Design, Synthesis, and SAR of New Pyrrole-Oxindole Progesterone Receptor Modulators Leading to 5-(7-Fluoro-3,3-dimethyl-2-oxo-2,3-dihydro-1H-indol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile (WAY-255348)
Fensome, Andrew, Adams, William R, Adams, Andrea L, Berrodin, Tom J, Cohen, Jeff, Huselton, Christine, Illenberger, Arthur, Kern, Jeffrey C, Hudak, Valerie A, Marella, Michael A, Melenski, Edward G, McComas, Casey C, Mugford, Cheryl A, Slayden, Ov D, Yudt, Matthew, Zhang, Zhiming, Zhang, Puwen, Zhu, Yuan, Winneker, Richard C, Wrobel, Jay E
Published in Journal of medicinal chemistry (27.03.2008)
Published in Journal of medicinal chemistry (27.03.2008)
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Effects of a Novel Beta Lactam Compound, MC-100093, on the Expression of Glutamate Transporters/Receptors and Ethanol Drinking Behavior of Alcohol-Preferring Rats
Alhaddad, Hasan, Wong, Woonyen, Abou-Gharbia, Magid, Childers, Wayne, Melenski, Edward, Bell, Richard L, Sari, Youssef
Published in The Journal of pharmacology and experimental therapeutics (01.12.2022)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2022)
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Facile synthesis of the glucosylceramide synthase inhibitor GZ667161
Hewlett, Elizabeth D., Melenski, Edward, Qiu, Frederick V., Leung, Hiu T., Jacobson, Marlene, Qiu, Feng, Abou-Gharbia, Magid, Childers, Wayne
Published in Tetrahedron letters (01.10.2020)
Published in Tetrahedron letters (01.10.2020)
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Novel compounds that reverse the disease phenotype in Type 2 Gaucher disease patient-derived cells
Childers, Wayne, Fan, Rong, Martinez, Rogelio, Colussi, Dennis J., Melenski, Edward, Liu, Yuxiao, Gordon, John, Abou-Gharbia, Magid, Jacobson, Marlene A.
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
Published in Bioorganic & medicinal chemistry letters (15.01.2020)
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Novel progesterone receptor modulators: 4-Aryl-phenylsulfonamides
McComas, Casey, Cohen, Jeffrey, Huselton, Christine, Marella, Michael, Melenski, Edward, Mugford, Cheryl, Slayden, Ov, Winneker, Richard, Wrobel, Jay, Yudt, Matthew R., Fensome, Andrew
Published in Bioorganic & medicinal chemistry letters (01.12.2012)
Published in Bioorganic & medicinal chemistry letters (01.12.2012)
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Journal Article
Design, Synthesis, and SAR of New Pyrrole-Oxindole Progesterone Receptor Modulators Leading to 5-(7-Fluoro-3,3-dimethyl-2-oxo-2,3-dihydro-1 H -indol-5-yl)-1-methyl-1 H -pyrrole-2-carbonitrile (WAY-255348)
Fensome, Andrew, Adams, William R., Adams, Andrea L., Berrodin, Tom J., Cohen, Jeff, Huselton, Christine, Illenberger, Arthur, Kern, Jeffrey C., Hudak, Valerie A., Marella, Michael A., Melenski, Edward G., McComas, Casey C., Mugford, Cheryl A., Slayden, Ov D., Yudt, Matthew, Zhang, Zhiming, Zhang, Puwen, Zhu, Yuan, Winneker, Richard C., Wrobel, Jay E.
Published in Journal of medicinal chemistry (01.03.2008)
Published in Journal of medicinal chemistry (01.03.2008)
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Journal Article
Functionalized N,N-dialkylamino phenyl ethers and their method of use
Jacobson, Marlene A, Abou-Gharbia, Magid A, Childers, Wayne E, Melenski, Edward G
Year of Publication 10.05.2022
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Year of Publication 10.05.2022
Patent
Novel Functionalized N,N-Dialkylamino Phenyl Ethers and Their Method of Use
Jacobson, Marlene A, Abou-Gharbia, Magid A, Childers, Wayne E, Melenski, Edward G
Year of Publication 12.11.2020
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Year of Publication 12.11.2020
Patent
NOVEL FUNCTIONALIZED N,N-DIALKYLAMINO PHENYL ETHERS AND THEIR METHOD OF USE
ABOU-GHARBIA, Magid A, MELENSKI, Edward G, CHILDERS, Wayne E, JACOBSON, Marlene A
Year of Publication 31.05.2019
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Year of Publication 31.05.2019
Patent