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Published in British journal of pharmacology (01.04.2009)
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Published in British journal of pharmacology (01.04.2009)
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Discovery and structure-activity relationships of a series of pyroglutamic acid amide antagonists of the P2X7 receptor
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Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Synthesis and biological activity of a series of tetrasubstituted-imidazoles as P2X(7) antagonists
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Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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AICA riboside both activates AMP‐activated protein kinase and competes with adenosine for the nucleoside transporter in the CA1 region of the rat hippocampus
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Published in Journal of neurochemistry (01.03.2004)
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Identification of 2-oxo-N-(phenylmethyl)-4-imidazolidinecarboxamide antagonists of the P2X(7) receptor
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Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Identification of 2-oxo-N-(phenylmethyl)-4-imidazolidinecarboxamide antagonists of the P2X7 receptor
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Structure-activity relationships and in vivo activity of (1H-pyrazol-4-yl)acetamide antagonists of the P2X(7) receptor
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Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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A novel series of benzimidazole NR2B-selective NMDA receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
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Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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The discovery of 6 -[2 -(5 -chloro -2 -{[ (2,4 -difluorophenyl )-methyl ]oxy}phenyl ) -1 -cyclopenten -1 -yl ] -2 -pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin EP1 receptor antagonist for the treatment of inflammatory pain
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Published in Bioorganic & medicinal chemistry letters (15.01.2007)
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Mechanism of action of species‐selective P2X7 receptor antagonists
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Published in British journal of pharmacology (01.04.2009)
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Structure-activity relationships of 1,5-biaryl pyrroles as EP1 receptor antagonists
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Structure–activity relationships and in vivo activity of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
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Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Identification of novel glycine sulfonamide antagonists for the EP1 receptor
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Published in Bioorganic & medicinal chemistry letters (15.03.2007)
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