ALARM NMR: A Rapid and Robust Experimental Method To Detect Reactive False Positives in Biochemical Screens
Huth, Jeffrey R, Mendoza, Renaldo, Olejniczak, Edward T, Johnson, Robert W, Cothron, Darlene A, Liu, Yaya, Lerner, Claude G, Chen, Jun, Hajduk, Philip J
Published in Journal of the American Chemical Society (12.01.2005)
Published in Journal of the American Chemical Society (12.01.2005)
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Journal Article
Discovery of a potent and selective Bcl-2 inhibitor using SAR by NMR
Petros, Andrew M., Huth, Jeffrey R., Oost, Thorsten, Park, Cheol-Min, Ding, Hong, Wang, Xilu, Zhang, Haichao, Nimmer, Paul, Mendoza, Renaldo, Sun, Chaohong, Mack, Jamey, Walter, Karl, Dorwin, Sarah, Gramling, Emily, Ladror, Uri, Rosenberg, Saul H., Elmore, Steven W., Fesik, Stephen W., Hajduk, Philip J.
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Journal Article
Toxicological Evaluation of Thiol-Reactive Compounds Identified Using a La Assay To Detect Reactive Molecules by Nuclear Magnetic Resonance
Huth, Jeffrey R, Song, Danying, Mendoza, Renaldo R, Black-Schaefer, Candice L, Mack, Jamey C, Dorwin, Sarah A, Ladror, Uri S, Severin, Jean M, Walter, Karl A, Bartley, Diane M, Hajduk, Philip J
Published in Chemical research in toxicology (01.12.2007)
Published in Chemical research in toxicology (01.12.2007)
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Journal Article
Novel p-Arylthio Cinnamides as Antagonists of Leukocyte Function-Associated Antigen-1/Intracellular Adhesion Molecule-1 Interaction. 2. Mechanism of Inhibition and Structure-Based Improvement of Pharmaceutical Properties
Liu, Gang, Huth, Jeffrey R, Olejniczak, Edward T, Mendoza, Renaldo, DeVries, Peter, Leitza, Sandra, Reilly, Edward B, Okasinski, Gregory F, Fesik, Stephen W, von Geldern, Thomas W
Published in Journal of medicinal chemistry (12.04.2001)
Published in Journal of medicinal chemistry (12.04.2001)
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Journal Article
Non-peptide entry inhibitors of HIV-1 that target the gp41 coiled coil pocket
Stewart, Kent D., Huth, Jeffrey R., Ng, Teresa I., McDaniel, Keith, Hutchinson, Rebecca Newlin, Stoll, Vincent S., Mendoza, Renaldo R., Matayoshi, Edmund D., Carrick, Robert, Mo, HongMei, Severin, Jean, Walter, Karl, Richardson, Paul L., Barrett, Leo W., Meadows, Robert, Anderson, Steve, Kohlbrenner, William, Maring, Clarence, Kempf, Dale J., Molla, Akhter, Olejniczak, Edward T.
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
NMR and Mutagenesis Evidence for an I Domain Allosteric Site That Regulates Lymphocyte Function-Associated Antigen 1 Ligand Binding
Huth, Jeffrey R., Olejniczak, Edward T., Mendoza, Renaldo, Liang, Heng, Edith A. S. Harris, Lupher, Mark L., Wilson, Amy E., Fesik, Stephen W., Staunton, Donald E.
Published in Proceedings of the National Academy of Sciences - PNAS (09.05.2000)
Published in Proceedings of the National Academy of Sciences - PNAS (09.05.2000)
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Journal Article
Design and characterization of an engineered gp41 protein from human immunodeficiency virus-1 as a tool for drug discovery
Stewart, Kent D, Steffy, Kevin, Harris, Kevin, Harlan, John E, Stoll, Vincent S, Huth, Jeffrey R, Walter, Karl A, Gramling-Evans, Emily, Mendoza, Renaldo R, Severin, Jean M, Richardson, Paul L, Barrett, Leo W, Matayoshi, Edmund D, Swift, Kerry M, Betz, Stephen F, Muchmore, Steve W, Kempf, Dale J, Molla, Akhter
Published in Journal of computer-aided molecular design (01.01.2007)
Published in Journal of computer-aided molecular design (01.01.2007)
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Journal Article
NMR-Based Screening of Proteins Containing 13C-Labeled Methyl Groups
Hajduk, Philip J, Augeri, David J, Mack, Jamey, Mendoza, Renaldo, Yang, Jianguo, Betz, Stephen F, Fesik, Stephen W
Published in Journal of the American Chemical Society (23.08.2000)
Published in Journal of the American Chemical Society (23.08.2000)
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Journal Article
Cracking the molecular weight barrier: Fragment screening of an aminotransferase using an NMR-based functional assay
Mendoza, Renaldo, Petros, Andrew M., Liu, Yaya, Thimmapaya, Rama, Surowy, Carol S., Leise, Walter F., Pereda-Lopez, Ana, Panchal, Sanjay C., Sun, Chaohong
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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Journal Article
Solution structure and calcium‐binding properties of EF‐hands 3 and 4 of calsenilin
Yu, Liping, Sun, Chaohong, Mendoza, Renaldo, Wang, Jie, Matayoshi, Edmund D., Hebert, Eric, Pereda‐Lopez, Ana, Hajduk, Philip J., Olejniczak, Edward T.
Published in Protein science (01.11.2007)
Published in Protein science (01.11.2007)
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Journal Article
NMR-Driven Discovery of Benzoylanthranilic Acid Inhibitors of Far Upstream Element Binding Protein Binding to the Human Oncogene c-myc Promoter
Huth, Jeffrey R, Yu, Liping, Collins, Irene, Mack, Jamey, Mendoza, Renaldo, Isaac, Binumol, Braddock, Demetrios T, Muchmore, Steven W, Comess, Kenneth M, Fesik, Stephen W, Clore, G. Marius, Levens, David, Hajduk, Philip J
Published in Journal of medicinal chemistry (23.09.2004)
Published in Journal of medicinal chemistry (23.09.2004)
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