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Published in British journal of cancer (14.02.2005)
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Bioactivation of 5-(aziridin-1-yl)-2,4-dinitrobenzamide (CB 1954) by human NAD(P)H quinone oxidoreductase 2 : A novel co-substrate-mediated antitumor prodrug therapy
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Published in Cancer research (Chicago, Ill.) (01.08.2000)
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Antibody-Enzyme Conjugates for Cancer Therapy
Melton, Roger G., Sherwood, Roger F.
Published in JNCI : Journal of the National Cancer Institute (21.02.1996)
Published in JNCI : Journal of the National Cancer Institute (21.02.1996)
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A cytotoxic agent can be generated selectively at cancer sites
BAGSHAWE, K. D, SPRINGER, C. J, SEARLE, F, ANTONIW, P, SHARMA, S. K, MELTON, R. G, SHERWOOD, R. F
Published in British journal of cancer (01.12.1988)
Published in British journal of cancer (01.12.1988)
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Bioactivation of dinitrobenzamide mustards by an E. coli B nitroreductase
Anlezark, G.M., Melton, R.G., Sherwood, R.F., Wilson, W.R., Denny, W.A., Palmer, B.D., Knox, R.J., Friedlos, F., Williams, A.
Published in Biochemical pharmacology (25.08.1995)
Published in Biochemical pharmacology (25.08.1995)
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Polyethylene glycol modification of a galactosylated streptavidin clearing agent: effects on immunogenicity and clearance of a biotinylated anti-tumour antibody
Marshall, D, Pedley, R B, Boden, J A, Boden, R, Melton, R G, Begent, R H
Published in British journal of cancer (01.03.1996)
Published in British journal of cancer (01.03.1996)
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Anti-tumour effects of an antibody-carboxypeptidase G2 conjugate in combination with phenol mustard prodrugs
BLAKEY, D. C, DAVIES, D. H, DOWELL, R. I, EAST, S. J, BURKE, P. J, SHARMA, S. K, SPRINGER, C. J, MAUGER, A. B, MELTON, R. G
Published in British journal of cancer (01.11.1995)
Published in British journal of cancer (01.11.1995)
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ZD2767, an improved system for antibody-directed enzyme prodrug therapy that results in tumor regressions in colorectal tumor xenografts
BLAKEY, D. C, BURKE, P. J, PINDER, P. E, SHARMA, S. K, WRIGHT, A. F, SPRINGER, C. J, DAVIES, D. H, DOWELL, R. I, EAST, S. J, ECKERSLEY, K. P, FITTON, J. E, MCDAID, J, MELTON, R. G, NICULESCU-DUVAZ, I. A
Published in Cancer research (Chicago, Ill.) (15.07.1996)
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Published in Cancer research (Chicago, Ill.) (15.07.1996)
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Investigation of alternative prodrugs for use with E. coli nitroreductase in 'suicide gene' approaches to cancer therapy
Bailey, S M, Knox, R J, Hobbs, S M, Jenkins, T C, Mauger, A B, Melton, R G, Burke, P J, Connors, T A, Hart, I R
Published in Gene therapy (01.12.1996)
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Published in Gene therapy (01.12.1996)
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Optimization of small-scale coupling of A5B7 monoclonal antibody to carboxypeptidase G2
MELTON, R. G, BOYLE, J. M. B, ROGERS, G. T, BURKE, P, BAGSHAWE, K. D, SHERWOOD, R. F
Published in Journal of immunological methods (14.01.1993)
Published in Journal of immunological methods (14.01.1993)
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New Mustard Prodrugs for Antibody-Directed Enzyme Prodrug Therapy: Alternatives to the Amide Link
Dowell, Robert I, Springer, Caroline J, Davies, David H, Hadley, Elizabeth M, Burke, Philip J, Boyle, F. Thomas, Melton, Roger G, Connors, Thomas A, Blakey, David C, Mauger, Anthony B
Published in Journal of medicinal chemistry (01.03.1996)
Published in Journal of medicinal chemistry (01.03.1996)
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Disposition of the prodrug 4-( (2-chloroethyl) amino) benzoyl-L-glutamic acid and its active parent drug in mice
ANTONIW, P, SPRINGER, C. J, BAGSHAWE, K. D, SEARLE, F, MELTON, R. G, ROGERS, G. T, BURKE, P. J, SHERWOOD, R. F
Published in British journal of cancer (01.12.1990)
Published in British journal of cancer (01.12.1990)
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Effect of cyclosporine on immunogenicity of a bacterial enzyme carboxypeptidase G2 in ADEPT
Sharma, S K, Bagshawe, K D, Melton, R G, Begent, R H
Published in Transplantation proceedings (01.12.1996)
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Published in Transplantation proceedings (01.12.1996)
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Galactosylated antibodies and antibody‐enzyme conjugates in antibody‐directed enzyme prodrug therapy
Sharma, Surinder K., Bagshawe, Kenneth D., Burke, Philip J., Boden, Joan A., Rogers, Gordon T., Springer, Caroline J., Melton, Roger G., Sherwood, Roger F.
Published in Cancer (01.02.1994)
Published in Cancer (01.02.1994)
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Antibody directed enzyme prodrug therapy (ADEPT): clinical report
Bagshawe, K D, Sharma, S K, Springer, C J, Antoniw, P, Boden, J A, Rogers, G T, Burke, P J, Melton, R G, Sherwood, R F
Published in Disease markers (01.05.1991)
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Published in Disease markers (01.05.1991)
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Virtual cofactors for an Escherichia coli nitroreductase enzyme: Relevance to reductively activated prodrugs in antibody directed enzyme prodrug therapy (ADEPT)
Knox, Richard J., Friedlos, Frank, Jarman, Michael, Davies, Lawrence C., Goddard, Phyllis, Anlezark, Gillian M., Melton, Roger G., Sherwood, Roger F.
Published in Biochemical pharmacology (26.05.1995)
Published in Biochemical pharmacology (26.05.1995)
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Antibody-directed enzyme prodrug therapy (ADEPT) for treatment of major solid tumour disease
Blakey, D C, Burke, P J, Davies, D H, Dowell, R I, Melton, R G, Springer, C J, Wright, A F
Published in Biochemical Society transactions (01.11.1995)
Published in Biochemical Society transactions (01.11.1995)
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