In vitro and in vivo characterization of a neutral boron-containing thrombin inhibitor
TAPPARELLI, C, METTERNICH, R, EHRHARDT, C, ZURINI, M, CLAESON, G, SCULLY, M. F, STONE, S. R
Published in The Journal of biological chemistry (05.03.1993)
Published in The Journal of biological chemistry (05.03.1993)
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Drug discovery process for kinase inhibitors
Weinmann, Hilmar, Metternich, Rainer
Published in Chembiochem : a European journal of chemical biology (01.03.2005)
Published in Chembiochem : a European journal of chemical biology (01.03.2005)
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Platelet aggregation and fibrinogen binding in human, rhesus monkey, guinea-pig, hamster and rat blood: activation by ADP and a thrombin receptor peptide and inhibition by glycoprotein IIb/IIIa antagonists
Cook, N S, Zerwes, H G, Tapparelli, C, Powling, M, Singh, J, Metternich, R, Hagenbach, A
Published in Thrombosis and haemostasis (01.09.1993)
Published in Thrombosis and haemostasis (01.09.1993)
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Benzyloxycarbonyl-D-Phe-Pro-methoxypropylboroglycine : a novel inhibitor of thrombin with high selectivity containing a neutral side chain at the P1 position
CLAESON, G, PHILIPP, M, AGNER, E, SCULLY, M. F, METTERNICH, R, KAKKAR, V. V, DESOYZA, T, LING-HAO NIU
Published in Biochemical journal (01.03.1993)
Published in Biochemical journal (01.03.1993)
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Toward a Total Synthesis of the Immunosuppressant Sanglifehrin A. Preparation of Two Relay Compounds by Degradation and Their Use in the Reassembly of the Natural Product
Metternich, Rainer, Denni, Donatienne, Thai, Binh, Sedrani, Richard
Published in Journal of organic chemistry (24.12.1999)
Published in Journal of organic chemistry (24.12.1999)
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A synthesis of the C1N12 tripeptide fragment of sanglifehrin A
Bänteli, Rolf, Brun, Ivan, Hall, Philip, Metternich, Rainer
Published in Tetrahedron letters (12.03.1999)
Published in Tetrahedron letters (12.03.1999)
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Design, synthesis and biological evaluation of selective boron-containing thrombin inhibitors
WIENAND, A, EHRHARDT, C, METTERNICH, R, TAPPARELLI, C
Published in Bioorganic & medicinal chemistry (01.07.1999)
Published in Bioorganic & medicinal chemistry (01.07.1999)
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Diastereoselective aldol reactions using .beta.-keto imide derived enolates. A versatile approach to the assemblage of polypropionate systems
Evans, David A, Clark, J. Stephen, Metternich, Rainer, Novack, Vance J, Sheppard, George S
Published in Journal of the American Chemical Society (01.01.1990)
Published in Journal of the American Chemical Society (01.01.1990)
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Thrombin inhibition in an ex vivo model of porcine heart xenograft hyperacute rejection
Robson, S C, Young, V K, Cook, N S, Metternich, R, Kasper-Konig, W, Lesnikoski, B A, Pierson, 3rd, R N, Hancock, W W, Candinas, D, White, D J, Bach, F H
Published in Transplantation (27.03.1996)
Published in Transplantation (27.03.1996)
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Structure and function of thrombin receptors
Tapparelli, Carlo, Metternich, Rainer, Cook, Nigel S.
Published in Trends in pharmacological sciences (Regular ed.) (01.12.1993)
Published in Trends in pharmacological sciences (Regular ed.) (01.12.1993)
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Thrombin Inhibition in discordant xenograft rejection
Lesnikoski, Beth-Ann, Candinas, Daniel, Otsu, Ichiro, Metternich, Rainer, Bach, Fritz H., Robson, Simon C.
Published in Xenotransplantation (Københaven) (01.08.1997)
Published in Xenotransplantation (Københaven) (01.08.1997)
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