, Switzerland) (23.09.2020)
Get full text
Journal Article
Antimalarial Pyrido[1,2‑a]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model
Singh, Kawaljit, Okombo, John, Brunschwig, Christel, Ndubi, Ferdinand, Barnard, Linley, Wilkinson, Chad, Njogu, Peter M, Njoroge, Mathew, Laing, Lizahn, Machado, Marta, Prudêncio, Miguel, Reader, Janette, Botha, Mariette, Nondaba, Sindisiwe, Birkholtz, Lyn-Marie, Lauterbach, Sonja, Churchyard, Alisje, Coetzer, Theresa L, Burrows, Jeremy N, Yeates, Clive, Denti, Paolo, Wiesner, Lubbe, Egan, Timothy J, Wittlin, Sergio, Chibale, Kelly
Published in Journal of medicinal chemistry (23.02.2017)
Published in Journal of medicinal chemistry (23.02.2017)
Get full text
Journal Article
The Impact of Antiretroviral Therapy on Malaria Parasite Transmission
Azevedo, Raquel, Mendes, António M, Prudêncio, Miguel
Published in Frontiers in microbiology (24.01.2020)
Published in Frontiers in microbiology (24.01.2020)
Get full text
Journal Article
Half-Sandwich Cyclopentadienylruthenium(II) Complexes: A New Antimalarial Chemotype
Milheiro, Sofia A, Gonçalves, Joana, Lopes, Ricardo M. R. M, Madureira, Margarida, Lobo, Lis, Lopes, Andreia, Nogueira, Fátima, Fontinha, Diana, Prudêncio, Miguel, M. Piedade, M. Fátima, Pinto, Sandra N, Florindo, Pedro R, Moreira, Rui
Published in Inorganic chemistry (08.09.2020)
Published in Inorganic chemistry (08.09.2020)
Get full text
Journal Article
Translation of liver stage activity of M5717, a Plasmodium elongation factor 2 inhibitor: from bench to bedside
Khandelwal, Akash, Arez, Francisca, Alves, Paula M, Badolo, Lassina, Brito, Catarina, Fischli, Christoph, Fontinha, Diana, Oeuvray, Claude, Prudêncio, Miguel, Rottmann, Matthias, Wilkins, Justin, Yalkinoglu, Özkan, Bagchus, Wilhelmina M, Spangenberg, Thomas
Published in Malaria journal (15.05.2022)
Published in Malaria journal (15.05.2022)
Get full text
Journal Article
Structure–Activity Relationship Studies and Plasmodium Life Cycle Profiling Identifies Pan-Active N‑Aryl-3-trifluoromethyl Pyrido[1,2‑a]benzimidazoles Which Are Efficacious in an in Vivo Mouse Model of Malaria
Mayoka, Godfrey, Njoroge, Mathew, Okombo, John, Gibhard, Liezl, Sanches-Vaz, Margarida, Fontinha, Diana, Birkholtz, Lyn-Marie, Reader, Janette, van der Watt, Mariëtte, Coetzer, Theresa L, Lauterbach, Sonja, Churchyard, Alisje, Bezuidenhout, Belinda, Egan, Timothy J, Yeates, Clive, Wittlin, Sergio, Prudêncio, Miguel, Chibale, Kelly
Published in Journal of medicinal chemistry (24.01.2019)
Published in Journal of medicinal chemistry (24.01.2019)
Get full text
Journal Article
Trypanosoma brucei infection protects mice against malaria
Sanches-Vaz, Margarida, Temporão, Adriana, Luis, Rafael, Nunes-Cabaço, Helena, Mendes, António M, Goellner, Sarah, Carvalho, Tânia, Figueiredo, Luisa M, Prudêncio, Miguel
Published in PLoS pathogens (08.11.2019)
Published in PLoS pathogens (08.11.2019)
Get full text
Journal Article
Tetraoxane–Pyrimidine Nitrile Hybrids as Dual Stage Antimalarials
Oliveira, Rudi, Guedes, Rita C, Meireles, Patrícia, Albuquerque, Inês S, Gonçalves, Lídia M, Pires, Elisabete, Bronze, Maria Rosário, Gut, Jiri, Rosenthal, Philip J, Prudêncio, Miguel, Moreira, Rui, O’Neill, Paul M, Lopes, Francisca
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
Get full text
Journal Article
Torins are potent antimalarials that block replenishment of Plasmodium liver stage parasitophorous vacuole membrane proteins
Hanson, Kirsten K., Ressurreição, Ana S., Buchholz, Kathrin, Prudêncio, Miguel, Herman-Ornelas, Jonathan D., Rebelo, Maria, Beatty, Wandy L., Wirth, Dyann F., Hänscheid, Thomas, Moreira, Rui, Marti, Matthias, Mota, Maria M.
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
Get full text
Journal Article
Visualisation and quantitative analysis of the rodent malaria liver stage by real time imaging
Ploemen, Ivo H J, Prudêncio, Miguel, Douradinha, Bruno G, Ramesar, Jai, Fonager, Jannik, van Gemert, Geert-Jan, Luty, Adrian J F, Hermsen, Cornelus C, Sauerwein, Robert W, Baptista, Fernanda G, Mota, Maria M, Waters, Andrew P, Que, Ivo, Lowik, Clemens W G M, Khan, Shahid M, Janse, Chris J, Franke-Fayard, Blandine M D
Published in PloS one (18.11.2009)
Published in PloS one (18.11.2009)
Get full text
Journal Article