The catalytic domain of free or ligand bound histone deacetylase 4 occurs in solution predominantly in closed conformation
Schweipert, Markus, Nehls, Thomas, Frühauf, Anton, Debarnot, Cecilé, Kumar, Adarsh, Knapp, Stefan, Lermyte, Frederik, Meyer‐Almes, Franz‐Josef
Published in Protein science (01.03.2024)
Published in Protein science (01.03.2024)
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Journal Article
Design and synthesis of peptides as stabilizers of histone deacetylase 4
Lill, Annika, Schweipert, Markus, Nehls, Thomas, Wurster, Eva, Lermyte, Frederik, Meyer‐Almes, Franz‐Josef, Schmitz, Katja
Published in Journal of peptide science (01.09.2024)
Published in Journal of peptide science (01.09.2024)
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Journal Article
Switching the Switch: Ligand Induced Disulfide Formation in HDAC8
Jänsch, Niklas, Sugiarto, Wisely Oki, Muth, Marius, Kopranovic, Aleksandra, Desczyk, Charlotte, Ballweg, Matthias, Kirschhöfer, Frank, Brenner‐Weiss, Gerald, Meyer‐Almes, Franz‐Josef
Published in Chemistry : a European journal (15.10.2020)
Published in Chemistry : a European journal (15.10.2020)
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Journal Article
Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine‐2,5‐dione Hybrids as Potential Antitumor Agents
Tilekar, Kalpana, Upadhyay, Neha, Meyer‐Almes, Franz‐Josef, Loiodice, Fulvio, Anisimova, Natalia Y., Spirina, Tatiana S., Sokolova, Darina V., Smirnova, Galina B., Choe, Jun‐yong, Pokrovsky, Vadim S., Lavecchia, Antonio, S Ramaa, C
Published in ChemMedChem (05.10.2020)
Published in ChemMedChem (05.10.2020)
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Journal Article
Assessment of Tractable Cysteines for Covalent Targeting by Screening Covalent Fragments
Petri, László, Ábrányi‐Balogh, Péter, Tímea, Imre, Pálfy, Gyula, Perczel, András, Knez, Damijan, Hrast, Martina, Gobec, Martina, Sosič, Izidor, Nyíri, Kinga, Vértessy, Beáta G., Jänsch, Niklas, Desczyk, Charlotte, Meyer‐Almes, Franz‐Josef, Ogris, Iza, Golič Grdadolnik, Simona, Iacovino, Luca Giacinto, Binda, Claudia, Gobec, Stanislav, Keserű, György M.
Published in Chembiochem : a European journal of chemical biology (15.02.2021)
Published in Chembiochem : a European journal of chemical biology (15.02.2021)
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Journal Article
Potent and Selective Non-hydroxamate Histone Deacetylase 8 Inhibitors
Kleinschek, Alexander, Meyners, Christian, Digiorgio, Eros, Brancolini, Claudio, Meyer-Almes, Franz-Josef
Published in ChemMedChem (06.12.2016)
Published in ChemMedChem (06.12.2016)
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Journal Article
Significance of Five-Membered Heterocycles in Human Histone Deacetylase Inhibitors
Frühauf, Anton, Behringer, Martin, Meyer-Almes, Franz-Josef
Published in Molecules (Basel, Switzerland) (27.07.2023)
Published in Molecules (Basel, Switzerland) (27.07.2023)
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Journal Article
A Fluorescence‐Lifetime‐Based Binding Assay for Class IIa Histone Deacetylases
Meyners, Christian, Mertens, Monique, Wessig, Pablo, Meyer‐Almes, Franz‐Josef
Published in Chemistry : a European journal (02.03.2017)
Published in Chemistry : a European journal (02.03.2017)
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Journal Article
Design, Synthesis, and Biological Evaluation of Novel Quinazolin-4(3H)-One-Based Histone Deacetylase 6 (HDAC6) Inhibitors for Anticancer Activity
Khetmalis, Yogesh Mahadu, Fathima, Ashna, Schweipert, Markus, Debarnot, Cécile, Bandaru, Naga Venkata Madhusudhan Rao, Murugesan, Sankaranarayanan, Jamma, Trinath, Meyer-Almes, Franz-Josef, Sekhar, Kondapalli Venkata Gowri Chandra
Published in International journal of molecular sciences (03.07.2023)
Published in International journal of molecular sciences (03.07.2023)
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Journal Article
3‐Chloro‐5‐Substituted‐1,2,4‐Thiadiazoles (TDZs) as Selective and Efficient Protein Thiol Modifiers
Jänsch, Niklas, Frühauf, Anton, Schweipert, Markus, Debarnot, Cécile, Erhardt, Miriam, Brenner‐Weiss, Gerald, Kirschhöfer, Frank, Jasionis, Tomas, Čapkauskaitė, Edita, Zubrienė, Asta, Matulis, Daumantas, Meyer‐Almes, Franz‐Josef
Published in Chembiochem : a European journal of chemical biology (04.11.2022)
Published in Chembiochem : a European journal of chemical biology (04.11.2022)
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Journal Article
The enzyme activity of histone deacetylase 8 is modulated by a redox-switch
Jänsch, Niklas, Meyners, Christian, Muth, Marius, Kopranovic, Aleksandra, Witt, Olaf, Oehme, Ina, Meyer-Almes, Franz-Josef
Published in Redox biology (01.01.2019)
Published in Redox biology (01.01.2019)
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Journal Article
Impact of binding mechanism on selective inhibition of histone deacetylase isoforms
Meyners, Christian, Meyer‐Almes, Franz‐Josef
Published in Chemical biology & drug design (01.12.2017)
Published in Chemical biology & drug design (01.12.2017)
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Journal Article
Class IIa HDACs repressive activities on MEF2-depedent transcription are associated with poor prognosis of ER⁺ breast tumors
Clocchiatti, Andrea, Di Giorgio, Eros, Ingrao, Sabrina, Meyer-Almes, Franz-Josef, Tripodo, Claudio, Brancolini, Claudio
Published in The FASEB journal (01.03.2013)
Published in The FASEB journal (01.03.2013)
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Journal Article
Defining the Mechanism of Action and Enzymatic Selectivity of Psammaplin A against Its Epigenetic Targets
Baud, Matthias G. J, Leiser, Thomas, Haus, Patricia, Samlal, Sharon, Wong, Ai Ching, Wood, Robert J, Petrucci, Vanessa, Gunaratnam, Mekala, Hughes, Siobhan M, Buluwela, Lakjaya, Turlais, Fabrice, Neidle, Stephen, Meyer-Almes, Franz-Josef, White, Andrew J. P, Fuchter, Matthew J
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
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Journal Article
Synthesis and HDAC inhibitory activity of pyrimidine-based hydroxamic acids
Jakubkiene, Virginija, Valiulis, Gabrielius Ernis, Schweipert, Markus, Zubriene, Asta, Matulis, Daumantas, Meyer-Almes, Franz-Josef, Tumkevicius, Sigitas
Published in Beilstein journal of organic chemistry (13.07.2022)
Published in Beilstein journal of organic chemistry (13.07.2022)
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Journal Article
Diaryl Pyrazoline, 1,3,4-Oxadizole, and 1,2,4-Triazole Pharmacophore Hybridization: Design, Synthesis, HDAC Inhibition, and Caspase 3/7 Activation Studies
Alzahrani, Abdullah Yahya Abdullah, Gupta, Pratibha, Patil, Vijay, Meyer-Almes, Franz-Josef, Sokolova, D. V., Pokrovsky, V. S., Ramaa, C. S.
Published in Russian journal of bioorganic chemistry (01.04.2024)
Published in Russian journal of bioorganic chemistry (01.04.2024)
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