Discovery of a Potent and Selective Covalent p300/CBP Inhibitor
Mastracchio, Anthony, Lai, Chunqiu, Digiammarino, Enrico, Ready, Damien B, Lasko, Loren M, Bromberg, Kenneth D, McClellan, William J, Montgomery, Debra, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Patterson, Melanie J, Sun, Chaohong C, Rosenberg, Saul, Lai, Albert, Michaelides, Michael R
Published in ACS medicinal chemistry letters (13.05.2021)
Published in ACS medicinal chemistry letters (13.05.2021)
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Journal Article
Discovery of potent and selective thienopyrimidine inhibitors of Aurora kinases
McClellan, William J., Dai, Yujia, Abad-Zapatero, Cele, Albert, Daniel H., Bouska, Jennifer J., Glaser, Keith B., Magoc, Terry J., Marcotte, Patrick A., Osterling, Donald J., Stewart, Kent D., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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Journal Article
Reduction of nanoparticle exposure to welding aerosols by modification of the ventilation system in a workplace
Lee, Myong-Hwa, McClellan, William J., Candela, Joe, Andrews, Dan, Biswas, Pratim
Published in Journal of nanoparticle research : an interdisciplinary forum for nanoscale science and technology (01.01.2007)
Published in Journal of nanoparticle research : an interdisciplinary forum for nanoscale science and technology (01.01.2007)
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Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors
Wang, Le, Pratt, John K, Soltwedel, Todd, Sheppard, George S, Fidanze, Steven D, Liu, Dachun, Hasvold, Lisa A, Mantei, Robert A, Holms, James H, McClellan, William J, Wendt, Michael D, Wada, Carol, Frey, Robin, Hansen, T. Matthew, Hubbard, Robert, Park, Chang H, Li, Leiming, Magoc, Terrance J, Albert, Daniel H, Lin, Xiaoyu, Warder, Scott E, Kovar, Peter, Huang, Xiaoli, Wilcox, Denise, Wang, Rongqi, Rajaraman, Ganesh, Petros, Andrew M, Hutchins, Charles W, Panchal, Sanjay C, Sun, Chaohong, Elmore, Steven W, Shen, Yu, Kati, Warren M, McDaniel, Keith F
Published in Journal of medicinal chemistry (11.05.2017)
Published in Journal of medicinal chemistry (11.05.2017)
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Discovery and Structure−Activity Relationship of Antagonists of B-Cell Lymphoma 2 Family Proteins with Chemopotentiation Activity in Vitro and in Vivo
Wendt, Michael D, Shen, Wang, Kunzer, Aaron, McClellan, William J, Bruncko, Milan, Oost, Thorsten K, Ding, Hong, Joseph, Mary K, Zhang, Haichao, Nimmer, Paul M, Ng, Shi-Chung, Shoemaker, Alexander R, Petros, Andrew M, Oleksijew, Anatol, Marsh, Kennan, Bauch, Joy, Oltersdorf, Tilman, Belli, Barbara A, Martineau, Darlene, Fesik, Stephen W, Rosenberg, Saul H, Elmore, Steven W
Published in Journal of medicinal chemistry (09.02.2006)
Published in Journal of medicinal chemistry (09.02.2006)
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Studies Leading to Potent, Dual Inhibitors of Bcl-2 and Bcl-xL
Bruncko, Milan, Oost, Thorsten K, Belli, Barbara A, Ding, Hong, Joseph, Mary K, Kunzer, Aaron, Martineau, Darlene, McClellan, William J, Mitten, Michael, Ng, Shi-Chung, Nimmer, Paul M, Oltersdorf, Tilman, Park, Cheol-Min, Petros, Andrew M, Shoemaker, Alexander R, Song, Xiaohong, Wang, Xilu, Wendt, Michael D, Zhang, Haichao, Fesik, Stephen W, Rosenberg, Saul H, Elmore, Steven W
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Journal Article
Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties
Bruncko, Milan, McClellan, William J., Wendt, Michael D., Sauer, Daryl R., Geyer, Andrew, Dalton, Christopher R., Kaminski, Michele A., Weitzberg, Moshe, Gong, Jane, Dellaria, Joseph F., Mantei, Robert, Zhao, Xumiao, Nienaber, Vicki L., Stewart, Kent, Klinghofer, Vered, Bouska, Jennifer, Rockway, Todd W., Giranda, Vincent L.
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
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Sulfonamide derivatives as Bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 18.01.2017
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Year of Publication 18.01.2017
Patent
Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 07.12.2016
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Year of Publication 07.12.2016
Patent
BROMODOMAIN INHIBITORS
HOLMS JAMES H, MANTEI ROBERT A, FIDANZE STEVEN D, HASVOLD LISA, WANG LE, DAI YUJIA, SHEPPARD GEORGE S, LIU DACHUN, KATI WARREN M, MCDANIEL KEITH F, MCCLELLAN WILLIAM J, WADA CAROL K, PRATT JOHN K
Year of Publication 24.09.2014
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Year of Publication 24.09.2014
Patent
APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, HANSEN TODD M, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, KUNZER AARON, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA
Year of Publication 09.04.2013
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Year of Publication 09.04.2013
Patent
SULFONAMIDE DERIVATIVES AS BCL-2-SELECTIVE APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, HANSEN TODD M, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, KUNZER AARON, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA
Year of Publication 12.12.2012
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Year of Publication 12.12.2012
Patent
SULFONAMIDE DERIVATIVES AS BCL-2-SELECTIVE APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 20.09.2011
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Year of Publication 20.09.2011
Patent
APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 05.09.2011
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Year of Publication 05.09.2011
Patent
Interaction with the S1β-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors
Wendt, Michael D., Geyer, Andrew, McClellan, William J., Rockway, Todd W., Weitzberg, Moshe, Zhao, Xumiao, Mantei, Robert, Stewart, Kent, Nienaber, Vicki, Klinghofer, Vered, Giranda, Vincent L.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Conformationally defined adrenergic agents. 1. Design and synthesis of novel .alpha.2-selective adrenergic agents: electrostatic repulsion based conformational prototypes
DeBernardis, John F, Kerkman, Daniel J, Winn, Martin, Bush, Eugene N, Arendsen, David L, McClellan, William J, Kyncl, John J, Basha, Fatima Z
Published in Journal of medicinal chemistry (01.10.1985)
Published in Journal of medicinal chemistry (01.10.1985)
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Interaction with the S1β-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors
WENDT, Michael D, GEYER, Andrew, GIRANDA, Vincent L, MCCLELLAN, William J, ROCKWAY, Todd W, WEITZBERG, Moshe, XUMIAO ZHAO, MANTEI, Robert, STEWART, Kent, NIENABER, Vicki, KLINGHOFER, Vered
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Journal Article
BROMODOMAIN INHIBITORS
Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
Patent