N‑Methyldihydroquinazolinone Derivatives of Retro‑2 with Enhanced Efficacy against Shiga Toxin
Noel, Romain, Gupta, Neetu, Pons, Valérie, Goudet, Amélie, Garcia-Castillo, Maria Daniela, Michau, Aurélien, Martinez, Jennifer, Buisson, David-Alexandre, Johannes, Ludger, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe
Published in Journal of medicinal chemistry (25.04.2013)
Published in Journal of medicinal chemistry (25.04.2013)
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Structure–Activity Relationship Studies of Retro‑1 Analogues against Shiga Toxin
Abdelkafi, Hajer, Michau, Aurélien, Pons, Valérie, Ngadjeua, Flora, Clerget, Alexandra, Ait Ouarab, Lilia, Buisson, David-Alexandre, Montoir, David, Caramelle, Lucie, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Metabolic Stress Impairs Pericyte Response to Optogenetic Stimulation in Pancreatic Islets
Michau, Aurélien, Lafont, Chrystel, Bargi-Souza, Paula, Kemkem, Yasmine, Guillou, Anne, Ravier, Magalie A., Bertrand, Gyslaine, Varrault, Annie, Fiordelisio, Tatiana, Hodson, David J., Mollard, Patrice, Schaeffer, Marie
Published in Frontiers in endocrinology (Lausanne) (23.06.2022)
Published in Frontiers in endocrinology (Lausanne) (23.06.2022)
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Journal Article
Detection of extracellular glucose by GLUT2 contributes to hypothalamic control of food intake
Stolarczyk, Emilie, Guissard, Christophe, Michau, Aurélien, Even, Patrick C, Grosfeld, Alexandra, Serradas, Patricia, Lorsignol, Anne, Pénicaud, Luc, Brot-Laroche, Edith, Leturque, Armelle, Le Gall, Maude
Published in American journal of physiology: endocrinology and metabolism (01.05.2010)
Published in American journal of physiology: endocrinology and metabolism (01.05.2010)
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Journal Article
(S)‑N‑Methyldihydroquinazolinones are the Active Enantiomers of Retro‑2 Derived Compounds against Toxins
Gupta, Neetu, Pons, Valérie, Noël, Romain, Buisson, David-Alexandre, Michau, Aurélien, Johannes, Ludger, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe
Published in ACS medicinal chemistry letters (09.01.2014)
Published in ACS medicinal chemistry letters (09.01.2014)
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Metabolism Regulates Exposure of Pancreatic Islets to Circulating Molecules In Vivo
Michau, Aurélien, Hodson, David J, Fontanaud, Pierre, Guillou, Anne, Espinosa-Carrasco, Gabriel, Molino, François, Peters, Catherine J, Robinson, Iain C, Le Tissier, Paul, Mollard, Patrice, Schaeffer, Marie
Published in Canadian journal of diabetes (01.02.2016)
Published in Canadian journal of diabetes (01.02.2016)
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Journal Article
Inhibitors of retrograde trafficking active against ricin and Shiga toxins also protect cells from several viruses, Leishmania and Chlamydiales
Gupta, Neetu, Noël, Romain, Goudet, Amélie, Hinsinger, Karen, Michau, Aurélien, Pons, Valérie, Abdelkafi, Hajer, Secher, Thomas, Shima, Ayaka, Shtanko, Olena, Sakurai, Yasuteru, Cojean, Sandrine, Pomel, Sébastien, Liévin-Le Moal, Vanessa, Leignel, Véronique, Herweg, Jo-Ana, Fischer, Annette, Johannes, Ludger, Harrison, Kate, Beard, Philippa M., Clayette, Pascal, Le Grand, Roger, Rayner, Jonathan O., Rudel, Thomas, Vacus, Joël, Loiseau, Philippe M., Davey, Robert A., Oswald, Eric, Cintrat, Jean-Christophe, Barbier, Julien, Gillet, Daniel
Published in Chemico-biological interactions (01.04.2017)
Published in Chemico-biological interactions (01.04.2017)
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Journal Article
Mutations in SLC2A2 Gene Reveal hGLUT2 Function in Pancreatic β Cell Development
Michau, Aurélien, Guillemain, Ghislaine, Grosfeld, Alexandra, Vuillaumier-Barrot, Sandrine, Grand, Teddy, Keck, Mathilde, L'Hoste, Sébastien, Chateau, Danielle, Serradas, Patricia, Teulon, Jacques, De Lonlay, Pascale, Scharfmann, Raphaël, Brot-Laroche, Edith, Leturque, Armelle, Le Gall, Maude
Published in The Journal of biological chemistry (25.10.2013)
Published in The Journal of biological chemistry (25.10.2013)
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Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro-1 as Potent Inhibitors of Shiga Toxin
Abdelkafi, Hajer, Michau, Aurélien, Clerget, Alexandra, Buisson, David-Alexandre, Johannes, Ludger, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe
Published in ChemMedChem (01.07.2015)
Published in ChemMedChem (01.07.2015)
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Journal Article
Metabolic Stress Impairs Pericyte Response to Optogenetic Stimulation in Pancreatic Islets
Michau, Aurélien, Lafont, Chrystel, Bargi-Souza, Paula, Kemkem, Yasmine, Guillou, Anne, Ravier, Magalie, Bertrand, Gyslaine, Varrault, Annie, Fiordelisio, Tatiana, Hodson, David, Mollard, Patrice, Schaeffer, Marie
Published in Frontiers in endocrinology (Lausanne) (23.06.2022)
Published in Frontiers in endocrinology (Lausanne) (23.06.2022)
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Journal Article
Metabolism Regulates Exposure of Pancreatic Islets to Circulating Molecules In Vivo
Michau, Aurélien, Hodson, David, Fontanaud, Pierre, Guillou, Anne, Espinosa-Carrasco, Gabriel, Molino, François, Peters, Catherine, Robinson, Iain, Le Tissier, Paul, Mollard, Patrice, Schaeffer, Marie
Published in Diabetes (New York, N.Y.) (01.02.2016)
Published in Diabetes (New York, N.Y.) (01.02.2016)
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Journal Article
Retro-2, a small molecule able to protect cells against a broad spectrum of menacing agents: Toxins, viruses, parasites and intracellular bacteria
Tepshi, Livia, Gupta, Neetu, Noel, Romain, Goudet, Amélie, Hinsinger, Karen, Michau, Aurélien, Pons, Valérie, Abdelkafi, Hajer, Secher, Thomas, Shima, Ayaka, Shtanko, Olena, Sakurai, Yasuteru, Cojean, Sandrine, Pomel, Sébastien, Lievin-Le Moal, Vanessa, Leignel, Véronique, Herweg, Jo-Ana, Fischer, Annette, Johannes, Ludger, Harrison, Kate, Beard, Philippa M., Rudel, Thomas, Vacus, Joël, Loiseau, Philippe M., Davey, Robert A., Oswald, Eric, Cintrat, Jean-Christophe, Barbier, Julien, Gillet, Daniel
Published in Toxicon (Oxford) (01.07.2018)
Published in Toxicon (Oxford) (01.07.2018)
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Journal Article
Inhibitors of retrograde trafficking active against ricin and Shiga toxins also protect cells from several viruses, Chlamydiales and Leishmania
Gupta, Neetu, Noël, Romain, Goudet, Amélie, Hinsinger, Karen, Michau, Aurélien, Pons, Valérie, Abdelkafi, Hajer, Secher, Thomas, Shima, Ayaka, Shtanko, Olena, Sakurai, Yasuteru, Cojean, Sandrine, Pomel, Sébastien, Liévin-Le Moal, Vanessa, Leignel, Véronique, Herweg, Jo-Ana, Fischer, Annette, Johannes, Ludger, Harrison, Kate, Beard, Philippa, Clayette, Pascal, Le Grand, Roger, Rayner, Jonathan, Rudel, Thomas, Vacus, Joël, Loiseau, Philippe, Davey, Robert, Oswald, Eric, Cintrat, Jean-Christophe, Barbier, Julien, Gillet, Daniel
Published in Chemico-biological interactions (01.04.2017)
Published in Chemico-biological interactions (01.04.2017)
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Journal Article
Inside Cover: Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro-1 as Potent Inhibitors of Shiga Toxin (ChemMedChem 7/2015)
Abdelkafi, Hajer, Michau, Aurélien, Clerget, Alexandra, Buisson, David-Alexandre, Johannes, Ludger, Gillet, Daniel, Barbier, Julien, Cintrat, Jean-Christophe
Published in ChemMedChem (01.07.2015)
Published in ChemMedChem (01.07.2015)
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Journal Article
Detection of extracellular glucose by GLUT2 contributes to hypothalamic control of food intake
STOLARCZYK, Emilie, GUISSARD, Christophe, LE GALL, Maude, MICHAU, Aurélien, EVEN, Patrick C, GROSFELD, Alexandra, SERRADAS, Patricia, LORSIGNOL, Anne, PENICAUD, Luc, BROT-LAROCHE, Edith, LETURQUE, Armelle
Published in American journal of physiology: endocrinology and metabolism (2010)
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Published in American journal of physiology: endocrinology and metabolism (2010)
Journal Article
Retro-1 Analogues Differentially Affect Oligonucleotide Delivery and Toxin Trafficking
Yang, Bing, Ming, Xin, Abdelkafi, Hajer, Pons, Valerie, Michau, Aurelien, Gillet, Daniel, Cintrat, Jean-Christophe, Barbier, Julien, Juliano, Rudy
Published in ChemMedChem (21.11.2016)
Published in ChemMedChem (21.11.2016)
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