Reply to Achieng and Riedel
Pham, Hanh Thi, Goring, Mark E, Mesplède, Thibault
Published in The Journal of infectious diseases (01.01.2019)
Published in The Journal of infectious diseases (01.01.2019)
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Journal Article
Erratum for Mesplède et al., "The R263K Dolutegravir Resistance-Associated Substitution Progressively Decreases HIV-1 Integration"
Mesplède, Thibault, Leng, Jing, Pham, Hanh Thi, Liang, Jiaming, Quan, Yudong, Han, Yingshan, Wainberg, Mark A
Published in mBio (25.09.2018)
Published in mBio (25.09.2018)
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Journal Article
Pharmaceutical, clinical, and resistance information on doravirine, a novel non-nucleoside reverse transcriptase inhibitor for the treatment of HIV-1 infection
Pham, Hanh Thi, Xiao, Meng A, Principe, Miguel Av, Wong, Alexander, Mesplède, Thibault
Published in Drugs in Context (03.03.2020)
Published in Drugs in Context (03.03.2020)
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Journal Article
Identification of a dibenzocyclooctadiene lignan as a HIV-1 non-nucleoside reverse transcriptase inhibitor
Han, Ying-Shan, Xiao, Wei-Lie, Xu, Hongtao, Kramer, Victor G, Quan, Yudong, Mesplède, Thibault, Oliveira, Maureen, Colby-Germinario, Susan P, Sun, Han-Dong, Wainberg, Mark A
Published in Antiviral chemistry & chemotherapy (01.02.2015)
Published in Antiviral chemistry & chemotherapy (01.02.2015)
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Journal Article
HIV‐1 group O integrase displays lower susceptibility to raltegravir and has a different mutational pathway for resistance than HIV‐1 group M
Depatureaux, Agnès, Mesplède, Thibault, Quashie, Peter, Oliveira, Maureen, Moisi, Daniela, Brenner, Bluma, Wainberg, Mark
Published in Journal of the International AIDS Society (01.11.2014)
Published in Journal of the International AIDS Society (01.11.2014)
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Journal Article
Antimalarial drugs and their metabolites are potent Zika virus inhibitors
Han, Yingshan, Pham, Hanh T., Xu, Hongtao, Quan, Yudong, Mesplède, Thibault
Published in Journal of medical virology (01.07.2019)
Published in Journal of medical virology (01.07.2019)
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Journal Article
The antimalarial drug amodiaquine possesses anti‐ZIKA virus activities
Han, Yingshan, Mesplède, Thibault, Xu, Hongtao, Quan, Yudong, Wainberg, Mark A.
Published in Journal of medical virology (01.05.2018)
Published in Journal of medical virology (01.05.2018)
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Journal Article
Cenicriviroc blocks HIV entry but does not lead to redistribution of HIV into extracellular space like maraviroc
Kramer, Victor, Hassounah, Said, Colby‐Germinario, Susan, Mesplède, Thibault, Lefebvre, Eric, Wainberg, Mark
Published in Journal of the International AIDS Society (01.11.2014)
Published in Journal of the International AIDS Society (01.11.2014)
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Journal Article
Characterization of the R263K Mutation in HIV-1 Integrase That Confers Low-Level Resistance to the Second-Generation Integrase Strand Transfer Inhibitor Dolutegravir
QUASHIE, Peter K, MESPLEDE, Thibault, HAN, Ying-Shan, OLIVEIRA, Maureen, SINGHROY, Diane N, FUJIWARA, Tamio, UNDERWOOD, Mark R, WAINBERG, Mark A
Published in Journal of Virology (01.03.2012)
Published in Journal of Virology (01.03.2012)
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Journal Article
Polymorphic substitution E157Q in HIV-1 integrase increases R263K-mediated dolutegravir resistance and decreases DNA binding activity
Anstett, Kaitlin, Cutillas, Vincent, Fusco, Robert, Mesplède, Thibault, Wainberg, Mark A
Published in Journal of antimicrobial chemotherapy (01.08.2016)
Published in Journal of antimicrobial chemotherapy (01.08.2016)
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Journal Article
Investigational drugs for HIV: trends, opportunities and key players
Overmars, Ronald J, Krullaars, Zoë, Mesplède, Thibault
Published in Expert opinion on investigational drugs (01.02.2023)
Published in Expert opinion on investigational drugs (01.02.2023)
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Journal Article
Selection of the R263K and H51Y resistance substitutions for DTG causes diminished integration and explains the lack of clinically significant drug resistance to this compound
Mesplède, Thibault, Liang, Jiaming, Anstett, Katlin, Osman, Nathan, Thi Pham, Hanh, Wainberg, Mark A.
Published in Journal of Virus Eradication (01.05.2016)
Published in Journal of Virus Eradication (01.05.2016)
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Journal Article
The G118R plus R263K Combination of Integrase Mutations Associated with Dolutegravir-Based Treatment Failure Reduces HIV-1 Replicative Capacity and Integration
Xiao, Meng A, Cleyle, Jenna, Yoo, Sunbin, Forrest, Mekayla, Krullaars, Zoë, Pham, Hanh Thi, Mesplède, Thibault
Published in Antimicrobial agents and chemotherapy (17.05.2023)
Published in Antimicrobial agents and chemotherapy (17.05.2023)
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Journal Article
Selective resistance profiles emerging in patient-derived clinical isolates with cabotegravir, bictegravir, dolutegravir, and elvitegravir
Oliveira, Maureen, Ibanescu, Ruxandra-Ilinca, Anstett, Kaitlin, Mésplède, Thibault, Routy, Jean-Pierre, Robbins, Marjorie A, Brenner, Bluma G
Published in Retrovirology (17.08.2018)
Published in Retrovirology (17.08.2018)
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Journal Article