Genome-wide and high-density CRISPR-Cas9 screens identify point mutations in PARP1 causing PARP inhibitor resistance
Pettitt, Stephen J, Krastev, Dragomir B, Brandsma, Inger, Dréan, Amy, Song, Feifei, Aleksandrov, Radoslav, Harrell, Maria I, Menon, Malini, Brough, Rachel, Campbell, James, Frankum, Jessica, Ranes, Michael, Pemberton, Helen N, Rafiq, Rumana, Fenwick, Kerry, Swain, Amanda, Guettler, Sebastian, Lee, Jung-Min, Swisher, Elizabeth M, Stoynov, Stoyno, Yusa, Kosuke, Ashworth, Alan, Lord, Christopher J
Published in Nature communications (10.05.2018)
Published in Nature communications (10.05.2018)
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Journal Article
Modeling Therapy Resistance in BRCA1/2 -Mutant Cancers
Dréan, Amy, Williamson, Chris T, Brough, Rachel, Brandsma, Inger, Menon, Malini, Konde, Asha, Garcia-Murillas, Isaac, Pemberton, Helen N, Frankum, Jessica, Rafiq, Rumana, Badham, Nicholas, Campbell, James, Gulati, Aditi, Turner, Nicholas C, Pettitt, Stephen J, Ashworth, Alan, Lord, Christopher J
Published in Molecular cancer therapeutics (01.09.2017)
Published in Molecular cancer therapeutics (01.09.2017)
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Journal Article
ATR Is a Therapeutic Target in Synovial Sarcoma
Jones, Samuel E, Fleuren, Emmy D G, Frankum, Jessica, Konde, Asha, Williamson, Chris T, Krastev, Dragomir B, Pemberton, Helen N, Campbell, James, Gulati, Aditi, Elliott, Richard, Menon, Malini, Selfe, Joanna L, Brough, Rachel, Pettitt, Stephen J, Niedzwiedz, Wojciech, van der Graaf, Winette T A, Shipley, Janet, Ashworth, Alan, Lord, Christopher J
Published in Cancer research (Chicago, Ill.) (15.12.2017)
Published in Cancer research (Chicago, Ill.) (15.12.2017)
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Journal Article
A novel tankyrase inhibitor, MSC2504877, enhances the effects of clinical CDK4/6 inhibitors
Menon, Malini, Elliott, Richard, Bowers, Leandra, Balan, Nicolae, Rafiq, Rumana, Costa-Cabral, Sara, Munkonge, Felix, Trinidade, Ines, Porter, Roderick, Campbell, Andrew D, Johnson, Emma R, Esdar, Christina, Buchstaller, Hans-Peter, Leuthner, Birgitta, Rohdich, Felix, Schneider, Richard, Sansom, Owen, Wienke, Dirk, Ashworth, Alan, Lord, Christopher J
Published in Scientific reports (17.01.2019)
Published in Scientific reports (17.01.2019)
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Journal Article
Small Molecule Inhibitors of the Neuropilin-1 Vascular Endothelial Growth Factor A (VEGF-A) Interaction
Jarvis, Ashley, Allerston, Charles K, Jia, Haiyan, Herzog, Birger, Garza-Garcia, Acely, Winfield, Natalie, Ellard, Katie, Aqil, Rehan, Lynch, Rosemary, Chapman, Chris, Hartzoulakis, Basil, Nally, James, Stewart, Mark, Cheng, Lili, Menon, Malini, Tickner, Michelle, Djordjevic, Snezana, Driscoll, Paul C, Zachary, Ian, Selwood, David L
Published in Journal of medicinal chemistry (11.03.2010)
Published in Journal of medicinal chemistry (11.03.2010)
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Journal Article
Myristoyl-CoA:Protein N-Myristoyltransferase, an Essential Enzyme and Potential Drug Target in Kinetoplastid Parasites
Price, Helen P, Menon, Malini R, Panethymitaki, Chrysoula, Goulding, David, McKean, Paul G, Smith, Deborah F
Published in The Journal of biological chemistry (28.02.2003)
Published in The Journal of biological chemistry (28.02.2003)
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Journal Article
The grafting of universal T-helper epitopes enhances immunogenicity of HIV-1 Tat concurrently improving its safety profile
Kashi, Venkatesh P, Jacob, Rajesh A, Shamanna, Raghavendra A, Menon, Malini, Balasiddaiah, Anangi, Varghese, Rebu K, Bachu, Mahesh, Ranga, Udaykumar
Published in PloS one (22.12.2014)
Published in PloS one (22.12.2014)
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Journal Article
Hammerhead ribozyme-mediated silencing of the mutant fibrillin-1 of tight skin mouse: Insight into the functional role of mutant fibrillin-1
Menon, Rajesh P., Menon, Malini R., Shi-Wen, Xu, Renzoni, Elisabetta, Bou-Gharios, George, Black, Carol M., Abraham, David J.
Published in Experimental cell research (15.05.2006)
Published in Experimental cell research (15.05.2006)
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Journal Article
Hi-JAK-ing the ubiquitin system: The design and physicochemical optimisation of JAK PROTACs
Shah, Rishi R., Redmond, Joanna M., Mihut, Andrei, Menon, Malini, Evans, John P., Murphy, John A., Bartholomew, Michelle A., Coe, Diane M.
Published in Bioorganic & medicinal chemistry (01.03.2020)
Published in Bioorganic & medicinal chemistry (01.03.2020)
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Journal Article
Astrocytes mediate HIV‐1 Tat‐induced neuronal damage via ligand‐gated ion channel P2X7R
Tewari, Manju, Monika, , Varghese, Rebu K, Menon, Malini, Seth, Pankaj
Published in Journal of neurochemistry (01.02.2015)
Published in Journal of neurochemistry (01.02.2015)
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Journal Article
RET mutation status in medullary thyroid cancer(MTC) patients and the significance of genetic screening for mutations in their immediate relatives--a preliminary report
Menon, Malini M, Simha, Mangala R
Published in Indian journal of pathology & microbiology (01.04.2005)
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Published in Indian journal of pathology & microbiology (01.04.2005)
Journal Article
E-Cadherin/ROS1 Inhibitor Synthetic Lethality in Breast Cancer
Bajrami, Ilirjana, Marlow, Rebecca, van de Ven, Marieke, Brough, Rachel, Pemberton, Helen N, Frankum, Jessica, Song, Feifei, Rafiq, Rumana, Konde, Asha, Krastev, Dragomir B, Menon, Malini, Campbell, James, Gulati, Aditi, Kumar, Rahul, Pettitt, Stephen J, Gurden, Mark D, Cardenosa, Marta Llorca, Chong, Irene, Gazinska, Patrycja, Wallberg, Fredrik, Sawyer, Elinor J, Martin, Lesley-Ann, Dowsett, Mitch, Linardopoulos, Spiros, Natrajan, Rachael, Ryan, Colm J, Derksen, Patrick W B, Jonkers, Jos, Tutt, Andrew N J, Ashworth, Alan, Lord, Christopher J
Published in Cancer discovery (01.04.2018)
Published in Cancer discovery (01.04.2018)
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Journal Article
PTAP motif duplication in the p6 Gag protein confers a replication advantage on HIV-1 subtype C
Sharma, Shilpee, Arunachalam, Prabhu S., Menon, Malini, Ragupathy, Viswanath, Satya, Ravi Vijaya, Jebaraj, Joshua, Aralaguppe, Shambhu Ganeshappa, Rao, Chaitra, Pal, Sreshtha, Saravanan, Shanmugam, Murugavel, Kailapuri G., Balakrishnan, Pachamuthu, Solomon, Suniti, Hewlett, Indira, Ranga, Udaykumar
Published in The Journal of biological chemistry (27.07.2018)
Published in The Journal of biological chemistry (27.07.2018)
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Journal Article
Abstract 2975: Synthetic lethality in synovial sarcoma: SS18-SSX fusions and DNA damage response (DDR) inhibitors
Fleuren, Emmy DG, Jones, Sam, Frankum, Jessica, Williamson, Chris, Menon, Malini, Shipley, Janet, Ashworth, Alan, Graaf, Winette van der, Lord, Christopher J.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract NTOC-093: SYNTHETIC LETHAL APPROACHES TO TARGET ARID1A DEFICIENT OVARIAN CANCERS
Khalique, Saira, Williamson, Chris T., Pemberton, Helen, Wai, Patty T., Menon, Malini, Brough, Rachel, Leonidou, Andri, Peck, Barrie, Banerjee, Susana, Natrajan, Rachael C., Lord, Christopher J.
Published in Clinical cancer research (01.06.2017)
Published in Clinical cancer research (01.06.2017)
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Journal Article
Chemosensitivity profiling of osteosarcoma tumour cell lines identifies a model of BRCAness
Holme, Harriett, Gulati, Aditi, Brough, Rachel, Fleuren, Emmy D G, Bajrami, Ilirjana, Campbell, James, Chong, Irene Y, Costa-Cabral, Sara, Elliott, Richard, Fenton, Tim, Frankum, Jessica, Jones, Samuel E, Menon, Malini, Miller, Rowan, Pemberton, Helen N, Postel-Vinay, Sophie, Rafiq, Rumana, Selfe, Joanna L, von Kriegsheim, Alex, Munoz, Amaya Garcia, Rodriguez, Javier, Shipley, Janet, van der Graaf, Winette T A, Williamson, Chris T, Ryan, Colm J, Pettitt, Stephen, Ashworth, Alan, Strauss, Sandra J, Lord, Christopher J
Published in Scientific reports (13.07.2018)
Published in Scientific reports (13.07.2018)
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Journal Article
Abstract 2986: E-cadherin/ROS1 inhibitor synthetic lethality in breast cancer
Bajrami, Ilirjana, Marlow, Rebecca, Ven, Marieke van de, Brough, Rachel, Pemberton, Helen N., Frankum, Jessica, Song, Fei Fei, Rafiq, Rumana, Konde, Asha, Menon, Malini, Campbell, James, Gulati, Aditi, Kumar, Rahul, Pettitt, Stephen J., Gurden, Mark D., Cardenosa, Marta Llorca, Chong, Irene, Gazinska, Patrycja, Wallberg, Fredrik, Sawyer, Elinor J., Martin, Lesley-Ann, Dowsett, Mitch, Linardopoulos, Spiros, Ryan, Colm, Derksen, Patrick W., Jonkers, Jos, Tutt, Andrew N.J., Ashworth, Alan, Lord, Christopher J.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Candidate drug therapies for molecularly defined subgroups of esophageal cancer identified from high-throughput drug screening
Chong, Irene Yu-Shing, Cunningham, David, Elliott, Richard, Konde, Asha, Campbell, James, Menon, Malini, Bowers, Leandra, Daley, Frances, Lord, Christopher J., Ashworth, Alan
Published in Journal of clinical oncology (20.05.2014)
Published in Journal of clinical oncology (20.05.2014)
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Journal Article
Author Correction: Chemosensitivity profiling of osteosarcoma tumour cell lines identifies a model of BRCAness
Holme, Harriett, Gulati, Aditi, Brough, Rachel, Fleuren, Emmy D G, Bajrami, Ilirjana, Campbell, James, Chong, Irene Y, Costa-Cabral, Sara, Elliott, Richard, Fenton, Tim, Frankum, Jessica, Jones, Samuel E, Menon, Malini, Miller, Rowan, Pemberton, Helen N, Postel-Vinay, Sophie, Rafiq, Rumana, Selfe, Joanna L, von Kriegsheim, Alex, Munoz, Amaya Garcia, Rodriguez, Javier, Shipley, Janet, van der Graaf, Winette T A, Williamson, Chris T, Ryan, Colm J, Pettitt, Stephen, Ashworth, Alan, Strauss, Sandra J, Lord, Christopher J
Published in Scientific reports (21.08.2018)
Published in Scientific reports (21.08.2018)
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Journal Article