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Das, Soumen, Yau, Mei‐Kwan, Noble, Jeffery, De Pascalis, Lucrezia, Finn, M. G.
Published in Angewandte Chemie International Edition (10.01.2022)
Published in Angewandte Chemie International Edition (10.01.2022)
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Programmable multistage drug delivery to lymph nodes
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Published in Nature nanotechnology (01.06.2020)
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Diet-induced obesity, adipose inflammation, and metabolic dysfunction correlating with PAR2 expression are attenuated by PAR2 antagonism
Lim, Junxian, Iyer, Abishek, Liu, Ligong, Suen, Jacky Y, Lohman, Rink-Jan, Seow, Vernon, Yau, Mei-Kwan, Brown, Lindsay, Fairlie, David P
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Published in The FASEB journal (01.12.2013)
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Mechanotransduction activates RhoA in the neighbors of apoptotic epithelial cells to engage apical extrusion
Duszyc, Kinga, Gomez, Guillermo A., Lagendijk, Anne K., Yau, Mei-Kwan, Nanavati, Bageshri Naimish, Gliddon, Briony L., Hall, Thomas E., Verma, Suzie, Hogan, Benjamin M., Pitson, Stuart M., Fairlie, David P., Parton, Robert G., Yap, Alpha S.
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Published in Current biology (22.03.2021)
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Published in Nature communications (24.08.2017)
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Toward Drugs for Protease-Activated Receptor 2 (PAR2)
Yau, Mei-Kwan, Liu, Ligong, Fairlie, David P
Published in Journal of medicinal chemistry (10.10.2013)
Published in Journal of medicinal chemistry (10.10.2013)
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A Potent Antagonist of Protease-Activated Receptor 2 That Inhibits Multiple Signaling Functions in Human Cancer Cells
Jiang, Yuhong, Yau, Mei-Kwan, Lim, Junxian, Wu, Kai-Chen, Xu, Weijun, Suen, Jacky Y, Fairlie, David P
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The Influence of Substitution on Thiol-Induced Oxanorbornadiene Fragmentation
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Published in Organic letters (07.05.2021)
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Protease activated receptor 2 (PAR2) modulators: a patent review (2010-2015)
Yau, Mei-Kwan, Lim, Junxian, Liu, Ligong, Fairlie, David P
Published in Expert opinion on therapeutic patents (02.04.2016)
Published in Expert opinion on therapeutic patents (02.04.2016)
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Potent Thiophene Antagonists of Human Complement C3a Receptor with Anti-Inflammatory Activity
Rowley, Jessica A, Reid, Robert C, Poon, Eunice K. Y, Wu, Kai-Chen, Lim, Junxian, Lohman, Rink-Jan, Hamidon, Johan K, Yau, Mei-Kwan, Halili, Maria A, Durek, Thomas, Iyer, Abishek, Fairlie, David P
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Published in Journal of medicinal chemistry (23.01.2020)
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Receptor residence time trumps drug-likeness and oral bioavailability in determining efficacy of complement C5a antagonists
Seow, Vernon, Lim, Junxian, Cotterell, Adam J, Yau, Mei-Kwan, Xu, Weijun, Lohman, Rink-Jan, Kok, W Mei, Stoermer, Martin J, Sweet, Matthew J, Reid, Robert C, Suen, Jacky Y, Fairlie, David P
Published in Scientific reports (20.04.2016)
Published in Scientific reports (20.04.2016)
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Publisher Correction: Programmable multistage drug delivery to lymph nodes
Schudel Alex, Chapman Asheley Poole, Mei-Kwan, Yau, Higginson, Cody James, Francis, David Mark, Manspeaker, Margaret Patricia, Avecilla Alexa Regina Chua, Rohner, Nathan Andrew, Finn, M G, Napier, Thomas Susan
Published in Nature nanotechnology (01.08.2020)
Published in Nature nanotechnology (01.08.2020)
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Transport of Molecular Cargo by Interaction with Virus‐Like Particle RNA
Das, Soumen, Yau, Mei‐Kwan, Noble, Jeffery, De Pascalis, Lucrezia, Finn, M. G.
Published in Angewandte Chemie (10.01.2022)
Published in Angewandte Chemie (10.01.2022)
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Potent Heterocyclic Ligands for Human Complement C3a Receptor
Reid, Robert C, Yau, Mei-Kwan, Singh, Ranee, Hamidon, Johan K, Lim, Junxian, Stoermer, Martin J, Fairlie, David P
Published in Journal of medicinal chemistry (23.10.2014)
Published in Journal of medicinal chemistry (23.10.2014)
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Three Homology Models of PAR2 Derived from Different Templates: Application to Antagonist Discovery
Perry, Samuel R, Xu, Weijun, Wirija, Anna, Lim, Junxian, Yau, Mei-Kwan, Stoermer, Martin J, Lucke, Andrew J, Fairlie, David P
Published in Journal of chemical information and modeling (22.06.2015)
Published in Journal of chemical information and modeling (22.06.2015)
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Repurposing Registered Drugs as Antagonists for Protease-Activated Receptor 2
Xu, Weijun, Lim, Junxian, Goh, Chai-Yeen, Suen, Jacky Y, Jiang, Yuhong, Yau, Mei-Kwan, Wu, Kai-Chen, Liu, Ligong, Fairlie, David P
Published in Journal of chemical information and modeling (26.10.2015)
Published in Journal of chemical information and modeling (26.10.2015)
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Downsizing a human inflammatory protein to a small molecule with equal potency and functionality
Reid, Robert C, Yau, Mei-Kwan, Singh, Ranee, Hamidon, Johan K, Reed, Anthony N, Chu, Peifei, Suen, Jacky Y, Stoermer, Martin J, Blakeney, Jade S, Lim, Junxian, Faber, Jonathan M, Fairlie, David P
Published in Nature communications (2013)
Published in Nature communications (2013)
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Efficient chemical synthesis of human complement protein C3a
Ghassemian, Artin, Wang, Ching-I Anderson, Yau, Mei-Kwan, Reid, Robert C, Lewis, Richard J, Fairlie, David P, Alewood, Paul F, Durek, Thomas
Published in Chemical communications (Cambridge, England) (21.03.2013)
Published in Chemical communications (Cambridge, England) (21.03.2013)
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Potent complement C3a receptor agonists derived from oxazole amino acids: Structure–activity relationships
Singh, Ranee, Reed, Anthony N., Chu, Peifei, Scully, Conor C.G., Yau, Mei-Kwan, Suen, Jacky Y., Durek, Thomas, Reid, Robert C., Fairlie, David P.
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
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